Results
|
1.
|
|
|
2.
|
|
|
3.
|
|
|
4.
|
Modeling aided design of potent glycogen phosphorylase inhibitors. [electronic resource] by
- Deng, Qiaolin
- Lu, Zhijian
- Bohn, Joann
- Ellsworth, Kenneth P
- Myers, Robert W
- Geissler, Wayne M
- Harris, Georgianna
- Willoughby, Christopher A
- Chapman, Kevin
- McKeever, Brian
- Mosley, Ralph
Producer: 20050728
In:
Journal of molecular graphics & modelling vol. 23
Availability: No items available.
|
|
5.
|
Novel 3,4-dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase a. [electronic resource] by
- Rosauer, Keith G
- Ogawa, Anthony K
- Willoughby, Chris A
- Ellsworth, Kenneth P
- Geissler, Wayne M
- Myers, Robert W
- Deng, Qiaolin
- Chapman, Kevin T
- Harris, Georgianna
- Moller, David E
Producer: 20040806
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
|
|
6.
|
A new class of glycogen phosphorylase inhibitors. [electronic resource] by
- Lu, Zhijian
- Bohn, Joann
- Bergeron, Raynald
- Deng, Qiaolin
- Ellsworth, Kenneth P
- Geissler, Wayne M
- Harris, Georgianna
- McCann, Peggy E
- McKeever, Brian
- Myers, Robert W
- Saperstein, Richard
- Willoughby, Christopher A
- Yao, Jun
- Chapman, Kevin
Producer: 20040706
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
|
|
7.
|
Design and synthesis of novel proline based factor XIa selective inhibitors as leads for potential new anticoagulants. [electronic resource] by
- Hussain, Zahid
- Cooke, Andrew J
- Neelamkavil, Santhosh
- Brown, Lindsay
- Carswell, Emma
- Geissler, Wayne M
- Guo, Zhuyan
- Hawes, Brian
- Kelly, Terri M
- Kiyoi, Yasuko
- Lai, KehDih
- Lesburg, Charles
- Pow, Eleanor
- Zang, Yi
- Wood, Harold B
- Edmondson, Scott D
- Liu, Weiguo
Producer: 20210528
In:
Bioorganic & medicinal chemistry letters vol. 30
Availability: No items available.
|
|
8.
|
Peptidomic profiling of human cerebrospinal fluid identifies YPRPIHPA as a novel substrate for prolylcarboxypeptidase. [electronic resource] by
- Zhao, Xuemei
- Southwick, Katie
- Cardasis, Helene L
- Du, Yi
- Lassman, Michael E
- Xie, Dan
- El-Sherbeini, Mohamed
- Geissler, Wayne M
- Pryor, KellyAnn D
- Verras, Andreas
- Garcia-Calvo, Margarita
- Shen, Dong-Ming
- Yates, Nathan A
- Pinto, Shirly
- Hendrickon, Ronald C
Producer: 20101123
In:
Proteomics vol. 10
Availability: No items available.
|
|
9.
|
Expression, purification and crystallization of human prolylcarboxypeptidase. [electronic resource] by
- Abeywickrema, Pravien D
- Patel, Sangita B
- Byrne, Noel J
- Diehl, Ronald E
- Hall, Dawn L
- Ford, Rachael E
- Rickert, Keith W
- Reid, John C
- Shipman, Jennifer M
- Geissler, Wayne M
- Pryor, Kelly D
- SinhaRoy, Ranabir
- Soisson, Stephen M
- Lumb, Kevin J
- Sharma, Sujata
Producer: 20101104
In:
Acta crystallographica. Section F, Structural biology and crystallization communications vol. 66
Availability: No items available.
|
|
10.
|
Design and synthesis of prolylcarboxypeptidase (PrCP) inhibitors to validate PrCP as a potential target for obesity. [electronic resource] by
- Zhou, Changyou
- Garcia-Calvo, Margareta
- Pinto, Shirly
- Lombardo, Matthew
- Feng, Zhe
- Bender, Kate
- Pryor, Kellyann D
- Bhatt, Urmi R
- Chabin, Renee M
- Geissler, Wayne M
- Shen, Zhu
- Tong, Xinchun
- Zhang, Zhoupeng
- Wong, Kenny K
- Roy, Ranabir Sinha
- Chapman, Kevin T
- Yang, Lihu
- Xiong, Yusheng
Producer: 20101109
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
|
|
11.
|
Definitive Metabolite Identification Coupled with Automated Ligand Identification System (ALIS) Technology: A Novel Approach to Uncover Structure-Activity Relationships and Guide Drug Design in a Factor IXa Inhibitor Program. [electronic resource] by
- Zhang, Ting
- Liu, Yong
- Yang, Xianshu
- Martin, Gary E
- Yao, Huifang
- Shang, Jackie
- Bugianesi, Randal M
- Ellsworth, Kenneth P
- Sonatore, Lisa M
- Nizner, Peter
- Sherer, Edward C
- Hill, Susan E
- Knemeyer, Ian W
- Geissler, Wayne M
- Dandliker, Peter J
- Helmy, Roy
- Wood, Harold B
Producer: 20160823
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
|
|
12.
|
Discovery and optimization of orally active cyclohexane-based prolylcarboxypeptidase (PrCP) inhibitors. [electronic resource] by
- Debenham, John S
- Graham, Thomas H
- Verras, Andreas
- Zhang, Yong
- Clements, Matthew J
- Kuethe, Jeffrey T
- Madsen-Duggan, Christina
- Liu, Wensheng
- Bhatt, Urmi R
- Chen, Dunlu
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- He, Huaibing
- Li, Xiaohua
- Lisnock, JeanMarie
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xu, Suoyu
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20140817
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
|
|
13.
|
A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes. [electronic resource] by
- Graham, Thomas H
- Liu, Wensheng
- Verras, Andreas
- Reibarkh, Mikhail
- Bleasby, Kelly
- Bhatt, Urmi R
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- Gorski, Judith N
- He, Huaibing
- Lassman, Michael E
- Lisnock, JeanMarie
- Li, Xiaohua
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xie, Dan
- Xu, Suoyu
- Xiao, Jianying
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|
|
14.
|
The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors. [electronic resource] by
- Graham, Thomas H
- Shen, Hong C
- Liu, Wensheng
- Xiong, Yusheng
- Verras, Andreas
- Bleasby, Kelly
- Bhatt, Urmi R
- Chabin, Renee M
- Chen, Dunlu
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- He, Huaibing
- Lassman, Michael E
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Xie, Dan
- Xu, Suoyu
- Colletti, Steven L
- Tata, James R
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120803
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|
|
15.
|
A new class of prolylcarboxypeptidase inhibitors, part 1: discovery and evaluation. [electronic resource] by
- Graham, Thomas H
- Liu, Wensheng
- Verras, Andreas
- Sebhat, Iyassu K
- Xiong, Yusheng
- Bleasby, Kelly
- Bhatt, Urmi R
- Chen, Qing
- Garcia-Calvo, Margarita
- Geissler, Wayne M
- Gorski, Judith N
- He, Huaibing
- Lassman, Michael E
- Lisnock, JeanMarie
- Li, Xiaohua
- Shen, Zhu
- Tong, Xinchun
- Tung, Elaine C
- Wiltsie, Judyann
- Xiao, Jianying
- Xie, Dan
- Xu, Suoyu
- Hale, Jeffrey J
- Pinto, Shirly
- Shen, Dong-Ming
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
|
|
16.
|
Development of a novel class of potent and selective FIXa inhibitors. [electronic resource] by
- Zhang, Ting
- Andre, Patrick
- Bateman, Thomas J
- Chen, Yi-Heng
- Desai, Kunal
- Ellsworth, Kenneth
- Geissler, Wayne M
- Guo, Liangqin
- Hruza, Alan
- Jian, Tianying
- Meng, Dongfang
- Parker, Dann L
- Qian, Xiaoxia
- Reichert, Paul
- Sherer, Edward C
- Shu, Min
- Smith, Cameron J
- Sonatore, Lisa M
- Tschirret-Guth, Richard
- Nolting, Andrew F
- Orr, Robert
- Campeau, Louis-Charles
- Araki, Kazuto
- Nishimura, Teruyuki
- Sakurada, Isao
- Wood, Harold B
Producer: 20160620
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
|
|
17.
|
Development of a novel tricyclic class of potent and selective FIXa inhibitors. [electronic resource] by
- Meng, Dongfang
- Andre, Patrick
- Bateman, Thomas J
- Berger, Richard
- Chen, Yi-Heng
- Desai, Kunal
- Dewnani, Sunita
- Ellsworth, Kenneth
- Feng, Daming
- Geissler, Wayne M
- Guo, Liangqin
- Hruza, Alan
- Jian, Tianying
- Li, Hong
- Metzger, Joe
- Parker, Dann L
- Reichert, Paul
- Sherer, Edward C
- Smith, Cameron J
- Sonatore, Lisa M
- Tschirret-Guth, Richard
- Wu, Jane
- Xu, Jiayi
- Zhang, Ting
- Campeau, Louis-Charles
- Orr, Robert
- Poirier, Marc
- McCabe-Dunn, Jamie
- Araki, Kazuto
- Nishimura, Teruyuki
- Sakurada, Isao
- Hirabayashi, Tomokazu
- Wood, Harold B
Producer: 20161216
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
|