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Discovery of Pyridazinone and Pyrazolo[1,5- [electronic resource] by
- O'Malley, Daniel P
- Ahuja, Vijay
- Fink, Brian
- Cao, Carolyn
- Wang, Cindy
- Swanson, Jesse
- Wee, Susan
- Gavai, Ashvinikumar V
- Tokarski, John
- Critton, David
- Paiva, Anthony A
- Johnson, Benjamin M
- Szapiel, Nicolas
- Xie, Dianlin
Publication details: ACS medicinal chemistry letters Oct 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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5.
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Discovery of novel 1-arylmethyl pyrrolidin-2-yl ethanol amines as calcium-sensing receptor antagonists. [electronic resource] by
- Gavai, Ashvinikumar V
- Vaz, Roy J
- Mikkilineni, Amarendra B
- Roberge, Jacques Y
- Liu, Yalei
- Lawrence, R Michael
- Corte, James R
- Yang, Wu
- Bednarz, Mark
- Dickson, John K
- Ma, Zhengping
- Seethala, Ramakrishna
- Feyen, Jean H M
Producer: 20060627
In:
Bioorganic & medicinal chemistry letters vol. 15
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Preclinical antitumor activity of BMS-599626, a pan-HER kinase inhibitor that inhibits HER1/HER2 homodimer and heterodimer signaling. [electronic resource] by
- Wong, Tai W
- Lee, Francis Y
- Yu, Chiang
- Luo, Feng R
- Oppenheimer, Simone
- Zhang, Hongjian
- Smykla, Richard A
- Mastalerz, Harold
- Fink, Brian E
- Hunt, John T
- Gavai, Ashvinikumar V
- Vite, Gregory D
Producer: 20061114
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 12
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7.
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Novel pyrrolo[2,1-f][1,2,4]triazin-4-amines: Dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Fink, Brian E
- Norris, Derek
- Mastalerz, Harold
- Chen, Ping
- Goyal, Bindu
- Zhao, Yufen
- Kim, Soong-Hoon
- Vite, Gregory D
- Lee, Francis Y
- Zhang, Hongjian
- Oppenheimer, Simone
- Tokarski, John S
- Wong, Tai W
- Gavai, Ashvinikumar V
Producer: 20110425
In:
Bioorganic & medicinal chemistry letters vol. 21
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Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17beta-hydroxysteroid dehydrogenase type 3. [electronic resource] by
- Fink, Brian E
- Gavai, Ashvinikumar V
- Tokarski, John S
- Goyal, Bindu
- Misra, Raj
- Xiao, Hai-Yun
- Kimball, S David
- Han, Wen-Ching
- Norris, Derek
- Spires, Thomas E
- You, Dan
- Gottardis, Marco M
- Lorenzi, Matthew V
- Vite, Gregory D
Producer: 20060417
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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9.
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Novel C-5 aminomethyl pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Mastalerz, Harold
- Chang, Ming
- Gavai, Ashvinikumar
- Johnson, Walter
- Langley, David
- Lee, Francis Y
- Marathe, Punit
- Mathur, Arvind
- Oppenheimer, Simone
- Tarrant, James
- Tokarski, John S
- Vite, Gregory D
- Vyas, Dolatrai M
- Wong, Henry
- Wong, Tai W
- Zhang, Hongjian
- Zhang, Guifen
Producer: 20070730
In:
Bioorganic & medicinal chemistry letters vol. 17
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10.
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Antitumor and antiangiogenic activities of BMS-690514, an inhibitor of human EGF and VEGF receptor kinase families. [electronic resource] by
- Wong, Tai W
- Lee, Francis Y
- Emanuel, Stuart
- Fairchild, Craig
- Fargnoli, Joseph
- Fink, Brian
- Gavai, Ashvinikumar
- Hammell, Amy
- Henley, Benjamin
- Hilt, Christine
- Hunt, John T
- Krishnan, Bala
- Kukral, Daniel
- Lewin, Anne
- Malone, Harold
- Norris, Derek
- Oppenheimer, Simone
- Vite, Gregory
- Yu, Chiang
Producer: 20111017
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 17
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11.
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[2.2.1]-Bicyclic sultams as potent androgen receptor antagonists. [electronic resource] by
- Shan, Weifang
- Balog, Aaron
- Nation, Andrew
- Zhu, Xiao
- Chen, Jing
- Cvijic, Mary Ellen
- Geng, Jieping
- Rizzo, Cheryl A
- Spires, Thomas
- Attar, Ricardo M
- Obermeier, Mary
- Traeger, Sarah
- Dai, Jun
- Zhang, Yingru
- Galella, Michael
- Trainor, George
- Vite, Gregory D
- Gavai, Ashvinikumar V
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
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12.
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Design and synthesis of a G-protein-coupled receptor antagonist library of aryloxyalkanolamines using a polymer-supported acyclic acetal linker. [electronic resource] by
- Roberge, Jacques Y
- Harikrishnan, Lalgudi S
- Kamau, Muthoni G
- Ruan, Zheming
- Van Kirk, Katy
- Liu, Yalei
- Cooper, Christopher B
- Poss, Michael A
- Dickson, John K
- Gavai, Ashvinikumar V
- Chao, Sam T
- Leith, Leslie W
- Bednarz, Mark S
- Mathur, Arvind
- Kakarla, Ramesh
- Schnur, Dora M
- Vaz, Roy
- Lawrence, R Michael
Producer: 20090227
In:
Journal of combinatorial chemistry vol. 11
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13.
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5-((4-Aminopiperidin-1-yl)methyl)pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Mastalerz, Harold
- Chang, Ming
- Chen, Ping
- Fink, Brian E
- Gavai, Ashvinikumar
- Han, Wen-Ching
- Johnson, Walter
- Langley, David
- Lee, Francis Y
- Leavitt, Kenneth
- Marathe, Punit
- Norris, Derek
- Oppenheimer, Simone
- Sleczka, Bogdan
- Tarrant, James
- Tokarski, John S
- Vite, Gregory D
- Vyas, Dolatrai M
- Wong, Henry
- Wong, Tai W
- Zhang, Hongjian
- Zhang, Guifen
Producer: 20071120
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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14.
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New C-5 substituted pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Mastalerz, Harold
- Chang, Ming
- Chen, Ping
- Dextraze, Pierre
- Fink, Brian E
- Gavai, Ashvinikumar
- Goyal, Bindu
- Han, Wen-Ching
- Johnson, Walter
- Langley, David
- Lee, Francis Y
- Marathe, Punit
- Mathur, Arvind
- Oppenheimer, Simone
- Ruediger, Edward
- Tarrant, James
- Tokarski, John S
- Vite, Gregory D
- Vyas, Dolatrai M
- Wong, Henry
- Wong, Tai W
- Zhang, Hongjian
- Zhang, Guifen
Producer: 20070725
In:
Bioorganic & medicinal chemistry letters vol. 17
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15.
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Design and synthesis of 4-[3,5-dioxo-11-oxa-4,9-diazatricyclo[5.3.1.0(2,6)]undec-4-yl]-2-trifluoromethyl-benzonitriles as androgen receptor antagonists. [electronic resource] by
- Xiao, Hai-Yun
- Balog, Aaron
- Attar, Ricardo M
- Fairfax, David
- Fleming, Linda B
- Holst, Christian L
- Martin, Gregory S
- Rossiter, Lana M
- Chen, Jing
- Cvjic, Mary-Ellen
- Dell-John, Janet
- Geng, Jieping
- Gottardis, Marco M
- Han, Wen-Ching
- Nation, Andrew
- Obermeier, Mary
- Rizzo, Cheryl A
- Schweizer, Liang
- Spires, Thomas
- Shan, Weifang
- Gavai, Ashvinikumar
- Salvati, Mark E
- Vite, Gregory
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
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16.
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Discovery and preclinical evaluation of [4-[[1-(3-fluorophenyl)methyl]-1H-indazol-5-ylamino]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamic acid, (3S)-3-morpholinylmethyl ester (BMS-599626), a selective and orally efficacious inhibitor of human epidermal growth factor receptor 1 and 2 kinases. [electronic resource] by
- Gavai, Ashvinikumar V
- Fink, Brian E
- Fairfax, David J
- Martin, Gregory S
- Rossiter, Lana M
- Holst, Christian L
- Kim, Soong-Hoon
- Leavitt, Kenneth J
- Mastalerz, Harold
- Han, Wen-Ching
- Norris, Derek
- Goyal, Bindu
- Swaminathan, Shankar
- Patel, Bharat
- Mathur, Arvind
- Vyas, Dolatrai M
- Tokarski, John S
- Yu, Chiang
- Oppenheimer, Simone
- Zhang, Hongjian
- Marathe, Punit
- Fargnoli, Joseph
- Lee, Francis Y
- Wong, Tai W
- Vite, Gregory D
Producer: 20091215
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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17.
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BMS-871: a novel orally active pan-Notch inhibitor as an anticancer agent. [electronic resource] by
- Shan, Weifang
- Balog, Aaron
- Quesnelle, Claude
- Gill, Patrice
- Han, Wen-Ching
- Norris, Derek
- Mandal, Sunilkumar
- Thiruvenkadam, Raja
- Gona, Kiran Babu
- Thiyagarajan, Kamalraj
- Kandula, Sathiah
- McGlinchey, Kelly
- Menard, Krista
- Wen, Mei-Li
- Rose, Anne
- White, Ronald
- Guarino, Victor
- Shen, Ding Ren
- Cvijic, Mary Ellen
- Ranasinghe, Asoka
- Dai, Jun
- Zhang, Yingru
- Wu, Dauh-Rurng
- Mathur, Arvind
- Rampulla, Richard
- Trainor, George
- Hunt, John T
- Vite, Gregory D
- Westhouse, Richard
- Lee, Francis Y
- Gavai, Ashvinikumar V
Producer: 20160219
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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18.
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Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors. [electronic resource] by
- Gavai, Ashvinikumar V
- Quesnelle, Claude
- Norris, Derek
- Han, Wen-Ching
- Gill, Patrice
- Shan, Weifang
- Balog, Aaron
- Chen, Ke
- Tebben, Andrew
- Rampulla, Richard
- Wu, Dauh-Rurng
- Zhang, Yingru
- Mathur, Arvind
- White, Ronald
- Rose, Anne
- Wang, Haiqing
- Yang, Zheng
- Ranasinghe, Asoka
- D'Arienzo, Celia
- Guarino, Victor
- Xiao, Lan
- Su, Ching
- Everlof, Gerry
- Arora, Vinod
- Shen, Ding Ren
- Cvijic, Mary Ellen
- Menard, Krista
- Wen, Mei-Li
- Meredith, Jere
- Trainor, George
- Lombardo, Louis J
- Olson, Richard
- Baran, Phil S
- Hunt, John T
- Vite, Gregory D
- Fischer, Bruce S
- Westhouse, Richard A
- Lee, Francis Y
Producer: 20150525
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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