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4-benzimidazolyl-3-phenylbutanoic acids as novel PIF-pocket-targeting allosteric inhibitors of protein kinase PKCζ. [electronic resource] by
- Fröhner, Wolfgang
- Lopez-Garcia, Laura A
- Neimanis, Sonja
- Weber, Nadja
- Navratil, Jeanette
- Maurer, Frauke
- Stroba, Adriana
- Zhang, Hua
- Biondi, Ricardo M
- Engel, Matthias
Producer: 20111212
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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10.
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2-(3-Oxo-1,3-diphenylpropyl)malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug concept. [electronic resource] by
- Wilhelm, Adriana
- Lopez-Garcia, Laura A
- Busschots, Katrien
- Fröhner, Wolfgang
- Maurer, Frauke
- Boettcher, Stefan
- Zhang, Hua
- Schulze, Jörg O
- Biondi, Ricardo M
- Engel, Matthias
Producer: 20130205
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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11.
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Regulation of the interaction between protein kinase C-related protein kinase 2 (PRK2) and its upstream kinase, 3-phosphoinositide-dependent protein kinase 1 (PDK1). [electronic resource] by
- Dettori, Rosalia
- Sonzogni, Silvina
- Meyer, Lucas
- Lopez-Garcia, Laura A
- Morrice, Nick A
- Zeuzem, Stefan
- Engel, Matthias
- Piiper, Albrecht
- Neimanis, Sonja
- Frödin, Morten
- Biondi, Ricardo M
Producer: 20091214
In:
The Journal of biological chemistry vol. 284
Availability: No items available.
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PLK1 phosphorylates PAX3-FOXO1, the inhibition of which triggers regression of alveolar Rhabdomyosarcoma. [electronic resource] by
- Thalhammer, Verena
- Lopez-Garcia, Laura A
- Herrero-Martin, David
- Hecker, Regina
- Laubscher, Dominik
- Gierisch, Maria E
- Wachtel, Marco
- Bode, Peter
- Nanni, Paolo
- Blank, Bernd
- Koscielniak, Ewa
- Schäfer, Beat W
Producer: 20150423
In:
Cancer research vol. 75
Availability: No items available.
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Structure and allosteric effects of low-molecular-weight activators on the protein kinase PDK1. [electronic resource] by
- Hindie, Valerie
- Stroba, Adriana
- Zhang, Hua
- Lopez-Garcia, Laura A
- Idrissova, Leila
- Zeuzem, Stefan
- Hirschberg, Daniel
- Schaeffer, Francis
- Jørgensen, Thomas J D
- Engel, Matthias
- Alzari, Pedro M
- Biondi, Ricardo M
Producer: 20091002
In:
Nature chemical biology vol. 5
Availability: No items available.
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14.
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Substrate-selective inhibition of protein kinase PDK1 by small compounds that bind to the PIF-pocket allosteric docking site. [electronic resource] by
- Busschots, Katrien
- Lopez-Garcia, Laura A
- Lammi, Carmen
- Stroba, Adriana
- Zeuzem, Stefan
- Piiper, Albrecht
- Alzari, Pedro M
- Neimanis, Sonja
- Arencibia, Jose M
- Engel, Matthias
- Schulze, Jörg O
- Biondi, Ricardo M
Producer: 20140710
In:
Chemistry & biology vol. 19
Availability: No items available.
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15.
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Allosteric activation of the protein kinase PDK1 with low molecular weight compounds. [electronic resource] by
- Engel, Matthias
- Hindie, Valerie
- Lopez-Garcia, Laura A
- Stroba, Adriana
- Schaeffer, Francis
- Adrian, Iris
- Imig, Jochen
- Idrissova, Leila
- Nastainczyk, Wolfgang
- Zeuzem, Stefan
- Alzari, Pedro M
- Hartmann, Rolf W
- Piiper, Albrecht
- Biondi, Ricardo M
Producer: 20070126
In:
The EMBO journal vol. 25
Availability: No items available.
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16.
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Allosteric regulation of protein kinase PKCζ by the N-terminal C1 domain and small compounds to the PIF-pocket. [electronic resource] by
- Lopez-Garcia, Laura A
- Schulze, Jörg O
- Fröhner, Wolfgang
- Zhang, Hua
- Süss, Evelyn
- Weber, Nadja
- Navratil, Jeanette
- Amon, Sabine
- Hindie, Valerie
- Zeuzem, Stefan
- Jørgensen, Thomas J D
- Alzari, Pedro M
- Neimanis, Sonja
- Engel, Matthias
- Biondi, Ricardo M
Producer: 20120326
In:
Chemistry & biology vol. 18
Availability: No items available.
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17.
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Molecular mechanism of regulation of the atypical protein kinase C by N-terminal domains and an allosteric small compound. [electronic resource] by
- Zhang, Hua
- Neimanis, Sonja
- Lopez-Garcia, Laura A
- Arencibia, José M
- Amon, Sabine
- Stroba, Adriana
- Zeuzem, Stefan
- Proschak, Ewgen
- Stark, Holger
- Bauer, Angelika F
- Busschots, Katrien
- Jørgensen, Thomas J D
- Engel, Matthias
- Schulze, Jörg O
- Biondi, Ricardo M
Producer: 20150331
In:
Chemistry & biology vol. 21
Availability: No items available.
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