Utility of frozen cell lines in medium throughput electrophysiology screening of hERG and NaV1.5 blockade. [electronic resource]
Producer: 20120608Description: 269-76 p. digitalISSN:- 1873-488X
- Amitriptyline -- pharmacology
- Cell Line, Transformed
- Cryopreservation -- methods
- Drug Evaluation, Preclinical -- methods
- ERG1 Potassium Channel
- Electrophysiological Phenomena -- drug effects
- Ether-A-Go-Go Potassium Channels -- antagonists & inhibitors
- Fluoxetine -- pharmacology
- HEK293 Cells
- Humans
- Imipramine -- pharmacology
- Membrane Potentials -- drug effects
- NAV1.5 Voltage-Gated Sodium Channel
- Patch-Clamp Techniques -- methods
- Potassium Channel Blockers -- pharmacology
- Quinidine -- pharmacology
- Sodium Channels -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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