Results
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Pronounced reduction in adenoma recurrence associated with aspirin use and a polymorphism in the ornithine decarboxylase gene. [electronic resource] by
- Martinez, Maria Elena
- O'Brien, Thomas G
- Fultz, Kimberly E
- Babbar, Naveen
- Yerushalmi, Hagit
- Qu, Ning
- Guo, Yongjun
- Boorman, David
- Einspahr, Janine
- Alberts, David S
- Gerner, Eugene W
Producer: 20030731
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 100
Availability: No items available.
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5.
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Discovery and SAR exploration of a novel series of imidazo[4,5-b]pyrazin-2-ones as potent and selective mTOR kinase inhibitors. [electronic resource] by
- Mortensen, Deborah S
- Perrin-Ninkovic, Sophie M
- Harris, Roy
- Lee, Branden G S
- Shevlin, Graziella
- Hickman, Matt
- Khambatta, Gody
- Bisonette, Rene R
- Fultz, Kimberly E
- Sankar, Sabita
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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6.
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Design and Optimization Leading to an Orally Active TTK Protein Kinase Inhibitor with Robust Single Agent Efficacy. [electronic resource] by
- Riggs, Jennifer R
- Elsner, Jan
- Cashion, Dan
- Robinson, Dale
- Tehrani, Lida
- Nagy, Mark
- Fultz, Kimberly E
- Krishna Narla, Rama
- Peng, Xiaohui
- Tran, Tam
- Kulkarni, Ashutosh
- Bahmanyar, Sogole
- Condroski, Kevin
- Pagarigan, Barbra
- Fenalti, Gustavo
- LeBrun, Laurie
- Leftheris, Katerina
- Zhu, Dan
- Boylan, John F
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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Use of core modification in the discovery of CC214-2, an orally available, selective inhibitor of mTOR kinase. [electronic resource] by
- Mortensen, Deborah S
- Sapienza, John
- Lee, Branden G S
- Perrin-Ninkovic, Sophie M
- Harris, Roy
- Shevlin, Graziella
- Parnes, Jason S
- Whitefield, Brandon
- Hickman, Matt
- Khambatta, Gody
- Bisonette, Rene R
- Peng, Sophie
- Gamez, Jim C
- Leisten, Jim
- Narla, Rama Krishna
- Fultz, Kimberly E
- Sankar, Sabita
Producer: 20130903
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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8.
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CC-223, a Potent and Selective Inhibitor of mTOR Kinase: In Vitro and In Vivo Characterization. [electronic resource] by
- Mortensen, Deborah S
- Fultz, Kimberly E
- Xu, Shuichan
- Xu, Weiming
- Packard, Garrick
- Khambatta, Godrej
- Gamez, James C
- Leisten, Jim
- Zhao, Jingjing
- Apuy, Julius
- Ghoreishi, Kamran
- Hickman, Matt
- Narla, Rama Krishna
- Bissonette, Rene
- Richardson, Samantha
- Peng, Sophie X
- Perrin-Ninkovic, Sophie
- Tran, Tam
- Shi, Tao
- Yang, Wen Qing
- Tong, Zeen
- Cathers, Brian E
- Moghaddam, Mehran F
- Canan, Stacie S
- Worland, Peter
- Sankar, Sabita
- Raymon, Heather K
Producer: 20160412
In:
Molecular cancer therapeutics vol. 14
Availability: No items available.
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9.
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Optimization of a Series of Triazole Containing Mammalian Target of Rapamycin (mTOR) Kinase Inhibitors and the Discovery of CC-115. [electronic resource] by
- Mortensen, Deborah S
- Perrin-Ninkovic, Sophie M
- Shevlin, Graziella
- Elsner, Jan
- Zhao, Jingjing
- Whitefield, Brandon
- Tehrani, Lida
- Sapienza, John
- Riggs, Jennifer R
- Parnes, Jason S
- Papa, Patrick
- Packard, Garrick
- Lee, Branden G S
- Harris, Roy
- Correa, Matthew
- Bahmanyar, Sogole
- Richardson, Samantha J
- Peng, Sophie X
- Leisten, Jim
- Khambatta, Godrej
- Hickman, Matt
- Gamez, James C
- Bisonette, René R
- Apuy, Julius
- Cathers, Brian E
- Canan, Stacie S
- Moghaddam, Mehran F
- Raymon, Heather K
- Worland, Peter
- Narla, Rama Krishna
- Fultz, Kimberly E
- Sankar, Sabita
Producer: 20151012
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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10.
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Discovery of mammalian target of rapamycin (mTOR) kinase inhibitor CC-223. [electronic resource] by
- Mortensen, Deborah S
- Perrin-Ninkovic, Sophie M
- Shevlin, Graziella
- Zhao, Jingjing
- Packard, Garrick
- Bahmanyar, Sogole
- Correa, Matthew
- Elsner, Jan
- Harris, Roy
- Lee, Branden G S
- Papa, Patrick
- Parnes, Jason S
- Riggs, Jennifer R
- Sapienza, John
- Tehrani, Lida
- Whitefield, Brandon
- Apuy, Julius
- Bisonette, René R
- Gamez, James C
- Hickman, Matt
- Khambatta, Godrej
- Leisten, Jim
- Peng, Sophie X
- Richardson, Samantha J
- Cathers, Brian E
- Canan, Stacie S
- Moghaddam, Mehran F
- Raymon, Heather K
- Worland, Peter
- Narla, Rama Krishna
- Fultz, Kimberly E
- Sankar, Sabita
Producer: 20151002
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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