Results
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Stereocontrolled total synthesis of (+)-UCS1025A. [electronic resource] by
- Uchida, Kenji
- Ogawa, Takahiro
- Yasuda, Yoshinori
- Mimura, Hiraku
- Fujimoto, Teppei
- Fukuyama, Tohru
- Wakimoto, Toshiyuki
- Asakawa, Tomohiro
- Hamashima, Yoshitaka
- Kan, Toshiyuki
Producer: 20130517
In:
Angewandte Chemie (International ed. in English) vol. 51
Availability: No items available.
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5.
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Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3-carboxamides as orally active renin inhibitors. [electronic resource] by
- Mori, Yutaka
- Ogawa, Yasuyuki
- Mochizuki, Akiyoshi
- Nakamura, Yuji
- Fujimoto, Teppei
- Sugita, Chie
- Miyazaki, Shojiro
- Tamaki, Kazuhiko
- Nagayama, Takahiro
- Nagai, Yoko
- Inoue, Shin-ichi
- Chiba, Katsuyoshi
- Nishi, Takahide
Producer: 20140326
In:
Bioorganic & medicinal chemistry vol. 21
Availability: No items available.
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6.
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Discovery of DS-8108b, a Novel Orally Bioavailable Renin Inhibitor. [electronic resource] by
- Nakamura, Yuji
- Fujimoto, Teppei
- Ogawa, Yasuyuki
- Sugita, Chie
- Miyazaki, Shojiro
- Tamaki, Kazuhiko
- Takahashi, Mizuki
- Matsui, Yumi
- Nagayama, Takahiro
- Manabe, Kenichi
- Mizuno, Makoto
- Masubuchi, Noriko
- Chiba, Katsuyoshi
- Nishi, Takahide
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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7.
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Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration. [electronic resource] by
- Matsufuji, Tetsuyoshi
- Shimada, Kousei
- Kobayashi, Shozo
- Kawamura, Asuka
- Fujimoto, Teppei
- Arita, Tsuyoshi
- Hara, Takashi
- Konishi, Masahiro
- Abe-Ohya, Rie
- Izumi, Masanori
- Sogawa, Yoshitaka
- Nagai, Youko
- Yoshida, Kazuhiro
- Takahashi, Hisashi
Producer: 20141104
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhexanamides to reduce a cardiac safety issue: discovery of DS-8108b, an orally active renin inhibitor. [electronic resource] by
- Nakamura, Yuji
- Fujimoto, Teppei
- Ogawa, Yasuyuki
- Namiki, Hidenori
- Suzuki, Sayaka
- Asano, Masayoshi
- Sugita, Chie
- Mochizuki, Akiyoshi
- Miyazaki, Shojiro
- Tamaki, Kazuhiko
- Nagai, Yoko
- Inoue, Shin-ichi
- Nagayama, Takahiro
- Kato, Mikio
- Chiba, Katsuyoshi
- Takasuna, Kiyoshi
- Nishi, Takahide
Producer: 20131203
In:
Bioorganic & medicinal chemistry vol. 21
Availability: No items available.
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9.
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Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach. [electronic resource] by
- Matsufuji, Tetsuyoshi
- Shimada, Kousei
- Kobayashi, Shozo
- Ichikawa, Masanori
- Kawamura, Asuka
- Fujimoto, Teppei
- Arita, Tsuyoshi
- Hara, Takashi
- Konishi, Masahiro
- Abe-Ohya, Rie
- Izumi, Masanori
- Sogawa, Yoshitaka
- Nagai, Yoko
- Yoshida, Kazuhiro
- Abe, Yasuyuki
- Kimura, Takako
- Takahashi, Hisashi
Producer: 20151022
In:
Bioorganic & medicinal chemistry vol. 23
Availability: No items available.
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