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Adamantane 11-beta-HSD-1 inhibitors: Application of an isocyanide multicomponent reaction. [electronic resource] by
- Sorensen, Bryan
- Rohde, Jeff
- Wang, Jiahong
- Fung, Steven
- Monzon, Katina
- Chiou, William
- Pan, Liping
- Deng, Xiaoqing
- Stolarik, DeAnne
- Frevert, Ernst U
- Jacobson, Peer
- Link, J T
Producer: 20070108
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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Bioequivalence of saxagliptin/metformin immediate release (IR) fixed-dose combination tablets and single-component saxagliptin and metformin IR tablets in healthy adult subjects. [electronic resource] by
- Upreti, Vijay V
- Keung, Chi-Fung
- Boulton, David W
- Chang, Ming
- Li, Li
- Tang, Angela
- Hsiang, Bonnie C
- Quamina-Edghill, Donette
- Frevert, Ernst U
- Lacreta, Frank P
Producer: 20131028
In:
Clinical drug investigation vol. 33
Availability: No items available.
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6.
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Discovery of potent and selective inhibitors of 11beta-HSD1 for the treatment of metabolic syndrome. [electronic resource] by
- Richards, Steven
- Sorensen, Bryan
- Jae, Hwan-Soo
- Winn, Marty
- Chen, Yixian
- Wang, Jiahong
- Fung, Steven
- Monzon, Katina
- Frevert, Ernst U
- Jacobson, Peer
- Sham, Hing
- Link, J T
Producer: 20070216
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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7.
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The synthesis and structure-activity relationship studies of selective acetyl-CoA carboxylase inhibitors containing 4-(thiazol-5-yl)but-3-yn-2-amino motif: polar region modifications. [electronic resource] by
- Xu, Xiangdong
- Weitzberg, Moshe
- Keyes, Robert F
- Li, Qun
- Wang, Rongqi
- Wang, Xiaojun
- Zhang, Xiaolin
- Frevert, Ernst U
- Camp, Heidi S
- Beutel, Bruce A
- Sham, Hing L
- Gu, Yu Gui
Producer: 20070529
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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Microarrayed compound screening (microARCS) to identify activators and inhibitors of AMP-activated protein kinase. [electronic resource] by
- Anderson, Steven N
- Cool, Barbara L
- Kifle, Lemma
- Chiou, William
- Egan, David A
- Barrett, Leo W
- Richardson, Paul L
- Frevert, Ernst U
- Warrior, Usha
- Kofron, James L
- Burns, David J
Producer: 20041223
In:
Journal of biomolecular screening vol. 9
Availability: No items available.
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Identification and characterization of a small molecule AMPK activator that treats key components of type 2 diabetes and the metabolic syndrome. [electronic resource] by
- Cool, Barbara
- Zinker, Bradley
- Chiou, William
- Kifle, Lemma
- Cao, Ning
- Perham, Matthew
- Dickinson, Robert
- Adler, Andrew
- Gagne, Gerard
- Iyengar, Rajesh
- Zhao, Gang
- Marsh, Kennan
- Kym, Philip
- Jung, Paul
- Camp, Heidi S
- Frevert, Ernst
Producer: 20060816
In:
Cell metabolism vol. 3
Availability: No items available.
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10.
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Structure-activity relationships for a novel series of thiazolyl phenyl ether derivatives exhibiting potent and selective acetyl-CoA carboxylase 2 inhibitory activity. [electronic resource] by
- Clark, Richard F
- Zhang, Tianyuan
- Xin, Zhili
- Liu, Gang
- Wang, Ying
- Hansen, T Matthew
- Wang, Xiaojun
- Wang, Rongqi
- Zhang, Xiaolin
- Frevert, Ernst U
- Camp, Heidi S
- Beutel, Bruce A
- Sham, Hing L
- Gu, Yu Gui
Producer: 20070108
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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11.
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Synthesis and structure-activity relationships of N-{3-[2-(4-alkoxyphenoxy)thiazol-5-yl]-1- methylprop-2-ynyl}carboxy derivatives as selective acetyl-CoA carboxylase 2 inhibitors. [electronic resource] by
- Gu, Yu Gui
- Weitzberg, Moshe
- Clark, Richard F
- Xu, Xiangdong
- Li, Qun
- Zhang, Tianyuan
- Hansen, T Matthew
- Liu, Gang
- Xin, Zhili
- Wang, Xiaojun
- Wang, Rongqi
- McNally, Teresa
- Zinker, Bradley A
- Frevert, Ernst U
- Camp, Heidi S
- Camp, Heidi
- Beutel, Bruce A
- Sham, Hing L
Producer: 20060816
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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12.
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Adamantane sulfone and sulfonamide 11-beta-HSD1 Inhibitors. [electronic resource] by
- Sorensen, Bryan
- Winn, Martin
- Rohde, Jeff
- Shuai, Qi
- Wang, Jiahong
- Fung, Steven
- Monzon, Katina
- Chiou, William
- Stolarik, DeAnne
- Imade, Hovis
- Pan, Liping
- Deng, Xiaoqing
- Chovan, Linda
- Longenecker, Kenton
- Judge, Russell
- Qin, Wenying
- Brune, Michael
- Camp, Heidi
- Frevert, Ernst U
- Jacobson, Peer
- Link, J T
Producer: 20070409
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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13.
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Discovery and metabolic stabilization of potent and selective 2-amino-N-(adamant-2-yl) acetamide 11beta-hydroxysteroid dehydrogenase type 1 inhibitors. [electronic resource] by
- Rohde, Jeffrey J
- Pliushchev, Marina A
- Sorensen, Bryan K
- Wodka, Dariusz
- Shuai, Qi
- Wang, Jiahong
- Fung, Steven
- Monzon, Katina M
- Chiou, William J
- Pan, Liping
- Deng, Xiaoqing
- Chovan, Linda E
- Ramaiya, Atul
- Mullally, Mark
- Henry, Rodger F
- Stolarik, DeAnne F
- Imade, Hovis M
- Marsh, Kennan C
- Beno, David W A
- Fey, Thomas A
- Droz, Brian A
- Brune, Michael E
- Camp, Heidi S
- Sham, Hing L
- Frevert, Ernst Uli
- Jacobson, Peer B
- Link, J T
Producer: 20070307
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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