Results
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Evaluation of indenoisoquinoline topoisomerase I inhibitors using a hollow fiber assay. [electronic resource] by
- Morrell, Andrew
- Jayaraman, Muthusamy
- Nagarajan, Muthukaman
- Fox, Brian M
- Meckley, Marintha Rae
- Ioanoviciu, Alexandra
- Pommier, Yves
- Antony, Smitha
- Hollingshead, Melinda
- Cushman, Mark
Producer: 20061006
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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4.
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Novel pyrrolidine melanin-concentrating hormone receptor 1 antagonists with reduced hERG inhibition. [electronic resource] by
- Fox, Brian M
- Natero, Reina
- Richard, Kevin
- Connors, Richard
- Roveto, Philip M
- Beckmann, Holger
- Haller, Katrin
- Golde, Justin
- Xiao, Shou-Hua
- Kayser, Frank
Producer: 20110719
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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Discovery of pyrrolopyridazines as novel DGAT1 inhibitors. [electronic resource] by
- Fox, Brian M
- Iio, Kiyosei
- Li, Kexue
- Choi, Rebeka
- Inaba, Takashi
- Jackson, Simon
- Sagawa, Shoichi
- Shan, Bei
- Tanaka, Masahiro
- Yoshida, Atsuhito
- Kayser, Frank
Producer: 20110113
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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A selective prostaglandin E2 receptor subtype 2 (EP2) antagonist increases the macrophage-mediated clearance of amyloid-beta plaques. [electronic resource] by
- Fox, Brian M
- Beck, Hilary P
- Roveto, Philip M
- Kayser, Frank
- Cheng, Qingwen
- Dou, Hannah
- Williamson, Toni
- Treanor, James
- Liu, Hantao
- Jin, Lixia
- Xu, Guifen
- Ma, Ji
- Wang, Songli
- Olson, Steven H
Producer: 20151002
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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Discovery of 6-phenylpyrimido[4,5-b][1,4]oxazines as potent and selective acyl CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitors with in vivo efficacy in rodents. [electronic resource] by
- Fox, Brian M
- Sugimoto, Kazuyuki
- Iio, Kiyosei
- Yoshida, Atsuhito
- Zhang, Jian Ken
- Li, Kexue
- Hao, Xiaolin
- Labelle, Marc
- Smith, Marie-Louise
- Rubenstein, Steven M
- Ye, Guosen
- McMinn, Dustin
- Jackson, Simon
- Choi, Rebekah
- Shan, Bei
- Ma, Ji
- Miao, Shichang
- Matsui, Takuya
- Ogawa, Nobuya
- Suzuki, Masahiro
- Kobayashi, Akio
- Ozeki, Hidekazu
- Okuma, Chihiro
- Ishii, Yukihito
- Tomimoto, Daisuke
- Furakawa, Noboru
- Tanaka, Masahiro
- Matsushita, Mutsuyoshi
- Takahashi, Mitsuru
- Inaba, Takashi
- Sagawa, Shoichi
- Kayser, Frank
Producer: 20140706
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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Novel inhibitors of the MDM2-p53 interaction featuring hydrogen bond acceptors as carboxylic acid isosteres. [electronic resource] by
- Gonzalez, Ana Z
- Li, Zhihong
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan
- Jin, Lixia
- Li, Yihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Sun, Daqing
- Medina, Julio C
Producer: 20140708
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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9.
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Discovery of AM-7209, a potent and selective 4-amidobenzoic acid inhibitor of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Yan, Xuelei
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Duquette, Jason
- Eksterowicz, John
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Houze, Jonathan
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- Oliner, Jonathan D
- Osgood, Tao
- Saiki, Anne Y
- Shaffer, Paul
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20150310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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10.
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Structure-based design of novel inhibitors of the MDM2-p53 interaction. [electronic resource] by
- Rew, Yosup
- Sun, Daqing
- Gonzalez-Lopez De Turiso, Felix
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Deignan, Jeffrey
- Fox, Brian M
- Gustin, Darin
- Huang, Xin
- Jiang, Min
- Jiao, Xianyun
- Jin, Lixia
- Kayser, Frank
- Kopecky, David J
- Li, Yihong
- Lo, Mei-Chu
- Long, Alexander M
- Michelsen, Klaus
- Oliner, Jonathan D
- Osgood, Tao
- Ragains, Mark
- Saiki, Anne Y
- Schneider, Steve
- Toteva, Maria
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Medina, Julio C
- Olson, Steven H
Producer: 20121001
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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11.
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Selective and potent morpholinone inhibitors of the MDM2-p53 protein-protein interaction. [electronic resource] by
- Gonzalez, Ana Z
- Eksterowicz, John
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chow, David
- Duquette, Jason
- Fox, Brian M
- Fu, Jiasheng
- Huang, Xin
- Houze, Jonathan B
- Jin, Lixia
- Li, Yihong
- Li, Zhihong
- Ling, Yun
- Lo, Mei-Chu
- Long, Alexander M
- McGee, Lawrence R
- McIntosh, Joel
- McMinn, Dustin L
- Oliner, Jonathan D
- Osgood, Tao
- Rew, Yosup
- Saiki, Anne Y
- Shaffer, Paul
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Zhao, Xiaoning
- Zhou, Jing
- Olson, Steven H
- Medina, Julio C
- Sun, Daqing
Producer: 20140527
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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12.
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Discovery of AMG 232, a potent, selective, and orally bioavailable MDM2-p53 inhibitor in clinical development. [electronic resource] by
- Sun, Daqing
- Li, Zhihong
- Rew, Yosup
- Gribble, Michael
- Bartberger, Michael D
- Beck, Hilary P
- Canon, Jude
- Chen, Ada
- Chen, Xiaoqi
- Chow, David
- Deignan, Jeffrey
- Duquette, Jason
- Eksterowicz, John
- Fisher, Benjamin
- Fox, Brian M
- Fu, Jiasheng
- Gonzalez, Ana Z
- Gonzalez-Lopez De Turiso, Felix
- Houze, Jonathan B
- Huang, Xin
- Jiang, Min
- Jin, Lixia
- Kayser, Frank
- Liu, Jiwen Jim
- Lo, Mei-Chu
- Long, Alexander M
- Lucas, Brian
- McGee, Lawrence R
- McIntosh, Joel
- Mihalic, Jeff
- Oliner, Jonathan D
- Osgood, Tao
- Peterson, Matthew L
- Roveto, Philip
- Saiki, Anne Y
- Shaffer, Paul
- Toteva, Maria
- Wang, Yingcai
- Wang, Yu Chung
- Wortman, Sarah
- Yakowec, Peter
- Yan, Xuelei
- Ye, Qiuping
- Yu, Dongyin
- Yu, Ming
- Zhao, Xiaoning
- Zhou, Jing
- Zhu, Jiang
- Olson, Steven H
- Medina, Julio C
Producer: 20140429
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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