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Design, synthesis, and evaluation of a novel dual FMS-like tyrosine kinase 3/stem cell factor receptor (FLT3/c-KIT) inhibitor for the treatment of acute myelogenous leukemia. [electronic resource] by
- Davies, Robert J
- Pierce, Albert C
- Forster, Cornelia
- Grey, Ron
- Xu, Jinwang
- Arnost, Michael
- Choquette, Deborah
- Galullo, Vincent
- Tian, Shi-Kai
- Henkel, Greg
- Chen, Guanjing
- Heidary, David K
- Ma, Joanne
- Stuver-Moody, Cameron
- Namchuk, Mark
Producer: 20120103
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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5.
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VX-322: a novel dual receptor tyrosine kinase inhibitor for the treatment of acute myelogenous leukemia. [electronic resource] by
- Heidary, David K
- Huang, George
- Boucher, Diane
- Ma, Jianguo
- Forster, Cornelia
- Grey, Ron
- Xu, Jinwang
- Arnost, Michael
- Choquette, Deborah
- Chen, Guanjing
- Zhou, Jie-Hua
- Yao, Yung-Mae
- Ball, Edward D
- Namchuk, Mark
- Davies, Robert J
- Henkel, Greg
Producer: 20120409
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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Discovery of diamide compounds as diacylglycerol acyltransferase 1 (DGAT1) inhibitors. [electronic resource] by
- Nakajima, Katsumasa
- April, Myriam
- Brewer, Jason T
- Daniels, Thomas
- Forster, Cornelia J
- Gilmore, Thomas A
- Jain, Monish
- Kanter, Aaron
- Kwak, Youngshin
- Li, Jingzhou
- McQuire, Les
- Serrano-Wu, Michael H
- Streeper, Ryan
- Szklennik, Paul
- Thompson, James
- Wang, Bing
Producer: 20160930
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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A new structural alert for benzimidazoles: 2,6-dimethylphenyl substituents increase mutagenic potential and time-dependent CYP3A4 inhibition risk. [electronic resource] by
- Kwak, Youngshin
- Coppola, Gary
- Forster, Cornelia J
- Gilmore, Thomas A
- Gong, Yongjin
- Kanter, Aaron
- Neubert, Alan
- Stroup, Bryan
- Szklennik, Paul
- Glowienke, Susanne
- Stadelmann, Pascal
- Bell, Leslie
- Bickford, Shari
- Gangl, Eric
- Gunduz, Mithat
- Jain, Monish
- Zhan, Jenny
- Serrano-Wu, Michael H
Producer: 20110614
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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8.
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Discovery of an Orally Bioavailable Benzimidazole Diacylglycerol Acyltransferase 1 (DGAT1) Inhibitor That Suppresses Body Weight Gain in Diet-Induced Obese Dogs and Postprandial Triglycerides in Humans. [electronic resource] by
- Nakajima, Katsumasa
- Chatelain, Ricardo
- Clairmont, Kevin B
- Commerford, Renee
- Coppola, Gary M
- Daniels, Thomas
- Forster, Cornelia J
- Gilmore, Thomas A
- Gong, Yongjin
- Jain, Monish
- Kanter, Aaron
- Kwak, Youngshin
- Li, Jingzhou
- Meyers, Charles D
- Neubert, Alan D
- Szklennik, Paul
- Tedesco, Vivienne
- Thompson, James
- Truong, David
- Yang, Qing
- Hubbard, Brian K
- Serrano-Wu, Michael H
Producer: 20170704
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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9.
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Discovery of 4-((2 [electronic resource] by
- Mainolfi, Nello
- Ehara, Takeru
- Karki, Rajeshri G
- Anderson, Karen
- Mac Sweeney, Aengus
- Liao, Sha-Mei
- Argikar, Upendra A
- Jendza, Keith
- Zhang, Chun
- Powers, James
- Klosowski, Daniel W
- Crowley, Maura
- Kawanami, Toshio
- Ding, Jian
- April, Myriam
- Forster, Cornelia
- Serrano-Wu, Michael
- Capparelli, Michael
- Ramqaj, Rrezarta
- Solovay, Catherine
- Cumin, Frederic
- Smith, Thomas M
- Ferrara, Luciana
- Lee, Wendy
- Long, Debby
- Prentiss, Melissa
- De Erkenez, Andrea
- Yang, Louis
- Liu, Fang
- Sellner, Holger
- Sirockin, Finton
- Valeur, Eric
- Erbel, Paulus
- Ostermeier, Daniela
- Ramage, Paul
- Gerhartz, Bernd
- Schubart, Anna
- Flohr, Stefanie
- Gradoux, Nathalie
- Feifel, Roland
- Vogg, Barbara
- Wiesmann, Christian
- Maibaum, Jürgen
- Eder, Jörg
- Sedrani, Richard
- Harrison, Richard A
- Mogi, Muneto
- Jaffee, Bruce D
- Adams, Christopher M
Producer: 20201112
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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