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Internalization of the chemokine receptor CCR4 can be evoked by orthosteric and allosteric receptor antagonists. [electronic resource] by
- Ajram, Laura
- Begg, Malcolm
- Slack, Robert
- Cryan, Jenni
- Hall, David
- Hodgson, Simon
- Ford, Alison
- Barnes, Ashley
- Swieboda, Dawid
- Mousnier, Aurelie
- Solari, Roberto
Producer: 20141203
In:
European journal of pharmacology vol. 729
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Lead identification of benzimidazolone and azabenzimidazolone arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists. [electronic resource] by
- Miah, Afjal H
- Abas, Hossay
- Begg, Malcolm
- Marsh, Benjamin J
- O'Flynn, Daniel E
- Ford, Alison J
- Percy, Jonathan M
- Procopiou, Panayiotis A
- Richards, Steve A
- Rumley, Sally-Anne
Producer: 20150904
In:
Bioorganic & medicinal chemistry vol. 22
Availability: No items available.
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Effect of lamotrigine on the activities of monoamine oxidases A and B in vitro and on monoamine disposition in vivo. [electronic resource] by
- Southam, Eric
- Pereira, Rui
- Stratton, Sharon C
- Sargent, Rebecca
- Ford, Alison J
- Butterfield, Lindsay J
- Wheable, Jane D
- Beckett, Simon R G
- Roe, Clare
- Marsden, Charles A
- Hagan, Russell M
Producer: 20051025
In:
European journal of pharmacology vol. 519
Availability: No items available.
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Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H [electronic resource] by
- Procopiou, Panayiotis A
- Ford, Alison J
- Gore, Paul M
- Hancock, Ashley P
- Hodgson, Simon T
- Holmes, Duncan S
- Looker, Brian E
- Vile, Sadie
- Clark, Kenneth L
- Saunders, Ken A
- Slack, Robert J
- Watts, Clarissa J
Producer: 20171206
In:
Bioorganic & medicinal chemistry letters vol. 27
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Design of Phthalazinone Amide Histamine H [electronic resource] by
- Procopiou, Panayiotis A
- Ford, Alison J
- Gore, Paul M
- Looker, Brian E
- Hodgson, Simon T
- Holmes, Duncan S
- Vile, Sadie
- Clark, Kenneth L
- Saunders, Ken A
- Slack, Robert J
- Rowedder, James E
- Watts, Clarissa J
Publication details: ACS medicinal chemistry letters May 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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Discovery of a rapidly metabolized, long-acting β(2) adrenergic receptor agonist with a short onset time incorporating a sulfone group suitable for once-daily dosing. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Biggadike, Keith
- Butchers, Peter R
- Craven, Andrew
- Ford, Alison J
- Guntrip, Stephen B
- Holmes, Duncan S
- Hughes, Sara C
- Jones, Anne E
- Looker, Brian E
- Mutch, Peter J
- Ruston, Mark
- Needham, Deborah
- Smith, Claire E
Producer: 20140310
In:
Journal of medicinal chemistry vol. 57
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The discovery of long-acting saligenin β₂ adrenergic receptor agonists incorporating hydantoin or uracil rings. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Butchers, Peter R
- Conroy, Richard
- Emmons, Amanda
- Ford, Alison J
- Jeulin, Séverine
- Looker, Brian E
- Lunniss, Gillian E
- Morrison, Valerie S
- Mutch, Peter J
- Perciaccante, Rossana
- Ruston, Mark
- Smith, Claire E
- Somers, Graham
Producer: 20111220
In:
Bioorganic & medicinal chemistry vol. 19
Availability: No items available.
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Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating arylsulfonamide groups. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Biggadike, Keith
- Butchers, Peter R
- Coe, Diane M
- Conroy, Richard
- Edney, Dean D
- Field, Rita N
- Ford, Alison J
- Guntrip, Stephen B
- Looker, Brian E
- McLay, Iain M
- Monteith, Michael J
- Morrison, Valerie S
- Mutch, Peter J
- Richards, Stephen A
- Sasse, Rosemary
- Smith, Claire E
Producer: 20090506
In:
Journal of medicinal chemistry vol. 52
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Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating metabolic inactivation: an antedrug approach. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, Victoria J
- Bevan, Nicola J
- Biggadike, Keith
- Box, Philip C
- Butchers, Peter R
- Coe, Diane M
- Conroy, Richard
- Emmons, Amanda
- Ford, Alison J
- Holmes, Duncan S
- Horsley, Helen
- Kerr, Fern
- Li-Kwai-Cheung, Anne-Marie
- Looker, Brian E
- Mann, Inderjit S
- McLay, Iain M
- Morrison, Valerie S
- Mutch, Peter J
- Smith, Claire E
- Tomlin, Paula
Producer: 20100701
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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Synthesis and structure-activity relationships of indazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists. [electronic resource] by
- Procopiou, Panayiotis A
- Barrett, John W
- Barton, Nicholas P
- Begg, Malcolm
- Clapham, David
- Copley, Royston C B
- Ford, Alison J
- Graves, Rebecca H
- Hall, David A
- Hancock, Ashley P
- Hill, Alan P
- Hobbs, Heather
- Hodgson, Simon T
- Jumeaux, Coline
- Lacroix, Yannick M L
- Miah, Afjal H
- Morriss, Karen M L
- Needham, Deborah
- Sheriff, Emma B
- Slack, Robert J
- Smith, Claire E
- Sollis, Steven L
- Staton, Hugo
Producer: 20130514
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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