Results
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Discovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor-Prolyl Hydroxylase Inhibitor for Anemia. [electronic resource] by
- Ariazi, Jennifer L
- Duffy, Kevin J
- Adams, David F
- Fitch, Duke M
- Luo, Lusong
- Pappalardi, Melissa
- Biju, Mangatt
- DiFilippo, Erin Hugger
- Shaw, Tony
- Wiggall, Ken
- Erickson-Miller, Connie
Producer: 20171121
In:
The Journal of pharmacology and experimental therapeutics vol. 363
Availability: No items available.
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4.
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Synthesis and biological activity of heteroaryl 3-(1,1-dioxo-2H-(1,2,4)-benzothiadizin-3-yl)-4-hydroxy-2(1H)-quinolinone derivatives as hepatitis C virus NS5B polymerase inhibitors. [electronic resource] by
- Tedesco, Rosanna
- Chai, Deping
- Darcy, Michael G
- Dhanak, Dashyant
- Fitch, Duke M
- Gates, Adam
- Johnston, Victor K
- Keenan, Richard M
- Lin-Goerke, Juili
- Sarisky, Robert T
- Shaw, Antony N
- Valko, Klara L
- Wiggall, Kenneth J
- Zimmerman, Michael N
- Duffy, Kevin J
Producer: 20091207
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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5.
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Substituted benzothiadizine inhibitors of Hepatitis C virus polymerase. [electronic resource] by
- Shaw, Antony N
- Tedesco, Rosanna
- Bambal, Ramesh
- Chai, Deping
- Concha, Nestor O
- Darcy, Michael G
- Dhanak, Dashyant
- Duffy, Kevin J
- Fitch, Duke M
- Gates, Adam
- Johnston, Victor K
- Keenan, Richard M
- Lin-Goerke, Juili
- Liu, Nannan
- Sarisky, Robert T
- Wiggall, Kenneth J
- Zimmerman, Michael N
Producer: 20091207
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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6.
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3-(1,1-dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones, potent inhibitors of hepatitis C virus RNA-dependent RNA polymerase. [electronic resource] by
- Tedesco, Rosanna
- Shaw, Antony N
- Bambal, Ramesh
- Chai, Deping
- Concha, Nestor O
- Darcy, Michael G
- Dhanak, Dashyant
- Fitch, Duke M
- Gates, Adam
- Gerhardt, Warren G
- Halegoua, Dina L
- Han, Chao
- Hofmann, Glenn A
- Johnston, Victor K
- Kaura, Arun C
- Liu, Nannan
- Keenan, Richard M
- Lin-Goerke, Juili
- Sarisky, Robert T
- Wiggall, Kenneth J
- Zimmerman, Michael N
- Duffy, Kevin J
Producer: 20060329
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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7.
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Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. [electronic resource] by
- Qian, Xiangping
- McDonald, Andrew
- Zhou, Han-Jie
- Adams, Nicholas D
- Parrish, Cynthia A
- Duffy, Kevin J
- Fitch, Duke M
- Tedesco, Rosanna
- Ashcraft, Luke W
- Yao, Bing
- Jiang, Hong
- Huang, Jennifer K
- Marin, Melchor V
- Aroyan, Carrie E
- Wang, Jianchao
- Ahmed, Seyed
- Burgess, Joelle L
- Chaudhari, Amita M
- Donatelli, Carla A
- Darcy, Michael G
- Ridgers, Lance H
- Newlander, Ken A
- Schmidt, Stanley J
- Chai, Deping
- Colón, Mariela
- Zimmerman, Michael N
- Lad, Latesh
- Sakowicz, Roman
- Schauer, Stephen
- Belmont, Lisa
- Baliga, Ramesh
- Pierce, Daniel W
- Finer, Jeffrey T
- Wang, Zhengping
- Morgan, Bradley P
- Morgans, David J
- Auger, Kurt R
- Sung, Chiu-Mei
- Carson, Jeff D
- Luo, Lusong
- Hugger, Erin D
- Copeland, Robert A
- Sutton, David
- Elliott, John D
- Jackson, Jeffrey R
- Wood, Kenneth W
- Dhanak, Dashyant
- Bergnes, Gustave
- Knight, Steven D
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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