Results
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1.
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Preclinical antitumor activity of BMS-599626, a pan-HER kinase inhibitor that inhibits HER1/HER2 homodimer and heterodimer signaling. [electronic resource] by
- Wong, Tai W
- Lee, Francis Y
- Yu, Chiang
- Luo, Feng R
- Oppenheimer, Simone
- Zhang, Hongjian
- Smykla, Richard A
- Mastalerz, Harold
- Fink, Brian E
- Hunt, John T
- Gavai, Ashvinikumar V
- Vite, Gregory D
Producer: 20061114
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 12
Availability: No items available.
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2.
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Novel pyrrolo[2,1-f][1,2,4]triazin-4-amines: Dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Fink, Brian E
- Norris, Derek
- Mastalerz, Harold
- Chen, Ping
- Goyal, Bindu
- Zhao, Yufen
- Kim, Soong-Hoon
- Vite, Gregory D
- Lee, Francis Y
- Zhang, Hongjian
- Oppenheimer, Simone
- Tokarski, John S
- Wong, Tai W
- Gavai, Ashvinikumar V
Producer: 20110425
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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3.
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New dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Fink, Brian E
- Vite, Gregory D
- Mastalerz, Harold
- Kadow, John F
- Kim, Soong-Hoon
- Leavitt, Kenneth J
- Du, Karen
- Crews, Donald
- Mitt, Toomas
- Wong, Tai W
- Hunt, John T
- Vyas, Dolatrai M
- Tokarski, John S
Producer: 20051223
In:
Bioorganic & medicinal chemistry letters vol. 15
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4.
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Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17beta-hydroxysteroid dehydrogenase type 3. [electronic resource] by
- Fink, Brian E
- Gavai, Ashvinikumar V
- Tokarski, John S
- Goyal, Bindu
- Misra, Raj
- Xiao, Hai-Yun
- Kimball, S David
- Han, Wen-Ching
- Norris, Derek
- Spires, Thomas E
- You, Dan
- Gottardis, Marco M
- Lorenzi, Matthew V
- Vite, Gregory D
Producer: 20060417
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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5.
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Identification of novel functional inhibitors of 17beta-hydroxysteroid dehydrogenase type III (17beta-HSD3). [electronic resource] by
- Spires, Thomas E
- Fink, Brian E
- Kick, Ellen K
- You, Dan
- Rizzo, Cheryl A
- Takenaka, Ivone
- Lawrence, R Michael
- Ruan, Zheming
- Salvati, Mark E
- Vite, Gregory D
- Weinmann, Roberto
- Attar, Ricardo M
- Gottardis, Marco M
- Lorenzi, Matthew V
Producer: 20051025
In:
The Prostate vol. 65
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6.
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Identification of 2-amino-5-(thioaryl)thiazoles as inhibitors of nerve growth factor receptor TrkA. [electronic resource] by
- Kim, Soong-Hoon
- Tokarski, John S
- Leavitt, Kenneth J
- Fink, Brian E
- Salvati, Mark E
- Moquin, Robert
- Obermeier, Mary T
- Trainor, George L
- Vite, Gregory G
- Stadnick, Linda K
- Lippy, Jonathan S
- You, Dan
- Lorenzi, Matthew V
- Chen, Ping
Producer: 20080527
In:
Bioorganic & medicinal chemistry letters vol. 18
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7.
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Constitutively active receptor tyrosine kinases as oncogenes in preclinical models for cancer therapeutics. [electronic resource] by
- Kellar, Kristen A
- Lorenzi, Matthew V
- Ho, Ching Ping
- You, Dan
- Wen, Mei-Li
- Ryseck, Rolf P
- Oppenheimer, Simone
- Fink, Brian E
- Vite, Gregory D
- Rowley, Bruce R
- Yu, Chiang
- Bol, David K
- Lee, Francis Y
- Wong, Tai W
Producer: 20061004
In:
Molecular cancer therapeutics vol. 5
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8.
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Discovery of 4-Azaindole Inhibitors of TGFβRI as Immuno-oncology Agents. [electronic resource] by
- Zhang, Yong
- Zhao, Yufen
- Tebben, Andrew J
- Sheriff, Steven
- Ruzanov, Max
- Fereshteh, Mark P
- Fan, Yi
- Lippy, Jonathan
- Swanson, Jesse
- Ho, Ching-Ping
- Wautlet, Barri S
- Rose, Anne
- Parrish, Karen
- Yang, Zheng
- Donnell, Andrew F
- Zhang, Liping
- Fink, Brian E
- Vite, Gregory D
- Augustine-Rauch, Karen
- Fargnoli, Joseph
- Borzilleri, Robert M
Publication details: ACS medicinal chemistry letters Nov 2018
In:
ACS medicinal chemistry letters vol. 9
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9.
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5-((4-Aminopiperidin-1-yl)methyl)pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Mastalerz, Harold
- Chang, Ming
- Chen, Ping
- Fink, Brian E
- Gavai, Ashvinikumar
- Han, Wen-Ching
- Johnson, Walter
- Langley, David
- Lee, Francis Y
- Leavitt, Kenneth
- Marathe, Punit
- Norris, Derek
- Oppenheimer, Simone
- Sleczka, Bogdan
- Tarrant, James
- Tokarski, John S
- Vite, Gregory D
- Vyas, Dolatrai M
- Wong, Henry
- Wong, Tai W
- Zhang, Hongjian
- Zhang, Guifen
Producer: 20071120
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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10.
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Heterobicyclic inhibitors of transforming growth factor beta receptor I (TGFβRI). [electronic resource] by
- Harikrishnan, Lalgudi S
- Warrier, Jayakumar
- Tebben, Andrew J
- Tonukunuru, Gopikishan
- Madduri, Sudhakara R
- Baligar, Vishweshwaraiah
- Mannoori, Raju
- Seshadri, Balaji
- Rahaman, Hasibur
- Arunachalam, P N
- Dikundwar, Amol G
- Fink, Brian E
- Fargnoli, Joseph
- Fereshteh, Mark
- Fan, Yi
- Lippy, Jonathan
- Ho, Ching-Ping
- Wautlet, Barri
- Sheriff, Steven
- Ruzanov, Max
- Borzilleri, Robert M
Producer: 20181001
In:
Bioorganic & medicinal chemistry vol. 26
Availability: No items available.
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11.
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New C-5 substituted pyrrolotriazine dual inhibitors of EGFR and HER2 protein tyrosine kinases. [electronic resource] by
- Mastalerz, Harold
- Chang, Ming
- Chen, Ping
- Dextraze, Pierre
- Fink, Brian E
- Gavai, Ashvinikumar
- Goyal, Bindu
- Han, Wen-Ching
- Johnson, Walter
- Langley, David
- Lee, Francis Y
- Marathe, Punit
- Mathur, Arvind
- Oppenheimer, Simone
- Ruediger, Edward
- Tarrant, James
- Tokarski, John S
- Vite, Gregory D
- Vyas, Dolatrai M
- Wong, Henry
- Wong, Tai W
- Zhang, Hongjian
- Zhang, Guifen
Producer: 20070725
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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12.
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Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists. [electronic resource] by
- Harikrishnan, Lalgudi S
- Gill, Patrice
- Kamau, Muthoni G
- Qin, Lan-Ying
- Ruan, Zheming
- O'Malley, Daniel
- Huynh, Tram
- Stachura, Sylwia
- Cavallaro, Cullen L
- Lu, Zhonghui
- J-W Duan, James
- Weigelt, Carolyn A
- Sack, John S
- Ruzanov, Max
- Khan, Javed
- Gururajan, Murali
- Wong, Jessica J
- Huang, Yanling
- Yarde, Melissa
- Li, Zhuyin
- Chen, Cliff
- Sun, Huadong
- Borowski, Virna
- Murtaza, Anwar
- Fink, Brian E
Producer: 20210512
In:
Bioorganic & medicinal chemistry letters vol. 30
Availability: No items available.
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13.
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Discovery and preclinical evaluation of [4-[[1-(3-fluorophenyl)methyl]-1H-indazol-5-ylamino]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamic acid, (3S)-3-morpholinylmethyl ester (BMS-599626), a selective and orally efficacious inhibitor of human epidermal growth factor receptor 1 and 2 kinases. [electronic resource] by
- Gavai, Ashvinikumar V
- Fink, Brian E
- Fairfax, David J
- Martin, Gregory S
- Rossiter, Lana M
- Holst, Christian L
- Kim, Soong-Hoon
- Leavitt, Kenneth J
- Mastalerz, Harold
- Han, Wen-Ching
- Norris, Derek
- Goyal, Bindu
- Swaminathan, Shankar
- Patel, Bharat
- Mathur, Arvind
- Vyas, Dolatrai M
- Tokarski, John S
- Yu, Chiang
- Oppenheimer, Simone
- Zhang, Hongjian
- Marathe, Punit
- Fargnoli, Joseph
- Lee, Francis Y
- Wong, Tai W
- Vite, Gregory D
Producer: 20091215
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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