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In vivo potent BM635 analogue with improved drug-like properties. [electronic resource] by
- Poce, Giovanna
- Cocozza, Martina
- Alfonso, Salvatore
- Consalvi, Sara
- Venditti, Giulia
- Fernandez-Menendez, Raquel
- Bates, Robert H
- Barros Aguirre, David
- Ballell, Lluis
- De Logu, Alessandro
- Vistoli, Giulio
- Biava, Mariangela
Producer: 20180302
In:
European journal of medicinal chemistry vol. 145
Availability: No items available.
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3.
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Novel Pyrazole-Containing Compounds Active against [electronic resource] by
- Poce, Giovanna
- Consalvi, Sara
- Venditti, Giulia
- Alfonso, Salvatore
- Desideri, Nicoletta
- Fernandez-Menendez, Raquel
- Bates, Robert H
- Ballell, Lluis
- Barros Aguirre, David
- Rullas, Joaquin
- De Logu, Alessandro
- Gardner, Michelle
- Ioerger, Thomas R
- Rubin, Eric J
- Biava, Mariangela
Publication details: ACS medicinal chemistry letters Oct 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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4.
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Design, synthesis, and evaluation of new thiadiazole-based direct inhibitors of enoyl acyl carrier protein reductase (InhA) for the treatment of tuberculosis. [electronic resource] by
- Šink, Roman
- Sosič, Izidor
- Živec, Matej
- Fernandez-Menendez, Raquel
- Turk, Samo
- Pajk, Stane
- Alvarez-Gomez, Daniel
- Lopez-Roman, Eva Maria
- Gonzales-Cortez, Carolina
- Rullas-Triconado, Joaquin
- Angulo-Barturen, Inigo
- Barros, David
- Ballell-Pages, Lluís
- Young, Robert J
- Encinas, Lourdes
- Gobec, Stanislav
Producer: 20150331
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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Discovery of heterocyclic replacements for the coumarin core of anti-tubercular FadD32 inhibitors. [electronic resource] by
- Fang, Chao
- Lee, Katie K
- Nietupski, Raymond
- Bates, Robert H
- Fernandez-Menendez, Raquel
- Lopez-Roman, Eva Maria
- Guijarro-Lopez, Laura
- Yin, Yunxing
- Peng, Zuozhong
- Gomez, James E
- Fisher, Stewart
- Barros-Aguirre, David
- Hubbard, Brian K
- Serrano-Wu, Michael H
- Hung, Deborah T
Producer: 20190610
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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6.
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Screening of a Novel Fragment Library with Functional Complexity against Mycobacterium tuberculosis InhA. [electronic resource] by
- Prati, Federica
- Zuccotto, Fabio
- Fletcher, Daniel
- Convery, Maire A
- Fernandez-Menendez, Raquel
- Bates, Robert
- Encinas, Lourdes
- Zeng, Jingkun
- Chung, Chun-Wa
- De Dios Anton, Paco
- Mendoza-Losana, Alfonso
- Mackenzie, Claire
- Green, Simon R
- Huggett, Margaret
- Barros, David
- Wyatt, Paul G
- Ray, Peter C
Producer: 20190318
In:
ChemMedChem vol. 13
Availability: No items available.
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7.
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Identification of Selective Inhibitors of [electronic resource] by
- Harupa, Anke
- De Las Heras, Laura
- Colmenarejo, Gonzalo
- Lyons-Abbott, Sally
- Reers, Alexandra
- Caballero Hernandez, Iván
- Chung, Chun-Wa
- Charter, David
- Myler, Peter J
- Fernández-Menéndez, Raquel M
- Calderón, Félix
- Palomo, Sara
- Rodríguez, Beatriz
- Berlanga, Manuela
- Herreros-Avilés, Esperanza
- Staker, Bart L
- Fernández Álvaro, Elena
- Kaushansky, Alexis
Producer: 20200727
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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8.
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Exploring the SAR of the β-Ketoacyl-ACP Synthase Inhibitor GSK3011724A and Optimization around a Genotoxic Metabolite. [electronic resource] by
- Cunningham, Fraser
- Esquivias, Jorge
- Fernández-Menéndez, Raquel
- Pérez, Arancha
- Guardia, Ana
- Escribano, Jaime
- Rivero, Cristina
- Vimal, Mythily
- Cacho, Mónica
- de Dios-Antón, Paco
- Martínez-Martínez, María Santos
- Jiménez, Elena
- Huertas Valentín, Leticia
- Rebollo-López, María José
- López-Román, Eva María
- Sousa-Morcuende, Verónica
- Rullas, Joaquín
- Neu, Margaret
- Chung, Chun-Wa
- Bates, Robert H
Producer: 20210616
In:
ACS infectious diseases vol. 6
Availability: No items available.
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9.
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Antitubercular drugs for an old target: GSK693 as a promising InhA direct inhibitor. [electronic resource] by
- Martínez-Hoyos, María
- Perez-Herran, Esther
- Gulten, Gulcin
- Encinas, Lourdes
- Álvarez-Gómez, Daniel
- Alvarez, Emilio
- Ferrer-Bazaga, Santiago
- García-Pérez, Adolfo
- Ortega, Fátima
- Angulo-Barturen, Iñigo
- Rullas-Trincado, Joaquin
- Blanco Ruano, Delia
- Torres, Pedro
- Castañeda, Pablo
- Huss, Sophie
- Fernández Menéndez, Raquel
- González Del Valle, Silvia
- Ballell, Lluis
- Barros, David
- Modha, Sundip
- Dhar, Neeraj
- Signorino-Gelo, François
- McKinney, John D
- García-Bustos, Jose Francisco
- Lavandera, Jose Luis
- Sacchettini, James C
- Jimenez, M Soledad
- Martín-Casabona, Nuria
- Castro-Pichel, Julia
- Mendoza-Losana, Alfonso
Producer: 20170214
In:
EBioMedicine vol. 8
Availability: No items available.
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