Results
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Antiplasmodial and cytotoxicity evaluation of 3-functionalized 2-azetidinone derivatives. [electronic resource] by
- Singh, Pardeep
- Sachdeva, Shaveta
- Raj, Raghu
- Kumar, Vipan
- Mahajan, Mohinder P
- Nasser, Shereen
- Vivas, Livia
- Gut, Jiri
- Rosenthal, Phillip J
- Feng, Tzu-Shean
- Chibale, Kelly
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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4.
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Novel orally active antimalarial thiazoles. [electronic resource] by
- González Cabrera, Diego
- Douelle, Frederic
- Feng, Tzu-Shean
- Nchinda, Aloysius T
- Younis, Yassir
- White, Karen L
- Wu, Quoc
- Ryan, Eileen
- Burrows, Jeremy N
- Waterson, David
- Witty, Michael J
- Wittlin, Sergio
- Charman, Susan A
- Chibale, Kelly
Producer: 20120207
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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5.
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Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization. [electronic resource] by
- Soares de Melo, Candice
- Candice, Soares de Melo
- Feng, Tzu-Shean
- van der Westhuyzen, Renier
- Gessner, Richard K
- Street, Leslie J
- Morgans, Garreth L
- Warner, Digby F
- Moosa, Atica
- Naran, Krupa
- Lawrence, Nina
- Boshoff, Helena I M
- Barry, Clifton E
- Harris, C John
- Gordon, Richard
- Chibale, Kelly
Producer: 20160818
In:
Bioorganic & medicinal chemistry vol. 23
Availability: No items available.
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Structure-activity relationship studies of orally active antimalarial 3,5-substituted 2-aminopyridines. [electronic resource] by
- González Cabrera, Diego
- Douelle, Frederic
- Younis, Yassir
- Feng, Tzu-Shean
- Le Manach, Claire
- Nchinda, Aloysius T
- Street, Leslie J
- Scheurer, Christian
- Kamber, Jolanda
- White, Karen L
- Montagnat, Oliver D
- Ryan, Eileen
- Katneni, Kasiram
- Zabiulla, K Mohammed
- Joseph, Jayan T
- Bashyam, Sridevi
- Waterson, David
- Witty, Michael J
- Charman, Susan A
- Wittlin, Sergio
- Chibale, Kelly
Producer: 20130314
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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2,4-Diaminothienopyrimidines as orally active antimalarial agents. [electronic resource] by
- González Cabrera, Diego
- Le Manach, Claire
- Douelle, Frederic
- Younis, Yassir
- Feng, Tzu-Shean
- Paquet, Tanya
- Nchinda, Aloysius T
- Street, Leslie J
- Taylor, Dale
- de Kock, Carmen
- Wiesner, Lubbe
- Duffy, Sandra
- White, Karen L
- Zabiulla, K Mohammed
- Sambandan, Yuvaraj
- Bashyam, Sridevi
- Waterson, David
- Witty, Michael J
- Charman, Susan A
- Avery, Vicky M
- Wittlin, Sergio
- Chibale, Kelly
Producer: 20140415
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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8.
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3,5-Diaryl-2-aminopyridines as a novel class of orally active antimalarials demonstrating single dose cure in mice and clinical candidate potential. [electronic resource] by
- Younis, Yassir
- Douelle, Frederic
- Feng, Tzu-Shean
- González Cabrera, Diego
- Le Manach, Claire
- Nchinda, Aloysius T
- Duffy, Sandra
- White, Karen L
- Shackleford, David M
- Morizzi, Julia
- Mannila, Janne
- Katneni, Kasiram
- Bhamidipati, Ravi
- Zabiulla, K Mohammed
- Joseph, Jayan T
- Bashyam, Sridevi
- Waterson, David
- Witty, Michael J
- Hardick, David
- Wittlin, Sergio
- Avery, Vicky
- Charman, Susan A
- Chibale, Kelly
Producer: 20120831
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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9.
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2-Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure-Activity Relationships, Mechanism of Action and Absorption, Distribution, Metabolism, and Excretion Characterization. [electronic resource] by
- Murugesan, Dinakaran
- Ray, Peter C
- Bayliss, Tracy
- Prosser, Gareth A
- Harrison, Justin R
- Green, Kirsteen
- Soares de Melo, Candice
- Feng, Tzu-Shean
- Street, Leslie J
- Chibale, Kelly
- Warner, Digby F
- Mizrahi, Valerie
- Epemolu, Ola
- Scullion, Paul
- Ellis, Lucy
- Riley, Jennifer
- Shishikura, Yoko
- Ferguson, Liam
- Osuna-Cabello, Maria
- Read, Kevin D
- Green, Simon R
- Lamprecht, Dirk A
- Finin, Peter M
- Steyn, Adrie J C
- Ioerger, Thomas R
- Sacchettini, Jim
- Rhee, Kyu Y
- Arora, Kriti
- Barry, Clifton E
- Wyatt, Paul G
- Boshoff, Helena I M
Producer: 20190911
In:
ACS infectious diseases vol. 4
Availability: No items available.
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