Design, synthesis and evaluation against Mycobacterium tuberculosis of azole piperazine derivatives as dicyclotyrosine (cYY) mimics. [electronic resource]
Producer: 20180105Description: 161-176 p. digitalISSN:- 1464-3391
- Antitubercular Agents -- chemical synthesis
- Azoles -- chemistry
- Binding Sites -- drug effects
- Cytochrome P-450 Enzyme System -- chemistry
- Dipeptides -- chemistry
- Dose-Response Relationship, Drug
- Drug Design
- Ligands
- Microbial Sensitivity Tests
- Models, Molecular
- Molecular Structure
- Mycobacterium tuberculosis -- drug effects
- Peptides, Cyclic -- chemistry
- Piperazine
- Piperazines -- chemistry
- Structure-Activity Relationship
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Publication Type: Journal Article
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