Identification, Characterization, and Optimization of 2,8-Disubstituted-1,5-naphthyridines as Novel Plasmodium falciparum Phosphatidylinositol-4-kinase Inhibitors with in Vivo Efficacy in a Humanized Mouse Model of Malaria. [electronic resource]
Producer: 20190607Description: 5692-5703 p. digitalISSN:- 1520-4804
- 1-Phosphatidylinositol 4-Kinase -- antagonists & inhibitors
- Animals
- Antimalarials -- chemistry
- Disease Models, Animal
- Drug Design
- Enzyme Inhibitors -- chemistry
- Humans
- Malaria -- drug therapy
- Mice
- Models, Molecular
- Naphthyridines -- chemistry
- Plasmodium falciparum -- drug effects
- Protein Conformation
- Structure-Activity Relationship
- Tissue Distribution
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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