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A novel mode of protein kinase inhibition exploiting hydrophobic motifs of autoinhibited kinases: discovery of ATP-independent inhibitors of fibroblast growth factor receptor. [electronic resource] by
- Eathiraj, Sudharshan
- Palma, Rocio
- Hirschi, Marscha
- Volckova, Erika
- Nakuci, Enkeleda
- Castro, Jennifer
- Chen, Chang-Rung
- Chan, Thomas C K
- France, Dennis S
- Ashwell, Mark A
Producer: 20110805
In:
The Journal of biological chemistry vol. 286
Availability: No items available.
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12.
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Preclinical efficacy for a novel tyrosine kinase inhibitor, ArQule 531 against acute myeloid leukemia. [electronic resource] by
- Elgamal, Ola A
- Mehmood, Abeera
- Jeon, Jae Yoon
- Carmichael, Bridget
- Lehman, Amy
- Orwick, Shelley J
- Truxall, Jean
- Goettl, Virginia M
- Wasmuth, Ronni
- Tran, Minh
- Mitchell, Shaneice
- Lapalombella, Rosa
- Eathiraj, Sudharshan
- Schwartz, Brian
- Stegmaier, Kimberly
- Baker, Sharyn D
- Hertlein, Erin
- Byrd, John C
Producer: 20210126
In:
Journal of hematology & oncology vol. 13
Availability: No items available.
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13.
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Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor. [electronic resource] by
- Lapierre, Jean-Marc
- Eathiraj, Sudharshan
- Vensel, David
- Liu, Yanbin
- Bull, Cathy O
- Cornell-Kennon, Susan
- Iimura, Shin
- Kelleher, Eugene W
- Kizer, Darin E
- Koerner, Steffi
- Makhija, Sapna
- Matsuda, Akihisa
- Moussa, Magdi
- Namdev, Nivedita
- Savage, Ronald E
- Szwaya, Jeff
- Volckova, Erika
- Westlund, Neil
- Wu, Hui
- Schwartz, Brian
Producer: 20170529
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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14.
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The BTK Inhibitor ARQ 531 Targets Ibrutinib-Resistant CLL and Richter Transformation. [electronic resource] by
- Reiff, Sean D
- Mantel, Rose
- Smith, Lisa L
- Greene, J T
- Muhowski, Elizabeth M
- Fabian, Catherine A
- Goettl, Virginia M
- Tran, Minh
- Harrington, Bonnie K
- Rogers, Kerry A
- Awan, Farrukh T
- Maddocks, Kami
- Andritsos, Leslie
- Lehman, Amy M
- Sampath, Deepa
- Lapalombella, Rosa
- Eathiraj, Sudharshan
- Abbadessa, Giovanni
- Schwartz, Brian
- Johnson, Amy J
- Byrd, John C
- Woyach, Jennifer A
Producer: 20191024
In:
Cancer discovery vol. 8
Availability: No items available.
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15.
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Discovery and optimization of a series of 3-(3-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amines: orally bioavailable, selective, and potent ATP-independent Akt inhibitors. [electronic resource] by
- Ashwell, Mark A
- Lapierre, Jean-Marc
- Brassard, Christopher
- Bresciano, Karen
- Bull, Cathy
- Cornell-Kennon, Susan
- Eathiraj, Sudharshan
- France, Dennis S
- Hall, Terence
- Hill, Jason
- Kelleher, Eoin
- Khanapurkar, Sampada
- Kizer, Darin
- Koerner, Steffi
- Link, Jeff
- Liu, Yanbin
- Makhija, Sapna
- Moussa, Magdi
- Namdev, Nivedita
- Nguyen, Khanh
- Nicewonger, Robert
- Palma, Rocio
- Szwaya, Jeff
- Tandon, Manish
- Uppalapati, Uma
- Vensel, David
- Volak, Laurie P
- Volckova, Erika
- Westlund, Neil
- Wu, Hui
- Yang, Rui-Yang
- Chan, Thomas C K
Producer: 20121001
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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