Results
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1.
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Determining direct binders of the Androgen Receptor using a high-throughput Cellular Thermal Shift Assay. [electronic resource] by
- Shaw, Joseph
- Leveridge, Mathew
- Norling, Charlotta
- Karén, Jakob
- Molina, Daniel Martinez
- O'Neill, Daniel
- Dowling, James E
- Davey, Paul
- Cowan, Suzanna
- Dabrowski, Michael
- Main, Martin
- Gianni, Davide
Producer: 20181116
In:
Scientific reports vol. 8
Availability: No items available.
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2.
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Synthesis of [1,2,4]triazolo[1,5-a]pyrazines as adenosine A2A receptor antagonists. [electronic resource] by
- Dowling, James E
- Vessels, Jeffrey T
- Haque, Serajul
- Chang, He Xi
- van Vloten, Kurt
- Kumaravel, Gnanasambandam
- Engber, Thomas
- Jin, Xiaowei
- Phadke, Deepali
- Wang, Joy
- Ayyub, Eman
- Petter, Russell C
Producer: 20051223
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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3.
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Potent and orally bioavailable 8-bicyclo[2.2.2]octylxanthines as adenosine A1 receptor antagonists. [electronic resource] by
- Kiesman, William F
- Zhao, Jin
- Conlon, Patrick R
- Dowling, James E
- Petter, Russell C
- Lutterodt, Frank
- Jin, Xiaowei
- Smits, Glenn
- Fure, Mary
- Jayaraj, Andrew
- Kim, John
- Sullivan, Gail
- Linden, Joel
Producer: 20070215
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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4.
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Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo. [electronic resource] by
- Dowling, James E
- Alimzhanov, Marat
- Bao, Larry
- Chuaqui, Claudio
- Denz, Christopher R
- Jenkins, Emma
- Larsen, Nicholas A
- Lyne, Paul D
- Pontz, Timothy
- Ye, Qing
- Holdgate, Geoff A
- Snow, Lindsay
- O'Connell, Nichole
- Ferguson, Andrew D
Producer: 20160317
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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5.
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Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors. [electronic resource] by
- McCoull, William
- Hennessy, Edward J
- Blades, Kevin
- Chuaqui, Claudio
- Dowling, James E
- Ferguson, Andrew D
- Goldberg, Frederick W
- Howe, Nicholas
- Jones, Christopher R
- Kemmitt, Paul D
- Lamont, Gillian
- Varnes, Jeffrey G
- Ward, Richard A
- Yang, Bin
Publication details: ACS medicinal chemistry letters Dec 2016
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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6.
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Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening. [electronic resource] by
- Yang, Bin
- Lamb, Michelle L
- Zhang, Tao
- Hennessy, Edward J
- Grewal, Gurmit
- Sha, Li
- Zambrowski, Mark
- Block, Michael H
- Dowling, James E
- Su, Nancy
- Wu, Jiaquan
- Deegan, Tracy
- Mikule, Keith
- Wang, Wenxian
- Kaspera, Rüdiger
- Chuaqui, Claudio
- Chen, Huawei
Producer: 20150226
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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7.
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Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases. [electronic resource] by
- Dakin, Les A
- Block, Michael H
- Chen, Huawei
- Code, Erin
- Dowling, James E
- Feng, Xiaomei
- Ferguson, Andrew D
- Green, Isabelle
- Hird, Alexander W
- Howard, Tina
- Keeton, Erika K
- Lamb, Michelle L
- Lyne, Paul D
- Pollard, Hannah
- Read, Jon
- Wu, Allan J
- Zhang, Tao
- Zheng, Xiaolan
Producer: 20130104
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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8.
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Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo. [electronic resource] by
- Dowling, James E
- Alimzhanov, Marat
- Bao, Larry
- Block, Michael H
- Chuaqui, Claudio
- Cooke, Emma L
- Denz, Christopher R
- Hird, Alex
- Huang, Shan
- Larsen, Nicholas A
- Peng, Bo
- Pontz, Timothy W
- Rivard-Costa, Caroline
- Saeh, Jamal Carlos
- Thakur, Kumar
- Ye, Qing
- Zhang, Tao
- Lyne, Paul D
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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9.
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Target Deconvolution Efforts on Wnt Pathway Screen Reveal Dual Modulation of Oxidative Phosphorylation and SERCA2. [electronic resource] by
- Casás-Selves, Matias
- Zhang, Andrew X
- Dowling, James E
- Hallén, Stefan
- Kawatkar, Aarti
- Pace, Nicholas J
- Denz, Christopher R
- Pontz, Timothy
- Garahdaghi, Farzin
- Cao, Qing
- Sabirsh, Alan
- Thakur, Kumar
- O'Connell, Nichole
- Hu, Jun
- Cornella-Taracido, Iván
- Weerapana, Eranthie
- Zinda, Michael
- Goodnow, Robert A
- Castaldi, M Paola
Producer: 20170929
In:
ChemMedChem vol. 12
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10.
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Discovery of 2,6-disubstituted pyrazine derivatives as inhibitors of CK2 and PIM kinases. [electronic resource] by
- Gingipalli, Lakshmaiah
- Block, Michael H
- Bao, Larry
- Cooke, Emma
- Dakin, Les A
- Denz, Christopher R
- Ferguson, Andrew D
- Johannes, Jeffrey W
- Larsen, Nicholas A
- Lyne, Paul D
- Pontz, Timothy W
- Wang, Tao
- Wu, Xiaoyun
- Wu, Allan
- Zhang, Hai-Jun
- Zheng, Xiaolan
- Dowling, James E
- Lamb, Michelle L
Producer: 20190227
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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11.
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Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization. [electronic resource] by
- Dowling, James E
- Chuaqui, Claudio
- Pontz, Timothy W
- Lyne, Paul D
- Larsen, Nicholas A
- Block, Michael H
- Chen, Huawei
- Su, Nancy
- Wu, Allan
- Russell, Daniel
- Pollard, Hannah
- Lee, John W
- Peng, Bo
- Thakur, Kumar
- Ye, Qing
- Zhang, Tao
- Brassil, Patrick
- Racicot, Vicki
- Bao, Larry
- Denz, Christopher R
- Cooke, Emma
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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12.
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Improving HIV Surveillance Data by Using the ATra Black Box System to Assist Regional Deduplication Activities. [electronic resource] by
- Ocampo, Joanne Michelle F
- Hamp, Auntré
- Rhodes, Anne
- Smart, J C
- Pemmaraju, Raghu
- Poschman, Karalee
- Hess, Kristen L
- Bhattacharjee, Reshma
- Flynn, Colin
- Anderson, Bridget J
- Dowling, James E
- Maccormack, Fred
- Doshi, Rupali
- Lum, Garret
- Maddox, Lorene
- Moncur, Brenda
- Barnhart, John E
- Maxwell, Jason
- Aurand, Sahithi Boggavarapu
- Hogan, Vicki
- Wills, David
- Prowell, Stacy
- Kassaye, Seble G
- Karn, Helen E
- Laffoon, Benjamin T
- Collmann, Jeff
Producer: 20200619
In:
Journal of acquired immune deficiency syndromes (1999) vol. 82 Suppl 1
Availability: No items available.
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13.
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Discovery and Optimization of Pyrrolopyrimidine Inhibitors of Interleukin-1 Receptor Associated Kinase 4 (IRAK4) for the Treatment of Mutant MYD88 [electronic resource] by
- Scott, James S
- Degorce, Sébastien L
- Anjum, Rana
- Culshaw, Janet
- Davies, Robert D M
- Davies, Nichola L
- Dillman, Keith S
- Dowling, James E
- Drew, Lisa
- Ferguson, Andrew D
- Groombridge, Sam D
- Halsall, Christopher T
- Hudson, Julian A
- Lamont, Scott
- Lindsay, Nicola A
- Marden, Stacey K
- Mayo, Michele F
- Pease, J Elizabeth
- Perkins, David R
- Pink, Jennifer H
- Robb, Graeme R
- Rosen, Alan
- Shen, Minhui
- McWhirter, Claire
- Wu, Dedong
Producer: 20190401
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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