A novel selective peroxisome proliferator-activator receptor-gamma modulator-SPPARgammaM5 improves insulin sensitivity with diminished adverse cardiovascular effects. [electronic resource]
Producer: 20080710Description: 192-201 p. digitalISSN:- 0014-2999
- 3T3-L1 Cells
- Acetates -- adverse effects
- Adipose Tissue, White -- drug effects
- Animals
- COS Cells
- Cardiomegaly -- chemically induced
- Cardiovascular Diseases -- chemically induced
- Chlorocebus aethiops
- Diabetes Mellitus, Type 2 -- drug therapy
- Disease Models, Animal
- Dose-Response Relationship, Drug
- Drug Partial Agonism
- Gene Expression Profiling
- Gene Expression Regulation -- drug effects
- Hemodilution
- Humans
- Hypoglycemic Agents -- adverse effects
- Indoles -- adverse effects
- Insulin Resistance -- genetics
- Male
- Mice
- Mice, Inbred Strains
- PPAR alpha -- drug effects
- PPAR delta -- drug effects
- PPAR gamma -- drug effects
- Propionates -- adverse effects
- Protein Binding
- Rats
- Rats, Zucker
- Rosiglitazone
- Thiazolidinediones -- adverse effects
- Transcriptional Activation -- drug effects
- Transfection
- Water-Electrolyte Balance -- drug effects
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Publication Type: Comparative Study; Journal Article
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