Design of (quinolin-4-ylthio)carboxylic acids as new Escherichia coli DNA gyrase B inhibitors: machine learning studies, molecular docking, synthesis and biological testing. [electronic resource]
Producer: 20210106Description: 107224 p. digitalISSN:- 1476-928X
- Anti-Bacterial Agents -- chemical synthesis
- Computational Biology
- DNA Gyrase -- metabolism
- Drug Design
- Escherichia coli -- drug effects
- Machine Learning
- Microbial Sensitivity Tests
- Molecular Docking Simulation
- Molecular Structure
- Quantitative Structure-Activity Relationship
- Quinolines -- chemical synthesis
- Topoisomerase II Inhibitors -- chemical synthesis
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Publication Type: Journal Article
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