High-throughput screening for novel inhibitors of Neisseria gonorrhoeae penicillin-binding protein 2. [electronic resource]
Producer: 20130422Description: e44918 p. digitalISSN:- 1932-6203
- Anti-Bacterial Agents -- chemistry
- Bacterial Proteins -- antagonists & inhibitors
- Boron Compounds -- analysis
- Catalytic Domain
- Cephalosporins -- pharmacology
- Dose-Response Relationship, Drug
- Fluorescence Polarization
- High-Throughput Screening Assays
- Microbial Sensitivity Tests
- Molecular Docking Simulation
- Neisseria gonorrhoeae -- drug effects
- Penicillin-Binding Proteins -- antagonists & inhibitors
- Penicillins -- analysis
- Protein Binding
- Recombinant Proteins -- antagonists & inhibitors
- Small Molecule Libraries -- chemistry
- beta-Lactam Resistance -- drug effects
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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