Evaluation of the in vivo receptor occupancy for the behavioral effects of cannabinoids using a radiolabeled cannabinoid receptor agonist, R-[125/131I]AM2233. [electronic resource]
Producer: 20060810Description: 93-101 p. digitalISSN:- 0887-4476
- Animals
- Behavior, Animal -- drug effects
- Benzoxazines
- Binding Sites -- drug effects
- Binding, Competitive -- drug effects
- Brain -- anatomy & histology
- Cannabinoids -- metabolism
- Dose-Response Relationship, Drug
- Drug Interactions
- Indoles -- metabolism
- Iodine Radioisotopes -- metabolism
- Male
- Mice
- Morpholines -- metabolism
- Motor Activity -- drug effects
- Naphthalenes -- metabolism
- Neurons -- drug effects
- Piperidines -- metabolism
- Protein Conformation -- drug effects
- Pyrazoles -- pharmacology
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptor, Cannabinoid, CB1 -- agonists
- Rimonabant
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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