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The chimpanzee (Pan troglodytes) as a pharmacokinetic model for selection of drug candidates: model characterization and application. [electronic resource] by
- Wong, Harvey
- Grossman, Scott J
- Bai, Stephen A
- Diamond, Sharon
- Wright, Matthew R
- Grace, James E
- Qian, Mingxin
- He, Kan
- Yeleswaram, Krishnaswamy
- Christ, David D
Producer: 20050408
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 32
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7.
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Roles of UGT, P450, and Gut Microbiota in the Metabolism of Epacadostat in Humans. [electronic resource] by
- Boer, Jason
- Young-Sciame, Ruth
- Lee, Fiona
- Bowman, Kevin J
- Yang, Xiaoqing
- Shi, Jack G
- Nedza, Frank M
- Frietze, William
- Galya, Laurine
- Combs, Andrew P
- Yeleswaram, Swamy
- Diamond, Sharon
Producer: 20180206
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 44
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8.
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Interaction of ritonavir on tissue distribution of a [(14)c]L-valinamide, a potent human immunodeficiency virus-1 protease inhibitor, in rats using quantitative whole-body autoradiography. [electronic resource] by
- Solon, Eric G
- Balani, Suresh K
- Luo, Gang
- Yang, Tian J
- Haines, Paula J
- Wang, Lifei
- Demond, Tonya
- Diamond, Sharon
- Christ, David D
- Gan, Liang-Shang
- Lee, Frank W
Producer: 20030507
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 30
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9.
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Species-specific, P450- and sulfotransferase-mediated novel ring contraction of a naphthyridine-N-oxide compound in cynomolgus monkey. [electronic resource] by
- Daniels, J Scott
- Espina, Robert
- Cao, Kevin
- Yuan, Haodan
- Lin, Jianrong
- Diamond, Sharon
- Johnson, Barry
- Rodgers, James
- Prakash, Shimoga
- Unger, Steve
- Christ, David
- Miwa, Gerald
- Gan, Liang-Shang
- Mutlib, Abdul
Producer: 20080116
In:
Chemical research in toxicology vol. 20
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10.
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The Janus kinase 2 inhibitor fedratinib inhibits thiamine uptake: a putative mechanism for the onset of Wernicke's encephalopathy. [electronic resource] by
- Zhang, Qiang
- Zhang, Yan
- Diamond, Sharon
- Boer, Jason
- Harris, Jennifer J
- Li, Yu
- Rupar, Mark
- Behshad, Elham
- Gardiner, Christine
- Collier, Paul
- Liu, Phillip
- Burn, Timothy
- Wynn, Richard
- Hollis, Gregory
- Yeleswaram, Swamy
Producer: 20150526
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 42
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11.
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Metabolism, excretion, and pharmacokinetics of [14C]INCB018424, a selective Janus tyrosine kinase 1/2 inhibitor, in humans. [electronic resource] by
- Shilling, Adam D
- Nedza, Frank M
- Emm, Thomas
- Diamond, Sharon
- McKeever, Edward
- Punwani, Naresh
- Williams, William
- Arvanitis, Argyrios
- Galya, Laurine G
- Li, Mei
- Shepard, Stacey
- Rodgers, James
- Yue, Tai-Yuen
- Yeleswaram, Swamy
Producer: 20110310
In:
Drug metabolism and disposition: the biological fate of chemicals vol. 38
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12.
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A novel kinase inhibitor, INCB28060, blocks c-MET-dependent signaling, neoplastic activities, and cross-talk with EGFR and HER-3. [electronic resource] by
- Liu, Xiangdong
- Wang, Qian
- Yang, Gengjie
- Marando, Cindy
- Koblish, Holly K
- Hall, Leslie M
- Fridman, Jordan S
- Behshad, Elham
- Wynn, Richard
- Li, Yu
- Boer, Jason
- Diamond, Sharon
- He, Chunhong
- Xu, Meizhong
- Zhuo, Jincong
- Yao, Wenqing
- Newton, Robert C
- Scherle, Peggy A
Producer: 20120325
In:
Clinical cancer research : an official journal of the American Association for Cancer Research vol. 17
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13.
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DPC 817: a cytidine nucleoside analog with activity against zidovudine- and lamivudine-resistant viral variants. [electronic resource] by
- Schinazi, Raymond F
- Mellors, John
- Bazmi, Holly
- Diamond, Sharon
- Garber, Sena
- Gallagher, Karen
- Geleziunas, Romas
- Klabe, Ron
- Pierce, Michael
- Rayner, Marlene
- Wu, Jing-Tao
- Zhang, Hangchun
- Hammond, Jennifer
- Bacheler, Lee
- Manion, Douglas J
- Otto, Michael J
- Stuyver, Lieven
- Trainor, George
- Liotta, Dennis C
- Erickson-Viitanen, Susan
Producer: 20020806
In:
Antimicrobial agents and chemotherapy vol. 46
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14.
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Discovery and pharmacological characterization of a novel rodent-active CCR2 antagonist, INCB3344. [electronic resource] by
- Brodmerkel, Carrie M
- Huber, Reid
- Covington, Maryanne
- Diamond, Sharon
- Hall, Leslie
- Collins, Robert
- Leffet, Lynn
- Gallagher, Karen
- Feldman, Patricia
- Collier, Paul
- Stow, Mark
- Gu, Xiaomei
- Baribaud, Frederic
- Shin, Niu
- Thomas, Beth
- Burn, Tim
- Hollis, Greg
- Yeleswaram, Swamy
- Solomon, Kim
- Friedman, Steve
- Wang, Anlai
- Xue, Chu Biao
- Newton, Robert C
- Scherle, Peggy
- Vaddi, Kris
Producer: 20051213
In:
Journal of immunology (Baltimore, Md. : 1950) vol. 175
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15.
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Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2. [electronic resource] by
- Xue, Chu-Biao
- Wang, Anlai
- Meloni, David
- Zhang, Ke
- Kong, Ling
- Feng, Hao
- Glenn, Joseph
- Huang, Taisheng
- Zhang, Yingxin
- Cao, Ganfeng
- Anand, Rajan
- Zheng, Changsheng
- Xia, Michael
- Han, Qi
- Robinson, D J
- Storace, Lou
- Shao, Lixin
- Li, Mei
- Brodmerkel, Carrie M
- Covington, Maryanne
- Scherle, Peggy
- Diamond, Sharon
- Yeleswaram, Swamy
- Vaddi, Kris
- Newton, Robert
- Hollis, Greg
- Friedman, Steven
- Metcalf, Brian
Producer: 20110314
In:
Bioorganic & medicinal chemistry letters vol. 20
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16.
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Preclinical characterization of INCB053914, a novel pan-PIM kinase inhibitor, alone and in combination with anticancer agents, in models of hematologic malignancies. [electronic resource] by
- Koblish, Holly
- Li, Yun-Long
- Shin, Niu
- Hall, Leslie
- Wang, Qian
- Wang, Kathy
- Covington, Maryanne
- Marando, Cindy
- Bowman, Kevin
- Boer, Jason
- Burke, Krista
- Wynn, Richard
- Margulis, Alex
- Reuther, Gary W
- Lambert, Que T
- Dostalik Roman, Valerie
- Zhang, Ke
- Feng, Hao
- Xue, Chu-Biao
- Diamond, Sharon
- Hollis, Greg
- Yeleswaram, Swamy
- Yao, Wenqing
- Huber, Reid
- Vaddi, Kris
- Scherle, Peggy
Producer: 20181231
In:
PloS one vol. 13
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17.
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INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models. [electronic resource] by
- Liu, Phillip C C
- Koblish, Holly
- Wu, Liangxing
- Bowman, Kevin
- Diamond, Sharon
- DiMatteo, Darlise
- Zhang, Yue
- Hansbury, Michael
- Rupar, Mark
- Wen, Xiaoming
- Collier, Paul
- Feldman, Patricia
- Klabe, Ronald
- Burke, Krista A
- Soloviev, Maxim
- Gardiner, Christine
- He, Xin
- Volgina, Alla
- Covington, Maryanne
- Ruggeri, Bruce
- Wynn, Richard
- Burn, Timothy C
- Scherle, Peggy
- Yeleswaram, Swamy
- Yao, Wenqing
- Huber, Reid
- Hollis, Gregory
Producer: 20200724
In:
PloS one vol. 15
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18.
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Discovery of INCB10820/PF-4178903, a potent, selective, and orally bioavailable dual CCR2 and CCR5 antagonist. [electronic resource] by
- Zheng, Changsheng
- Cao, Ganfeng
- Xia, Michael
- Feng, Hao
- Glenn, Joseph
- Anand, Rajan
- Zhang, Ke
- Huang, Taisheng
- Wang, Anlai
- Kong, Ling
- Li, Mei
- Galya, Laurine
- Hughes, Robert O
- Devraj, Rajesh
- Morton, Phillip A
- Rogier, D Joseph
- Covington, Maryanne
- Baribaud, Fred
- Shin, Niu
- Scherle, Peggy
- Diamond, Sharon
- Yeleswaram, Swamy
- Vaddi, Kris
- Newton, Robert
- Hollis, Greg
- Friedman, Steven
- Metcalf, Brian
- Xue, Chu-Biao
Producer: 20110614
In:
Bioorganic & medicinal chemistry letters vol. 21
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19.
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Discovery of INCB9471, a Potent, Selective, and Orally Bioavailable CCR5 Antagonist with Potent Anti-HIV-1 Activity. [electronic resource] by
- Xue, Chu-Biao
- Chen, Lihua
- Cao, Ganfeng
- Zhang, Ke
- Wang, Anlai
- Meloni, David
- Glenn, Joseph
- Anand, Rajan
- Xia, Michael
- Kong, Ling
- Huang, Taisheng
- Feng, Hao
- Zheng, Changsheng
- Li, Mei
- Galya, Laurine
- Zhou, Jiacheng
- Shin, Niu
- Baribaud, Fredric
- Solomon, Kim
- Scherle, Peggy
- Zhao, Bitao
- Diamond, Sharon
- Emm, Tom
- Keller, Douglas
- Contel, Nancy
- Yeleswaram, Swamy
- Vaddi, Kris
- Hollis, Gregory
- Newton, Robert
- Friedman, Steven
- Metcalf, Brian
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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20.
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INCB040093 Is a Novel PI3K [electronic resource] by
- Shin, Niu
- Li, Yun-Long
- Mei, Song
- Wang, Kathy He
- Hall, Leslie
- Katiyar, Kamna
- Wang, Qian
- Yang, Gengjie
- Rumberger, Beth
- Leffet, Lynn
- He, Xin
- Rupar, Mark
- Bowman, Kevin
- Favata, Margaret
- Li, Jun
- Liu, Mike
- Li, Yanlong
- Covington, Maryanne
- Koblish, Holly
- Soloviev, Maxim
- Shuey, Dana
- Burn, Timothy
- Diamond, Sharon
- Fridman, Jordan
- Combs, Andrew
- Yao, Wenqing
- Yeleswaram, Swamy
- Hollis, Gregory
- Vaddi, Kris
- Huber, Reid
- Newton, Robert
- Scherle, Peggy
Producer: 20171227
In:
The Journal of pharmacology and experimental therapeutics vol. 364
Availability: No items available.
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