Results
|
1.
|
ARRY-520, a novel KSP inhibitor with potent activity in hematological and taxane-resistant tumor models. [electronic resource] by
- Woessner, Richard
- Tunquist, Brian
- Lemieux, Christine
- Chlipala, Elizabeth
- Jackinsky, Steve
- Dewolf, Walter
- Voegtli, Walter
- Cox, April
- Rana, Sumeet
- Lee, Patrice
- Walker, Duncan
Producer: 20100126
In:
Anticancer research vol. 29
Availability: No items available.
|
|
2.
|
The kinetic model of the shikimate pathway as a tool to optimize enzyme assays for high-throughput screening. [electronic resource] by
- Noble, Michael
- Sinha, Yugesh
- Kolupaev, Aleksey
- Demin, Oleg
- Earnshaw, David
- Tobin, Frank
- West, Joshua
- Martin, John D
- Qiu, Chunyan
- Liu, Wu-Schyong
- DeWolf, Walter E
- Tew, David
- Goryanin, Igor I
Producer: 20061208
In:
Biotechnology and bioengineering vol. 95
Availability: No items available.
|
|
3.
|
Identification of a new class of glucokinase activators through structure-based design. [electronic resource] by
- Hinklin, Ronald J
- Boyd, Steven A
- Chicarelli, Mark J
- Condroski, Kevin R
- DeWolf, Walter E
- Lee, Patrice A
- Lee, Waiman
- Singh, Ajay
- Thomas, Laurie
- Voegtli, Walter C
- Williams, Lance
- Aicher, Thomas D
Producer: 20131223
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
|
|
4.
|
Characterization of Streptococcus pneumoniae enoyl-(acyl-carrier protein) reductase (FabK). [electronic resource] by
- Marrakchi, Hedia
- Dewolf, Walter E
- Quinn, Chad
- West, Joshua
- Polizzi, Brian J
- So, Chi Y
- Holmes, David J
- Reed, Shannon L
- Heath, Richard J
- Payne, David J
- Rock, Charles O
- Wallis, Nicola G
Producer: 20030423
In:
The Biochemical journal vol. 370
Availability: No items available.
|
|
5.
|
Characterization of a novel glucokinase activator in rat and mouse models. [electronic resource] by
- Lu, Min
- Li, Pingping
- Bandyopadhyay, Gautam
- Lagakos, William
- Dewolf, Walter E
- Alford, Taylor
- Chicarelli, Mark Joseph
- Williams, Lance
- Anderson, Deborah A
- Baer, Brian R
- McVean, Maralee
- Conn, Marion
- Véniant, Murielle M
- Coward, Peter
Producer: 20150106
In:
PloS one vol. 9
Availability: No items available.
|
|
6.
|
Discovery of 2-pyridylureas as glucokinase activators. [electronic resource] by
- Hinklin, Ronald J
- Aicher, Thomas D
- Anderson, Deborah A
- Baer, Brian R
- Boyd, Steven A
- Condroski, Kevin R
- DeWolf, Walter E
- Kraser, Christopher F
- McVean, Maralee
- Rhodes, Susan P
- Sturgis, Hillary L
- Voegtli, Walter C
- Williams, Lance
- Houze, Jonathan B
Producer: 20141218
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
|
|
7.
|
Defining and combating the mechanisms of triclosan resistance in clinical isolates of Staphylococcus aureus. [electronic resource] by
- Fan, Frank
- Yan, Kang
- Wallis, Nicola G
- Reed, Shannon
- Moore, Terrance D
- Rittenhouse, Stephen F
- DeWolf, Walter E
- Huang, Jianzhong
- McDevitt, Damien
- Miller, William H
- Seefeld, Mark A
- Newlander, Kenneth A
- Jakas, Dalia R
- Head, Martha S
- Payne, David J
Producer: 20030324
In:
Antimicrobial agents and chemotherapy vol. 46
Availability: No items available.
|
|
8.
|
Prodrug thiamine analogs as inhibitors of the enzyme transketolase. [electronic resource] by
- Le Huerou, Yvan
- Gunawardana, Indrani
- Thomas, Allen A
- Boyd, Steven A
- de Meese, Jason
- Dewolf, Walter
- Gonzales, Steven S
- Han, May
- Hayter, Laura
- Kaplan, Tomas
- Lemieux, Christine
- Lee, Patrice
- Pheneger, Jed
- Poch, Gregory
- Romoff, Todd T
- Sullivan, Francis
- Weiler, Solly
- Wright, S Kirk
- Lin, Jie
Producer: 20080527
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
|
|
9.
|
5-Alkyl-2-urea-Substituted Pyridines: Identification of Efficacious Glucokinase Activators with Improved Properties. [electronic resource] by
- Kohn, Todd J
- Du, Xiaohui
- Lai, SuJen
- Xiong, YuMei
- Komorowski, Renee
- Veniant, Murielle
- Fu, Zice
- Jiao, Xianyun
- Pattaropong, Vatee
- Chow, David
- Cardozo, Mario
- Jin, Lixia
- Conn, Marion
- DeWolf, Walter E
- Kraser, Christopher F
- Hinklin, Ronald J
- Boys, Mark L
- Medina, Julio C
- Houze, Jonathan
- Dransfield, Paul
- Coward, Peter
Producer: 20160720
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
|
|
10.
|
Non-charged thiamine analogs as inhibitors of enzyme transketolase. [electronic resource] by
- Thomas, Allen A
- De Meese, J
- Le Huerou, Y
- Boyd, Steven A
- Romoff, Todd T
- Gonzales, Steven S
- Gunawardana, Indrani
- Kaplan, Tomas
- Sullivan, Francis
- Condroski, Kevin
- Lyssikatos, Joseph P
- Aicher, Thomas D
- Ballard, Josh
- Bernat, Bryan
- DeWolf, Walter
- Han, May
- Lemieux, Christine
- Smith, Darin
- Weiler, Solly
- Wright, S Kirk
- Vigers, Guy
- Brandhuber, Barb
Producer: 20080527
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
|
|
11.
|
Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator. [electronic resource] by
- Hinklin, Ronald J
- Baer, Brian R
- Boyd, Steven A
- Chicarelli, Mark D
- Condroski, Kevin R
- DeWolf, Walter E
- Fischer, John
- Frank, Michele
- Hingorani, Gary P
- Lee, Patrice A
- Neitzel, Nickolas A
- Pratt, Scott A
- Singh, Ajay
- Sullivan, Francis X
- Turner, Timothy
- Voegtli, Walter C
- Wallace, Eli M
- Williams, Lance
- Aicher, Thomas D
Producer: 20210120
In:
Bioorganic & medicinal chemistry vol. 28
Availability: No items available.
|
|
12.
|
Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394. [electronic resource] by
- Dransfield, Paul J
- Pattaropong, Vatee
- Lai, Sujen
- Fu, Zice
- Kohn, Todd J
- Du, Xiaohui
- Cheng, Alan
- Xiong, Yumei
- Komorowski, Renee
- Jin, Lixia
- Conn, Marion
- Tien, Eric
- DeWolf, Walter E
- Hinklin, Ronald J
- Aicher, Thomas D
- Kraser, Christopher F
- Boyd, Steven A
- Voegtli, Walter C
- Condroski, Kevin R
- Veniant-Ellison, Murielle
- Medina, Julio C
- Houze, Jonathan
- Coward, Peter
Producer: 20160720
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
|
|
13.
|
Indole naphthyridinones as inhibitors of bacterial enoyl-ACP reductases FabI and FabK. [electronic resource] by
- Seefeld, Mark A
- Miller, William H
- Newlander, Kenneth A
- Burgess, Walter J
- DeWolf, Walter E
- Elkins, Patricia A
- Head, Martha S
- Jakas, Dalia R
- Janson, Cheryl A
- Keller, Paul M
- Manley, Peter J
- Moore, Terrance D
- Payne, David J
- Pearson, Stewart
- Polizzi, Brian J
- Qiu, Xiayang
- Rittenhouse, Stephen F
- Uzinskas, Irene N
- Wallis, Nicola G
- Huffman, William F
Producer: 20030527
In:
Journal of medicinal chemistry vol. 46
Availability: No items available.
|
|
14.
|
Discovery of aminopyridine-based inhibitors of bacterial enoyl-ACP reductase (FabI). [electronic resource] by
- Miller, William H
- Seefeld, Mark A
- Newlander, Kenneth A
- Uzinskas, Irene N
- Burgess, Walter J
- Heerding, Dirk A
- Yuan, Catherine C K
- Head, Martha S
- Payne, David J
- Rittenhouse, Stephen F
- Moore, Terrance D
- Pearson, Stewart C
- Berry, Valerie
- DeWolf, Walter E
- Keller, Paul M
- Polizzi, Brian J
- Qiu, Xiayang
- Janson, Cheryl A
- Huffman, William F
Producer: 20020812
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
|
|
15.
|
Synthesis, in vitro and in vivo activity of thiamine antagonist transketolase inhibitors. [electronic resource] by
- Thomas, Allen A
- Le Huerou, Y
- De Meese, J
- Gunawardana, Indrani
- Kaplan, Tomas
- Romoff, Todd T
- Gonzales, Stephen S
- Condroski, Kevin
- Boyd, Steven A
- Ballard, Josh
- Bernat, Bryan
- DeWolf, Walter
- Han, May
- Lee, Patrice
- Lemieux, Christine
- Pedersen, Robin
- Pheneger, Jed
- Poch, Greg
- Smith, Darin
- Sullivan, Francis
- Weiler, Solly
- Wright, S Kirk
- Lin, Jie
- Brandhuber, Barb
- Vigers, Guy
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
|
|
16.
|
C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators. [electronic resource] by
- Du, Xiaohui
- Hinklin, Ronald J
- Xiong, Yumei
- Dransfield, Paul
- Park, Jaehyeon
- Kohn, Todd J
- Pattaropong, Vatee
- Lai, SuJen
- Fu, Zice
- Jiao, Xianyun
- Chow, David
- Jin, Lixia
- Davda, Jasmine
- Veniant, Murielle M
- Anderson, Deborah A
- Baer, Brian R
- Bencsik, Josef R
- Boyd, Steven A
- Chicarelli, Mark Joseph
- Mohr, Peter J
- Wang, Bin
- Condroski, Kevin R
- DeWolf, Walter E
- Conn, Marion
- Tran, Thanhvien
- Yang, Jerry
- Aicher, Thomas D
- Medina, Julio C
- Coward, Peter
- Houze, Jonathan B
Producer: 20141217
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
|
|
17.
|
Discovery of a novel and potent class of FabI-directed antibacterial agents. [electronic resource] by
- Payne, David J
- Miller, William H
- Berry, Valerie
- Brosky, John
- Burgess, Walter J
- Chen, Emile
- DeWolf, Walter E
- Fosberry, Andrew P
- Greenwood, Rebecca
- Head, Martha S
- Heerding, Dirk A
- Janson, Cheryl A
- Jaworski, Deborah D
- Keller, Paul M
- Manley, Peter J
- Moore, Terrance D
- Newlander, Kenneth A
- Pearson, Stewart
- Polizzi, Brian J
- Qiu, Xiayang
- Rittenhouse, Stephen F
- Slater-Radosti, Courtney
- Salyers, Kevin L
- Seefeld, Mark A
- Smyth, Martin G
- Takata, Dennis T
- Uzinskas, Irene N
- Vaidya, Kalindi
- Wallis, Nicola G
- Winram, Scott B
- Yuan, Catherine C K
- Huffman, William F
Producer: 20030225
In:
Antimicrobial agents and chemotherapy vol. 46
Availability: No items available.
|
|
18.
|
A Next-Generation TRK Kinase Inhibitor Overcomes Acquired Resistance to Prior TRK Kinase Inhibition in Patients with TRK Fusion-Positive Solid Tumors. [electronic resource] by
- Drilon, Alexander
- Nagasubramanian, Ramamoorthy
- Blake, James F
- Ku, Nora
- Tuch, Brian B
- Ebata, Kevin
- Smith, Steve
- Lauriault, Veronique
- Kolakowski, Gabrielle R
- Brandhuber, Barbara J
- Larsen, Paul D
- Bouhana, Karyn S
- Winski, Shannon L
- Hamor, Robyn
- Wu, Wen-I
- Parker, Andrew
- Morales, Tony H
- Sullivan, Francis X
- DeWolf, Walter E
- Wollenberg, Lance A
- Gordon, Paul R
- Douglas-Lindsay, Dorothea N
- Scaltriti, Maurizio
- Benayed, Ryma
- Raj, Sandeep
- Hanusch, Bethany
- Schram, Alison M
- Jonsson, Philip
- Berger, Michael F
- Hechtman, Jaclyn F
- Taylor, Barry S
- Andrews, Steve
- Rothenberg, S Michael
- Hyman, David M
Producer: 20180629
In:
Cancer discovery vol. 7
Availability: No items available.
|