Results
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The discovery and synthesis of highly potent subtype selective phosphodiesterase 4D inhibitors. [electronic resource] by
- Aspiotis, Renee
- Deschênes, Denis
- Dubé, Daniel
- Girard, Yves
- Huang, Zheng
- Laliberté, France
- Liu, Susana
- Papp, Robert
- Nicholson, Donald W
- Young, Robert N
Producer: 20101228
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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3.
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Synthesis and biological activity of a potent and orally bioavailable SCD inhibitor (MF-438). [electronic resource] by
- Léger, Serge
- Black, W Cameron
- Deschenes, Denis
- Dolman, Sarah
- Falgueyret, Jean-Pierre
- Gagnon, Marc
- Guiral, Sébastien
- Huang, Zheng
- Guay, Jocelyne
- Leblanc, Yves
- Li, Chun-Sing
- Massé, Frédéric
- Oballa, Renata
- Zhang, Lei
Producer: 20100420
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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4.
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Nitrogen-bridged substituted 8-arylquinolines as potent PDE IV inhibitors. [electronic resource] by
- Lacombe, Patrick
- Deschênes, Denis
- Dubé, Daniel
- Dubé, Laurence
- Gallant, Michel
- Macdonald, Dwight
- Mastracchio, Antony
- Perrier, Hélène
- Charleson, Stella
- Huang, Zheng
- Laliberté, France
- Liu, Susana
- Mancini, Joseph A
- Masson, Paul
- Salem, Myriam
- Styhler, Angela
- Girard, Yves
Producer: 20060809
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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5.
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Structure-activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP(4) receptor. [electronic resource] by
- Burch, Jason D
- Belley, Michel
- Fortin, Réjean
- Deschênes, Denis
- Girard, Mario
- Colucci, John
- Farand, Julie
- Therien, Alex G
- Mathieu, Marie-Claude
- Denis, Danielle
- Vigneault, Erika
- Lévesque, Jean-François
- Gagné, Sébastien
- Wrona, Mark
- Xu, Daigen
- Clark, Patsy
- Rowland, Steve
- Han, Yongxin
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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6.
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Nicotinic acids: liver-targeted SCD inhibitors with preclinical anti-diabetic efficacy. [electronic resource] by
- Powell, David A
- Black, W Cameron
- Bleasby, Kelly
- Chan, Chi-Chung
- Deschenes, Denis
- Gagnon, Marc
- Gordon, Rob
- Guay, Jocelyne
- Guiral, Sebastien
- Hafey, Michael J
- Huang, Zheng
- Isabel, Elise
- Leblanc, Yves
- Styhler, Angela
- Xu, Li-Jing
- Zhang, Lei
- Oballa, Renata M
Producer: 20120312
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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7.
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Identification of a potent and selective non-basic cathepsin K inhibitor. [electronic resource] by
- Li, Chun Sing
- Deschenes, Denis
- Desmarais, Sylvie
- Falgueyret, Jean-Pierre
- Gauthier, Jacques Yves
- Kimmel, Donald B
- Léger, Serge
- Massé, Frédéric
- McGrath, Mary E
- McKay, Daniel J
- Percival, M David
- Riendeau, Denis
- Rodan, Sevgi B
- Thérien, Michel
- Truong, Vouy-Linh
- Wesolowski, Gregg
- Zamboni, Robert
- Black, W Cameron
Producer: 20060719
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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8.
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Alkyl-bridged substituted 8-arylquinolines as highly potent PDE IV inhibitors. [electronic resource] by
- Lacombe, Patrick
- Chauret, Nathalie
- Claveau, David
- Day, Stephen
- Deschênes, Denis
- Dubé, Daniel
- Gallant, Michel
- Girard, Yves
- Huang, Zheng
- Laliberté, France
- Lévesque, Jean-Francois
- Liu, Susana
- Macdonald, Dwight
- Mancini, Joseph A
- Masson, Paul
- Nicholson, Donald W
- Nicoll-Griffith, Deborah A
- Salem, Myriam
- Styhler, Angela
- Young, Robert N
Producer: 20091124
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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9.
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Design, synthesis, and biological evaluation of 8-biarylquinolines: a novel class of PDE4 inhibitors. [electronic resource] by
- Gallant, Michel
- Chauret, Nathalie
- Claveau, David
- Day, Stephen
- Deschênes, Denis
- Dubé, Daniel
- Huang, Zheng
- Lacombe, Patrick
- Laliberté, France
- Lévesque, Jean-François
- Liu, Susana
- Macdonald, Dwight
- Mancini, Joseph
- Masson, Paul
- Mastracchio, Anthony
- Nicholson, Donald
- Nicoll-Griffith, Deborah A
- Perrier, Hélène
- Salem, Myriam
- Styhler, Angela
- Young, Robert N
- Girard, Yves
Producer: 20080512
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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10.
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The identification of 4,7-disubstituted naphthoic acid derivatives as UDP-competitive antagonists of P2Y14. [electronic resource] by
- Gauthier, Jacques Yves
- Belley, Michel
- Deschênes, Denis
- Fournier, Jean-François
- Gagné, Sébastien
- Gareau, Yves
- Hamel, Martine
- Hénault, Martin
- Hyjazie, Huda
- Kargman, Stacia
- Lavallée, Geneviève
- Levesque, Jean-François
- Li, Lianhai
- Mamane, Yaël
- Mancini, Joseph
- Morin, Nicolas
- Mulrooney, Erin
- Robichaud, Joël
- Thérien, Michel
- Tranmer, Geoffrey
- Wang, Zhaoyin
- Wu, Jin
- Black, W Cameron
Producer: 20110823
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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11.
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Difluoroethylamines as an amide isostere in inhibitors of cathepsin K. [electronic resource] by
- Isabel, Elise
- Mellon, Christophe
- Boyd, Michael J
- Chauret, Nathalie
- Deschênes, Denis
- Desmarais, Sylvie
- Falgueyret, Jean-Pierre
- Gauthier, Jacques Yves
- Khougaz, Karine
- Lau, Cheuk K
- Léger, Serge
- Levorse, Dorothy A
- Li, Chun Sing
- Massé, Frédéric
- Percival, M David
- Roy, Bruno
- Scheigetz, John
- Thérien, Michel
- Truong, Vouy Linh
- Wesolowski, Gregg
- Young, Robert N
- Zamboni, Robert
- Black, W Cameron
Producer: 20110502
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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12.
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Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: structure-activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitor. [electronic resource] by
- Macdonald, Dwight
- Mastracchio, Anthony
- Perrier, Hélène
- Dubé, Daniel
- Gallant, Michel
- Lacombe, Patrick
- Deschênes, Denis
- Roy, Bruno
- Scheigetz, John
- Bateman, Kevin
- Li, Chun
- Trimble, Laird A
- Day, Stephen
- Chauret, Nathalie
- Nicoll-Griffith, Deborah A
- Silva, Jose M
- Huang, Zheng
- Laliberté, France
- Liu, Susana
- Ethier, Diane
- Pon, Doug
- Muise, Eric
- Boulet, Louise
- Chan, Chi Chung
- Styhler, Angela
- Charleson, Stella
- Mancini, Joseph
- Masson, Paul
- Claveau, David
- Nicholson, Donald
- Turner, Mervyn
- Young, Robert N
- Girard, Yves
Producer: 20060123
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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13.
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Discovery of MK-1439, an orally bioavailable non-nucleoside reverse transcriptase inhibitor potent against a wide range of resistant mutant HIV viruses. [electronic resource] by
- Côté, Bernard
- Burch, Jason D
- Asante-Appiah, Ernest
- Bayly, Chris
- Bédard, Leanne
- Blouin, Marc
- Campeau, Louis-Charles
- Cauchon, Elizabeth
- Chan, Manuel
- Chefson, Amandine
- Coulombe, Nathalie
- Cromlish, Wanda
- Debnath, Smita
- Deschênes, Denis
- Dupont-Gaudet, Kristina
- Falgueyret, Jean-Pierre
- Forget, Robert
- Gagné, Sébastien
- Gauvreau, Danny
- Girardin, Melina
- Guiral, Sébastien
- Langlois, Eric
- Li, Chun Sing
- Nguyen, Natalie
- Papp, Rob
- Plamondon, Serge
- Roy, Amélie
- Roy, Stéphanie
- Seliniotakis, Ria
- St-Onge, Miguel
- Ouellet, Stéphane
- Tawa, Paul
- Truchon, Jean-François
- Vacca, Joe
- Wrona, Marc
- Yan, Youwei
- Ducharme, Yves
Producer: 20141104
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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