Results
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1.
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High-resolution crystal structures of factor XIa coagulation factor in complex with nonbasic high-affinity synthetic inhibitors. [electronic resource] by
- Fradera, Xavier
- Kazemier, Bert
- Carswell, Emma
- Cooke, Andrew
- Oubrie, Arthur
- Hamilton, William
- Dempster, Maureen
- Krapp, Stephan
- Nagel, Susanna
- Jestel, Anja
Producer: 20120625
In:
Acta crystallographica. Section F, Structural biology and crystallization communications vol. 68
Availability: No items available.
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2.
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Dioxo-triazines as a novel series of cathepsin K inhibitors. [electronic resource] by
- Rankovic, Zoran
- Cai, Jiaqiang
- Fradera, Xavier
- Dempster, Maureen
- Mistry, Ashvin
- Mitchell, Ann
- Long, Clive
- Hamilton, Emma
- King, Angela
- Boucharens, Sylviane
- Jamieson, Craig
- Gillespie, Jonathan
- Cumming, Iain
- Uitdehaag, Joost
- van Zeeland, Mario
Producer: 20100527
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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3.
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4-(3-Trifluoromethylphenyl)-pyrimidine-2-carbonitrile as cathepsin S inhibitors: N3, not N1 is critically important. [electronic resource] by
- Cai, Jiaqiang
- Fradera, Xavier
- van Zeeland, Mario
- Dempster, Maureen
- Cameron, Kenneth S
- Bennett, D Jonathan
- Robinson, John
- Popplestone, Lucy
- Baugh, Mark
- Westwood, Paul
- Bruin, John
- Hamilton, William
- Kinghorn, Emma
- Long, Clive
- Uitdehaag, Joost C M
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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4.
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Identification of potent, soluble, and orally active TRPV1 antagonists. [electronic resource] by
- Ratcliffe, Paul
- Maclean, John
- Abernethy, Lynn
- Clarkson, Tom
- Dempster, Maureen
- Easson, Anna-Marie
- Edwards, Darren
- Everett, Katy
- Feilden, Helen
- Littlewood, Peter
- McArthur, Duncan
- McGregor, Deborah
- McLuskey, Hazel
- Nimz, Olaf
- Nisbet, Lesley-Anne
- Palin, Ronnie
- Tracey, Heather
- Walker, Glenn
Producer: 20110719
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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1H-imidazo[4,5-c]pyridine-4-carbonitrile as cathepsin S inhibitors: separation of desired cellular activity from undesired tissue accumulation through optimization of basic nitrogen pka. [electronic resource] by
- Arbuckle, Wullie
- Baugh, Mark
- Belshaw, Simone
- Bennett, D Jonathan
- Bruin, John
- Cai, Jiaqiang
- Cameron, Kenneth S
- Claxton, Chris
- Dempster, Maureen
- Everett, Kathryn
- Fradera, Xavier
- Hamilton, William
- Jones, Philip S
- Kinghorn, Emma
- Long, Clive
- Martin, Iain
- Robinson, John
- Westwood, Paul
Producer: 20110502
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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6.
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Therapeutic dosing of an orally active, selective cathepsin S inhibitor suppresses disease in models of autoimmunity. [electronic resource] by
- Baugh, Mark
- Black, Darcey
- Westwood, Paul
- Kinghorn, Emma
- McGregor, Kieran
- Bruin, John
- Hamilton, William
- Dempster, Maureen
- Claxton, Christopher
- Cai, Jiaqiang
- Bennett, Jonathan
- Long, Clive
- McKinnon, Heather
- Vink, Paul
- den Hoed, Leontien
- Gorecka, Monika
- Vora, Kalpit
- Grant, Ethan
- Percival, M David
- Boots, A Mieke H
- van Lierop, Marie-José
Producer: 20110801
In:
Journal of autoimmunity vol. 36
Availability: No items available.
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7.
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Trifluoromethylphenyl as P2 for ketoamide-based cathepsin S inhibitors. [electronic resource] by
- Cai, Jiaqiang
- Robinson, John
- Belshaw, Simone
- Everett, Kathryn
- Fradera, Xavier
- van Zeeland, Mario
- van Berkom, Leon
- van Rijnsbergen, Peter
- Popplestone, Lucy
- Baugh, Mark
- Dempster, Maureen
- Bruin, John
- Hamilton, William
- Kinghorn, Emma
- Westwood, Paul
- Kerr, Jennifer
- Rankovic, Zoran
- Arbuckle, Wullie
- Bennett, D Jonathan
- Jones, Philip S
- Long, Clive
- Martin, Iain
- Uitdehaag, Joost C M
- Meulemans, Tommi
Producer: 20110223
In:
Bioorganic & medicinal chemistry letters vol. 20
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8.
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2-Phenyl-9H-purine-6-carbonitrile derivatives as selective cathepsin S inhibitors. [electronic resource] by
- Cai, Jiaqiang
- Bennett, D Jonathan
- Rankovic, Zoran
- Dempster, Maureen
- Fradera, Xavier
- Gillespie, Jonathan
- Cumming, Iain
- Finlay, William
- Baugh, Mark
- Boucharens, Sylviane
- Bruin, John
- Cameron, Kenneth S
- Hamilton, William
- Kerr, Jennifer
- Kinghorn, Emma
- McGarry, George
- Robinson, John
- Scullion, Paul
- Uitdehaag, Joost C M
- van Zeeland, Mario
- Potin, Dominique
- Saniere, Laurent
- Fouquet, Andre
- Chevallier, Francois
- Deronzier, Hortense
- Dorleans, Cecile
- Nicolai, Eric
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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9.
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Design and optimization of a series of novel 2-cyano-pyrimidines as cathepsin K inhibitors. [electronic resource] by
- Rankovic, Zoran
- Cai, Jiaqiang
- Kerr, Jennifer
- Fradera, Xavier
- Robinson, John
- Mistry, Ashvin
- Hamilton, Emma
- McGarry, George
- Andrews, Fiona
- Caulfield, Wilson
- Cumming, Iain
- Dempster, Maureen
- Waller, John
- Scullion, Paul
- Martin, Iain
- Mitchell, Ann
- Long, Clive
- Baugh, Mark
- Westwood, Paul
- Kinghorn, Emma
- Bruin, John
- Hamilton, William
- Uitdehaag, Joost
- van Zeeland, Mario
- Potin, Dominique
- Saniere, Laurent
- Fouquet, Andre
- Chevallier, François
- Deronzier, Hortense
- Dorleans, Cecile
- Nicolai, Eric
Producer: 20100527
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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10.
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Discovery of potent, soluble and orally active TRPV1 antagonists. Structure-activity relationships of a series of isoxazoles. [electronic resource] by
- Ratcliffe, Paul
- Abernethy, Lynn
- Ansari, Nasrin
- Cameron, Ken
- Clarkson, Tom
- Dempster, Maureen
- Dunn, David
- Easson, Anna-Marie
- Edwards, Darren
- Everett, Katy
- Feilden, Helen
- Ho, Koc-Kan
- Kultgen, Steve
- Littlewood, Peter
- Maclean, John
- McArthur, Duncan
- McGregor, Deborah
- McLuskey, Hazel
- Neagu, Irina
- Nimz, Olaf
- Nisbet, Lesley-Anne
- Ohlmeyer, Michael
- Palin, Ronnie
- Pham, Quynhchi
- Rong, Yajing
- Roughton, Andrew
- Sammons, Melanie
- Swanson, Robert
- Tracey, Heather
- Walker, Glenn
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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11.
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Structure-activity studies of a novel series of isoxazole-3-carboxamide derivatives as TRPV1 antagonists. [electronic resource] by
- Palin, Ronald
- Abernethy, Lynn
- Ansari, Nasrin
- Cameron, Kenneth
- Clarkson, Tom
- Dempster, Maureen
- Dunn, David
- Easson, Anna-Marie
- Edwards, Darren
- Maclean, John
- Everett, Katy
- Feilden, Helen
- Ho, Koc-Kan
- Kultgen, Steve
- Littlewood, Peter
- McArthur, Duncan
- McGregor, Deborah
- McLuskey, Hazel
- Neagu, Irina
- Neale, Stuart
- Nisbet, Lesley-Anne
- Ohlmeyer, Michael
- Pham, Quynhchi
- Ratcliffe, Paul
- Rong, Yajing
- Roughton, Andrew
- Sammons, Melanie
- Swanson, Robert
- Tracey, Heather
- Walker, Glenn
Producer: 20110502
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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12.
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6-Phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile as cathepsin S inhibitors. [electronic resource] by
- Cai, Jiaqiang
- Baugh, Mark
- Black, Darcey
- Long, Clive
- Jonathan Bennett, D
- Dempster, Maureen
- Fradera, Xavier
- Gillespie, Jonathan
- Andrews, Fiona
- Boucharens, Sylviane
- Bruin, John
- Cameron, Kenneth S
- Cumming, Iain
- Hamilton, William
- Jones, Philip S
- Kaptein, Allard
- Kinghorn, Emma
- Maidment, Maurice
- Martin, Iain
- Mitchell, Ann
- Rankovic, Zoran
- Robinson, John
- Scullion, Paul
- Uitdehaag, Joost C M
- Vink, Paul
- Westwood, Paul
- van Zeeland, Mario
- van Berkom, Leon
- Bastiani, Martijn
- Meulemans, Tommi
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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13.
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Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: improving selectivity over hERG. [electronic resource] by
- Rankovic, Zoran
- Cai, Jiaqiang
- Kerr, Jennifer
- Fradera, Xavier
- Robinson, John
- Mistry, Ashvin
- Finlay, William
- McGarry, George
- Andrews, Fiona
- Caulfield, Wilson
- Cumming, Iain
- Dempster, Maureen
- Waller, John
- Arbuckle, Wullie
- Anderson, Mark
- Martin, Iain
- Mitchell, Ann
- Long, Clive
- Baugh, Mark
- Westwood, Paul
- Kinghorn, Emma
- Jones, Phil
- Uitdehaag, Joost C M
- van Zeeland, Mario
- Potin, Dominique
- Saniere, Laurent
- Fouquet, Andre
- Chevallier, François
- Deronzier, Hortense
- Dorleans, Cecile
- Nicolai, Eric
Producer: 20110124
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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