Results
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Inhibition of Hsp90 with resorcylic acid macrolactones: synthesis and binding studies. [electronic resource] by
- Day, James E H
- Sharp, Swee Y
- Rowlands, Martin G
- Aherne, Wynne
- Lewis, William
- Roe, S Mark
- Prodromou, Chrisostomos
- Pearl, Laurence H
- Workman, Paul
- Moody, Christopher J
Producer: 20101221
In:
Chemistry (Weinheim an der Bergstrasse, Germany) vol. 16
Availability: No items available.
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4.
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Targeting the Hsp90 molecular chaperone with novel macrolactams. Synthesis, structural, binding, and cellular studies. [electronic resource] by
- Day, James E H
- Sharp, Swee Y
- Rowlands, Martin G
- Aherne, Wynne
- Hayes, Angela
- Raynaud, Florence I
- Lewis, William
- Roe, S Mark
- Prodromou, Chrisostomos
- Pearl, Laurence H
- Workman, Paul
- Moody, Christopher J
Producer: 20120416
In:
ACS chemical biology vol. 6
Availability: No items available.
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5.
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Discovery of a Potent Nonpeptidomimetic, Small-Molecule Antagonist of Cellular Inhibitor of Apoptosis Protein 1 (cIAP1) and X-Linked Inhibitor of Apoptosis Protein (XIAP). [electronic resource] by
- Tamanini, Emiliano
- Buck, Ildiko M
- Chessari, Gianni
- Chiarparin, Elisabetta
- Day, James E H
- Frederickson, Martyn
- Griffiths-Jones, Charlotte M
- Hearn, Keisha
- Heightman, Tom D
- Iqbal, Aman
- Johnson, Christopher N
- Lewis, Edward J
- Martins, Vanessa
- Peakman, Torren
- Reader, Michael
- Rich, Sharna J
- Ward, George A
- Williams, Pamela A
- Wilsher, Nicola E
Producer: 20170704
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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6.
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Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Discovery of a Non-Alanine Lead Series with Dual Activity Against cIAP1 and XIAP. [electronic resource] by
- Chessari, Gianni
- Buck, Ildiko M
- Day, James E H
- Day, Philip J
- Iqbal, Aman
- Johnson, Christopher N
- Lewis, Edward J
- Martins, Vanessa
- Miller, Darcey
- Reader, Michael
- Rees, David C
- Rich, Sharna J
- Tamanini, Emiliano
- Vitorino, Marc
- Ward, George A
- Williams, Pamela A
- Williams, Glyn
- Wilsher, Nicola E
- Woolford, Alison J-A
Producer: 20151116
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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7.
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Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors. [electronic resource] by
- Murray, Christopher W
- Berdini, Valerio
- Buck, Ildiko M
- Carr, Maria E
- Cleasby, Anne
- Coyle, Joseph E
- Curry, Jayne E
- Day, James E H
- Day, Phillip J
- Hearn, Keisha
- Iqbal, Aman
- Lee, Lydia Y W
- Martins, Vanessa
- Mortenson, Paul N
- Munck, Joanne M
- Page, Lee W
- Patel, Sahil
- Roomans, Susan
- Smith, Kirsten
- Tamanini, Emiliano
- Saxty, Gordon
Producer: 20150720
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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8.
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A Fragment-Derived Clinical Candidate for Antagonism of X-Linked and Cellular Inhibitor of Apoptosis Proteins: 1-(6-[(4-Fluorophenyl)methyl]-5-(hydroxymethyl)-3,3-dimethyl-1 H,2 H,3 H-pyrrolo[3,2- b]pyridin-1-yl)-2-[(2 R,5 R)-5-methyl-2-([(3R)-3-methylmorpholin-4-yl]methyl)piperazin-1-yl]ethan-1-one (ASTX660). [electronic resource] by
- Johnson, Christopher N
- Ahn, Jong Sook
- Buck, Ildiko M
- Chiarparin, Elisabetta
- Day, James E H
- Hopkins, Anna
- Howard, Steven
- Lewis, Edward J
- Martins, Vanessa
- Millemaggi, Alessia
- Munck, Joanne M
- Page, Lee W
- Peakman, Torren
- Reader, Michael
- Rich, Sharna J
- Saxty, Gordon
- Smyth, Tomoko
- Thompson, Neil T
- Ward, George A
- Williams, Pamela A
- Wilsher, Nicola E
- Chessari, Gianni
Producer: 20191014
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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9.
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Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. [electronic resource] by
- Heightman, Tom D
- Berdini, Valerio
- Braithwaite, Hannah
- Buck, Ildiko M
- Cassidy, Megan
- Castro, Juan
- Courtin, Aurélie
- Day, James E H
- East, Charlotte
- Fazal, Lynsey
- Graham, Brent
- Griffiths-Jones, Charlotte M
- Lyons, John F
- Martins, Vanessa
- Muench, Sandra
- Munck, Joanne M
- Norton, David
- O'Reilly, Marc
- Palmer, Nick
- Pathuri, Puja
- Reader, Michael
- Rees, David C
- Rich, Sharna J
- Richardson, Caroline
- Saini, Harpreet
- Thompson, Neil T
- Wallis, Nicola G
- Walton, Hugh
- Wilsher, Nicola E
- Woolford, Alison J-A
- Cooke, Michael
- Cousin, David
- Onions, Stuart
- Shannon, Jonathan
- Watts, John
- Murray, Christopher W
Producer: 20190520
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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