Results
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1.
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2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists. 2. Synthesis, chirality, and pharmacokinetics. [electronic resource] by
- Borthwick, Alan D
- Davies, Dave E
- Exall, Anne M
- Livermore, David G
- Sollis, Steve L
- Nerozzi, Fabrizio
- Allen, Michael J
- Perren, Marion
- Shabbir, Shalia S
- Woollard, Patrick M
- Wyatt, Paul G
Producer: 20051220
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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2.
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Design and synthesis of pyrrolidine-5,5'-trans-lactams (5-oxo-hexahydropyrrolo[3,2-b]pyrroles) as novel mechanism-based inhibitors of human cytomegalovirus protease. 4. Antiviral activity and plasma stability. [electronic resource] by
- Borthwick, Alan D
- Davies, Dave E
- Ertl, Peter F
- Exall, Anne M
- Haley, Terry M
- Hart, Graham J
- Jackson, Deborah L
- Parry, Nigel R
- Patikis, Angela
- Trivedi, Naimisha
- Weingarten, Gordon G
- Woolven, James M
Producer: 20031112
In:
Journal of medicinal chemistry vol. 46
Availability: No items available.
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3.
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2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: Identification, stereochemistry and initial SAR. [electronic resource] by
- Wyatt, Paul G
- Allen, Michael J
- Borthwick, Alan D
- Davies, Dave E
- Exall, Anne M
- Hatley, Richard J D
- Irving, Wendy R
- Livermore, David G
- Miller, Neil D
- Nerozzi, Fabrizio
- Sollis, Steve L
- Szardenings, Anna Katrin
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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4.
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2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists. 3. Synthesis, pharmacokinetics, and in vivo potency. [electronic resource] by
- Borthwick, Alan D
- Davies, Dave E
- Exall, Anne M
- Hatley, Richard J D
- Hughes, Jennifer A
- Irving, Wendy R
- Livermore, David G
- Sollis, Steve L
- Nerozzi, Fabrizio
- Valko, Klara L
- Allen, Michael J
- Perren, Marion
- Shabbir, Shalia S
- Woollard, Patrick M
- Price, Mark A
Producer: 20060911
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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5.
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Pyridyl-2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists: synthesis, pharmacokinetics, and in vivo potency. [electronic resource] by
- Borthwick, Alan D
- Liddle, John
- Davies, Dave E
- Exall, Anne M
- Hamlett, Christopher
- Hickey, Deirdre M
- Mason, Andrew M
- Smith, Ian E D
- Nerozzi, Fabrizio
- Peace, Simon
- Pollard, Derek
- Sollis, Steve L
- Allen, Michael J
- Woollard, Patrick M
- Pullen, Mark A
- Westfall, Timothy D
- Stanislaus, Dinesh J
Producer: 20120409
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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