Substrate-dependent modulation of CYP3A4 catalytic activity: analysis of 27 test compounds with four fluorometric substrates. [electronic resource]
Producer: 20010202Description: 1440-8 p. digitalISSN:- 0090-9556
- Algorithms
- Calcium Channel Blockers -- metabolism
- Chromatography, High Pressure Liquid
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme Inhibitors
- Cytochrome P-450 Enzyme System -- metabolism
- Fluorescent Dyes -- pharmacokinetics
- GABA Modulators -- metabolism
- Humans
- In Vitro Techniques
- Kinetics
- Mass Spectrometry
- Midazolam -- metabolism
- Mixed Function Oxygenases -- antagonists & inhibitors
- Nifedipine -- metabolism
- Spectrometry, Fluorescence
- Spectrophotometry, Ultraviolet
- Testosterone -- metabolism
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Publication Type: Journal Article
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