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Synthesis and in vitro evaluation of SG3227, a pyrrolobenzodiazepine dimer antibody-drug conjugate payload based on sibiromycin. [electronic resource] by
- Kemp, Gary C
- Tiberghien, Arnaud C
- Patel, Neki V
- D'Hooge, Francois
- Nilapwar, Sanjay M
- Adams, Lauren R
- Corbett, Simon
- Williams, David G
- Hartley, John A
- Howard, Philip W
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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Uptake of unnatural trehalose analogs as a reporter for Mycobacterium tuberculosis. [electronic resource] by
- Backus, Keriann M
- Boshoff, Helena I
- Barry, Conor S
- Boutureira, Omar
- Patel, Mitul K
- D'Hooge, François
- Lee, Seung Seo
- Via, Laura E
- Tahlan, Kapil
- Barry, Clifton E
- Davis, Benjamin G
Producer: 20110513
In:
Nature chemical biology vol. 7
Availability: No items available.
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The development of boronic acids as sensors and separation tools. [electronic resource] by
- Fossey, John S
- D'Hooge, Francois
- van den Elsen, Jean M H
- Pereira Morais, Marta P
- Pascu, Sofia I
- Bull, Steven D
- Marken, Frank
- Jenkins, A Toby A
- Jiang, Yun-Bao
- James, Tony D
Producer: 20130304
In:
Chemical record (New York, N.Y.) vol. 12
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8.
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Boronate affinity saccharide electrophoresis: a novel carbohydrate analysis tool. [electronic resource] by
- Jackson, Thomas R
- Springall, Jeremy S
- Rogalle, Damien
- Masumoto, Naoko
- Ching Li, Hung
- D'Hooge, François
- Perera, Semali P
- Jenkins, A Toby A
- James, Tony D
- Fossey, John S
- van den Elsen, Jean M H
Producer: 20090126
In:
Electrophoresis vol. 29
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9.
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Synthesis and evaluation of pyrrolobenzodiazepine dimer antibody-drug conjugates with dual β-glucuronide and dipeptide triggers. [electronic resource] by
- Gregson, Stephen J
- Barrett, Allison M
- Patel, Neki V
- Kang, Gyoung-Dong
- Schiavone, Davide
- Sult, Erin
- Barry, Conor S
- Vijayakrishnan, Balakumar
- Adams, Lauren R
- Masterson, Luke A
- D'Hooge, Francois
- Snaith, Mike
- Harper, Jay
- Hartley, John A
- Howard, Philip W
Producer: 20191104
In:
European journal of medicinal chemistry vol. 179
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10.
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ADCT-402, a PBD dimer-containing antibody drug conjugate targeting CD19-expressing malignancies. [electronic resource] by
- Zammarchi, Francesca
- Corbett, Simon
- Adams, Lauren
- Tyrer, Peter C
- Kiakos, Konstantinos
- Janghra, Narinder
- Marafioti, Teresa
- Britten, Charles E
- Havenith, Carin E G
- Chivers, Simon
- D'Hooge, Francois
- Williams, David G
- Tiberghien, Arnaud
- Howard, Philip W
- Hartley, John A
- van Berkel, Patrick H
Producer: 20190319
In:
Blood vol. 131
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11.
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TR1801-ADC: a highly potent cMet antibody-drug conjugate with high activity in patient-derived xenograft models of solid tumors. [electronic resource] by
- Gymnopoulos, Marco
- Betancourt, Oscar
- Blot, Vincent
- Fujita, Ryo
- Galvan, Diana
- Lieuw, Vincent
- Nguyen, Sophie
- Snedden, Jeanette
- Stewart, Christine
- Villicana, Jose
- Wojciak, Jon
- Wong, Eley
- Pardo, Raul
- Patel, Neki
- D'Hooge, Francois
- Vijayakrishnan, Balakumar
- Barry, Conor
- Hartley, John A
- Howard, Philip W
- Newman, Roland
- Coronella, Julia
Producer: 20210203
In:
Molecular oncology vol. 14
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12.
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A single dose of antibody-drug conjugate cures a stage 1 model of African trypanosomiasis. [electronic resource] by
- MacGregor, Paula
- Gonzalez-Munoz, Andrea L
- Jobe, Fatoumatta
- Taylor, Martin C
- Rust, Steven
- Sandercock, Alan M
- Macleod, Olivia J S
- Van Bocxlaer, Katrien
- Francisco, Amanda F
- D'Hooge, Francois
- Tiberghien, Arnaud
- Barry, Conor S
- Howard, Philip
- Higgins, Matthew K
- Vaughan, Tristan J
- Minter, Ralph
- Carrington, Mark
Producer: 20191028
In:
PLoS neglected tropical diseases vol. 13
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13.
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Genetically Encoded Azide Containing Amino Acid in Mammalian Cells Enables Site-Specific Antibody-Drug Conjugates Using Click Cycloaddition Chemistry. [electronic resource] by
- VanBrunt, Michael P
- Shanebeck, Kurt
- Caldwell, Zachary
- Johnson, Jeffrey
- Thompson, Pamela
- Martin, Thomas
- Dong, Huifang
- Li, Gary
- Xu, Hengyu
- D'Hooge, Francois
- Masterson, Luke
- Bariola, Pauline
- Tiberghien, Arnaud
- Ezeadi, Ebele
- Williams, David G
- Hartley, John A
- Howard, Philip W
- Grabstein, Kenneth H
- Bowen, Michael A
- Marelli, Marcello
Producer: 20160829
In:
Bioconjugate chemistry vol. 26
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14.
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ADCT-301, a Pyrrolobenzodiazepine (PBD) Dimer-Containing Antibody-Drug Conjugate (ADC) Targeting CD25-Expressing Hematological Malignancies. [electronic resource] by
- Flynn, Michael J
- Zammarchi, Francesca
- Tyrer, Peter C
- Akarca, Ayse U
- Janghra, Narinder
- Britten, Charles E
- Havenith, Carin E G
- Levy, Jean-Noel
- Tiberghien, Arnaud
- Masterson, Luke A
- Barry, Conor
- D'Hooge, Francois
- Marafioti, Teresa
- Parren, Paul W H I
- Williams, David G
- Howard, Philip W
- van Berkel, Patrick H
- Hartley, John A
Producer: 20170615
In:
Molecular cancer therapeutics vol. 15
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15.
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Preclinical Evaluation of MEDI0641, a Pyrrolobenzodiazepine-Conjugated Antibody-Drug Conjugate Targeting 5T4. [electronic resource] by
- Harper, Jay
- Lloyd, Christopher
- Dimasi, Nazzareno
- Toader, Dorin
- Marwood, Rose
- Lewis, Leeanne
- Bannister, David
- Jovanovic, Jelena
- Fleming, Ryan
- D'Hooge, Francois
- Mao, Shenlan
- Marrero, Allison M
- Korade, Martin
- Strout, Patrick
- Xu, Linda
- Chen, Cui
- Wetzel, Leslie
- Breen, Shannon
- van Vlerken-Ysla, Lilian
- Jalla, Sanjoo
- Rebelatto, Marlon
- Zhong, Haihong
- Hurt, Elaine M
- Hinrichs, Mary Jane
- Huang, Keven
- Howard, Philip W
- Tice, David A
- Hollingsworth, Robert E
- Herbst, Ronald
- Kamal, Adeela
Producer: 20180626
In:
Molecular cancer therapeutics vol. 16
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16.
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Antitumor Activity of MEDI3726 (ADCT-401), a Pyrrolobenzodiazepine Antibody-Drug Conjugate Targeting PSMA, in Preclinical Models of Prostate Cancer. [electronic resource] by
- Cho, Song
- Zammarchi, Francesca
- Williams, David G
- Havenith, Carin E G
- Monks, Noel R
- Tyrer, Peter
- D'Hooge, Francois
- Fleming, Ryan
- Vashisht, Kapil
- Dimasi, Nazzareno
- Bertelli, Francois
- Corbett, Simon
- Adams, Lauren
- Reinert, Halla W
- Dissanayake, Sandamali
- Britten, Charles E
- King, Wanda
- Dacosta, Karma
- Tammali, Ravinder
- Schifferli, Kevin
- Strout, Patrick
- Korade, Martin
- Masson Hinrichs, Mary Jane
- Chivers, Simon
- Corey, Eva
- Liu, He
- Kim, Sae
- Bander, Neil H
- Howard, Philip W
- Hartley, John A
- Coats, Steve
- Tice, David A
- Herbst, Ronald
- van Berkel, Patrick H
Producer: 20190909
In:
Molecular cancer therapeutics vol. 17
Availability: No items available.
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