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Substituted 2H-isoquinolin-1-one as potent Rho-Kinase inhibitors. Part 1: Hit-to-lead account. [electronic resource] by
- Wu, Frank
- Büttner, Frank H
- Chen, Rhonda
- Hickey, Eugene
- Jakes, Scott
- Kaplita, Paul
- Kashem, Mohammed A
- Kerr, Steven
- Kugler, Stanley
- Paw, Zofia
- Prokopowicz, Anthony
- Shih, Cheng-Kon
- Snow, Roger
- Young, Erick
- Cywin, Charles L
Producer: 20100810
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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5.
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Substituted 2H-isoquinolin-1-ones as potent Rho-kinase inhibitors: part 2, optimization for blood pressure reduction in spontaneously hypertensive rats. [electronic resource] by
- Ginn, John D
- Bosanac, Todd
- Chen, Rhonda
- Cywin, Charles
- Hickey, Eugene
- Kashem, Mohammed
- Kerr, Steven
- Kugler, Stanley
- Li, Xiang
- Prokopowicz, Anthony
- Schlyer, Sabine
- Smith, James D
- Turner, Michael R
- Wu, Frank
- Young, Erick R R
Producer: 20101206
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Hit to lead account of the discovery of bisbenzamide and related ureidobenzamide inhibitors of Rho kinase. [electronic resource] by
- Morwick, Tina
- Büttner, Frank H
- Cywin, Charles L
- Dahmann, Georg
- Hickey, Eugene
- Jakes, Scott
- Kaplita, Paul
- Kashem, Mohammed A
- Kerr, Steven
- Kugler, Stanley
- Mao, Wang
- Marshall, Daniel
- Paw, Zofia
- Shih, Cheng-Kon
- Wu, Frank
- Young, Erick
Producer: 20100302
In:
Journal of medicinal chemistry vol. 53
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7.
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Hit to lead account of the discovery of a new class of inhibitors of Pim kinases and crystallographic studies revealing an unusual kinase binding mode. [electronic resource] by
- Qian, Kevin
- Wang, Lian
- Cywin, Charles L
- Farmer, Bennett T
- Hickey, Eugene
- Homon, Carol
- Jakes, Scott
- Kashem, Mohammed A
- Lee, George
- Leonard, Scott
- Li, Jun
- Magboo, Ronald
- Mao, Wang
- Pack, Edward
- Peng, Charlene
- Prokopowicz, Anthony
- Welzel, Morgan
- Wolak, John
- Morwick, Tina
Producer: 20090428
In:
Journal of medicinal chemistry vol. 52
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8.
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Hit-to-lead studies on benzimidazole inhibitors of ITK: discovery of a novel class of kinase inhibitors. [electronic resource] by
- Snow, Roger J
- Abeywardane, Asitha
- Campbell, Scot
- Lord, John
- Kashem, Mohammed A
- Khine, Hnin Hnin
- King, Josephine
- Kowalski, Jennifer A
- Pullen, Steven S
- Roma, Teresa
- Roth, Gregory P
- Sarko, Christopher R
- Wilson, Noel S
- Winters, Michael P
- Wolak, John P
- Cywin, Charles L
Producer: 20070906
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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9.
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Bicyclic [3.3.0]-Octahydrocyclopenta[c]pyrrolo Antagonists of Retinol Binding Protein 4: Potential Treatment of Atrophic Age-Related Macular Degeneration and Stargardt Disease. [electronic resource] by
- Cioffi, Christopher L
- Racz, Boglarka
- Freeman, Emily E
- Conlon, Michael P
- Chen, Ping
- Stafford, Douglas G
- Schwarz, Daniel M C
- Zhu, Lei
- Kitchen, Douglas B
- Barnes, Keith D
- Dobri, Nicoleta
- Michelotti, Enrique
- Cywin, Charles L
- Martin, William H
- Pearson, Paul G
- Johnson, Graham
- Petrukhin, Konstantin
Producer: 20151208
In:
Journal of medicinal chemistry vol. 58
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10.
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Discovery and SAR of novel Naphthyridines as potent inhibitors of spleen tyrosine kinase (SYK). [electronic resource] by
- Cywin, Charles L
- Zhao, Bao-Ping
- McNeil, Daniel W
- Hrapchak, Matt
- Prokopowicz, Anthony S
- Goldberg, Daniel R
- Morwick, Tina M
- Gao, Amy
- Jakes, Scott
- Kashem, Mohammed
- Magolda, Ronald L
- Soll, Richard M
- Player, Mark R
- Bobko, Mark A
- Rinker, James
- DesJarlais, Renee L
- Winters, Michael P
Producer: 20031205
In:
Bioorganic & medicinal chemistry letters vol. 13
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11.
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The design of potent hydrazones and disulfides as cathepsin S inhibitors. [electronic resource] by
- Cywin, Charles L
- Firestone, Raymond A
- McNeil, Daniel W
- Grygon, Christine A
- Crane, Kathryn M
- White, Della M
- Kinkade, Peter R
- Hopkins, Jerry L
- Davidson, Walter
- Labadia, Mark E
- Wildeson, Jessi
- Morelock, Maurice M
- Peterson, Jeffrey D
- Raymond, Ernest L
- Brown, Maryanne L
- Spero, Denice M
Producer: 20030826
In:
Bioorganic & medicinal chemistry vol. 11
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12.
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Design, synthesis, and evaluation of nonretinoid retinol binding protein 4 antagonists for the potential treatment of atrophic age-related macular degeneration and Stargardt disease. [electronic resource] by
- Cioffi, Christopher L
- Dobri, Nicoleta
- Freeman, Emily E
- Conlon, Michael P
- Chen, Ping
- Stafford, Douglas G
- Schwarz, Daniel M C
- Golden, Kathy C
- Zhu, Lei
- Kitchen, Douglas B
- Barnes, Keith D
- Racz, Boglarka
- Qin, Qiong
- Michelotti, Enrique
- Cywin, Charles L
- Martin, William H
- Pearson, Paul G
- Johnson, Graham
- Petrukhin, Konstantin
Producer: 20141203
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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13.
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5-Aminomethyl-1H-benzimidazoles as orally active inhibitors of inducible T-cell kinase (Itk). [electronic resource] by
- Winters, Michael P
- Robinson, Darius J
- Khine, Hnin Hnin
- Pullen, Steven S
- Woska, Joseph R
- Raymond, Ernest L
- Sellati, Rosemarie
- Cywin, Charles L
- Snow, Roger J
- Kashem, Mohammed A
- Wolak, John P
- King, Josephine
- Kaplita, Paul V
- Liu, Lisa H
- Farrell, Thomas M
- DesJarlais, Renee
- Roth, Gregory P
- Takahashi, Hidenori
- Moriarty, Kevin J
Producer: 20090424
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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14.
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Evolution of the thienopyridine class of inhibitors of IkappaB kinase-beta: part I: hit-to-lead strategies. [electronic resource] by
- Morwick, Tina
- Berry, Angela
- Brickwood, Janice
- Cardozo, Mario
- Catron, Katrina
- DeTuri, Molly
- Emeigh, Jonathan
- Homon, Carol
- Hrapchak, Matt
- Jacober, Stephen
- Jakes, Scott
- Kaplita, Paul
- Kelly, Terence A
- Ksiazek, John
- Liuzzi, Michel
- Magolda, Ronald
- Mao, Can
- Marshall, Daniel
- McNeil, Daniel
- Prokopowicz, Anthony
- Sarko, Christopher
- Scouten, Erika
- Sledziona, Cynthia
- Sun, Sanxing
- Watrous, Jane
- Wu, Jiang Ping
- Cywin, Charles L
Producer: 20060606
In:
Journal of medicinal chemistry vol. 49
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15.
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Design and synthesis of dipeptide nitriles as reversible and potent Cathepsin S inhibitors. [electronic resource] by
- Ward, Yancey D
- Thomson, David S
- Frye, Leah L
- Cywin, Charles L
- Morwick, Tina
- Emmanuel, Michel J
- Zindell, Renée
- McNeil, Daniel
- Bekkali, Younes
- Girardot, Marc
- Hrapchak, Matt
- DeTuri, Molly
- Crane, Kathy
- White, Della
- Pav, Susan
- Wang, Yong
- Hao, Ming-Hong
- Grygon, Christine A
- Labadia, Mark E
- Freeman, Dorothy M
- Davidson, Walter
- Hopkins, Jerry L
- Brown, Maryanne L
- Spero, Denice M
- Giradot, Marc
Producer: 20030107
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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16.
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Discovery of potent and selective PKC-theta inhibitors. [electronic resource] by
- Cywin, Charles L
- Dahmann, Georg
- Prokopowicz, Anthony S
- Young, Erick R R
- Magolda, Ronald L
- Cardozo, Mario G
- Cogan, Derek A
- Disalvo, Darren
- Ginn, John D
- Kashem, Mohammed A
- Wolak, John P
- Homon, Carol A
- Farrell, Thomas M
- Grbic, Heather
- Hu, Hanbo
- Kaplita, Paul V
- Liu, Lisa H
- Spero, Denice M
- Jeanfavre, Deborah D
- O'Shea, Kathy M
- White, Della M
- Woska, Joseph R
- Brown, Maryanne L
Producer: 20070424
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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17.
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The discovery of thienopyridine analogues as potent IkappaB kinase beta inhibitors. Part II. [electronic resource] by
- Wu, Jiang-Ping
- Fleck, Roman
- Brickwood, Janice
- Capolino, Alison
- Catron, Katrina
- Chen, Zhidong
- Cywin, Charles
- Emeigh, Jonathan
- Foerst, Melissa
- Ginn, John
- Hrapchak, Matt
- Hickey, Eugene
- Hao, Ming-Hong
- Kashem, Mohammed
- Li, Jun
- Liu, Weimin
- Morwick, Tina
- Nelson, Richard
- Marshall, Daniel
- Martin, Leslie
- Nemoto, Peter
- Potocki, Ian
- Liuzzi, Michel
- Peet, Gregory W
- Scouten, Erika
- Stefany, David
- Turner, Michael
- Weldon, Steve
- Zimmitti, Clare
- Spero, Denise
- Kelly, Terence A
Producer: 20091130
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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