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The synthesis of 2,3,6-trisubstituted 1-oxo-1,2-dihydroisoquinolines as potent CRTh [electronic resource] by
- Huang, Xianhai
- Rao, Ashwin
- Zhou, Wei
- Aslanian, Robert
- Nargund, Ravi
- Buevich, Alexei
- Zhang, Li-Kang
- Qiu, Hongchen
- Yang, Xiaoxin
- Garlisi, Charles G
- Correll, Craig
- Palani, Anandan
Producer: 20171201
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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11.
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Anti-inflammatory actions of Chemoattractant Receptor-homologous molecule expressed on Th2 by the antagonist MK-7246 in a novel rat model of Alternaria alternata elicited pulmonary inflammation. [electronic resource] by
- Gil, Malgorzata A
- Caniga, Michael
- Woodhouse, Janice D
- Eckman, Joseph
- Lee, Hyun-Hee
- Salmon, Michael
- Naber, John
- Hamilton, Valerie T
- Sevilla, Raquel S
- Bettano, Kimberly
- Klappenbach, Joel
- Moy, Lily
- Correll, Craig C
- Gervais, Francois G
- Siliphaivanh, Phieng
- Zhang, Weisheng
- Zhang-Hoover, Jie
- McLeod, Robbie L
- Cicmil, Milenko
Producer: 20150811
In:
European journal of pharmacology vol. 743
Availability: No items available.
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12.
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Quality by design (QbD) of amide isosteres: 5,5-Disubstituted isoxazolines as potent CRTh2 antagonists with favorable pharmacokinetic and drug-like properties. [electronic resource] by
- Xiao, Dong
- Zhu, Xiaohong
- Yu, Younong
- Shao, Ning
- Wu, Jie
- McCormick, Kevin D
- Dhondi, Pawan
- Qin, Jun
- Mazzola, Robert
- Tang, Haiqun
- Rao, Ashwin
- Siliphaivanh, Phieng
- Qiu, Hongchen
- Yang, Xiaoxin
- Rivelli, Maria
- Garlisi, Charles G
- Eckel, Steve
- Mukhopadhyay, Gitali
- Correll, Craig
- Rindgen, Diane
- Aslanian, Robert
- Palani, Anandan
Producer: 20141104
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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13.
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Identification of an allosteric binding site for RORγt inhibition. [electronic resource] by
- Scheepstra, Marcel
- Leysen, Seppe
- van Almen, Geert C
- Miller, J Richard
- Piesvaux, Jennifer
- Kutilek, Victoria
- van Eenennaam, Hans
- Zhang, Hongjun
- Barr, Kenneth
- Nagpal, Sunil
- Soisson, Stephen M
- Kornienko, Maria
- Wiley, Kristen
- Elsen, Nathaniel
- Sharma, Sujata
- Correll, Craig C
- Trotter, B Wesley
- van der Stelt, Mario
- Oubrie, Arthur
- Ottmann, Christian
- Parthasarathy, Gopal
- Brunsveld, Luc
Producer: 20160628
In:
Nature communications vol. 6
Availability: No items available.
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14.
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T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones-optimization, design and synthesis. [electronic resource] by
- Smith, Elizabeth M
- Sorota, Steve
- Kim, Hyunjin M
- McKittrick, Brian A
- Nechuta, Terry L
- Bennett, Chad
- Knutson, Chad
- Burnett, Duane A
- Kieselgof, Jane
- Tan, Zheng
- Rindgen, Diane
- Bridal, Terry
- Zhou, Xiaoping
- Jia, Yu-Ping
- Dong, Zoe
- Mullins, Debbie
- Zhang, Xiaoping
- Priestley, Tony
- Correll, Craig C
- Tulshian, Deen
- Czarniecki, Michael
- Greenlee, William J
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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15.
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RORγt inhibitors suppress T(H)17 responses in inflammatory arthritis and inflammatory bowel disease. [electronic resource] by
- de Wit, Jelle
- Al-Mossawi, M Hussein
- Hühn, Michael H
- Arancibia-Cárcamo, Carolina V
- Doig, Karen
- Kendrick, Benjamin
- Gundle, Roger
- Taylor, Peter
- Mcclanahan, Terri
- Murphy, Erin
- Zhang, Hongjun
- Barr, Ken
- Miller, J Richard
- Hu, Xiao
- Aicher, Thomas D
- Morgan, Rodney W
- Glick, Gary D
- Zaller, Dennis
- Correll, Craig
- Powrie, Fiona
- Bowness, Paul
Producer: 20160808
In:
The Journal of allergy and clinical immunology vol. 137
Availability: No items available.
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16.
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Discovery of [electronic resource] by
- Zhang, Hongjun
- Lapointe, Blair T
- Anthony, Neville
- Azevedo, Rita
- Cals, Jos
- Correll, Craig C
- Daniels, Matthew
- Deshmukh, Sujal
- van Eenenaam, Hans
- Ferguson, Heidi
- Hegde, Laxminarayan G
- Karstens, Willem Jan
- Maclean, John
- Miller, J Richard
- Moy, Lily Y
- Simov, Vladimir
- Nagpal, Sunil
- Oubrie, Arthur
- Palte, Rachel L
- Parthasarathy, Gopal
- Sciammetta, Nunzio
- van der Stelt, Mario
- Woodhouse, Janice D
- Trotter, B Wesley
- Barr, Kenneth
Publication details: ACS medicinal chemistry letters Feb 2020
In:
ACS medicinal chemistry letters vol. 11
Availability: No items available.
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17.
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Inhibition of RORγT Skews TCRα Gene Rearrangement and Limits T Cell Repertoire Diversity. [electronic resource] by
- Guo, Yanxia
- MacIsaac, Kenzie D
- Chen, Yi
- Miller, Richard J
- Jain, Renu
- Joyce-Shaikh, Barbara
- Ferguson, Heidi
- Wang, I-Ming
- Cristescu, Razvan
- Mudgett, John
- Engstrom, Laura
- Piers, Kyle J
- Baltus, Gretchen A
- Barr, Kenneth
- Zhang, Hongjun
- Mehmet, Huseyin
- Hegde, Laxminarayan G
- Hu, Xiao
- Carter, Laura L
- Aicher, Thomas D
- Glick, Gary
- Zaller, Dennis
- Hawwari, Abbas
- Correll, Craig C
- Jones, Dallas C
- Cua, Daniel J
Producer: 20171120
In:
Cell reports vol. 17
Availability: No items available.
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18.
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Discovery of MK-8318, a Potent and Selective CRTh2 Receptor Antagonist for the Treatment of Asthma. [electronic resource] by
- Huang, Xianhai
- Brubaker, Jason
- Zhou, Wei
- Biju, Purakkattle J
- Xiao, Li
- Shao, Ning
- Huang, Ying
- Dong, Li
- Liu, Zhidan
- Bitar, Rema
- Buevich, Alexei
- Jung, Joon
- Peterson, Scott L
- Butcher, John W
- Close, Joshua
- Martinez, Michelle
- MacCoss, Rachel N
- Zhang, Hongjun
- Crawford, Scott
- McCormick, Kevin D
- Aslanian, Robert
- Nargund, Ravi
- Correll, Craig
- Gervais, Francois
- Qiu, Hongchen
- Yang, Xiaoxin
- Garlisi, Charles
- Rindgen, Diane
- Maloney, Kevin M
- Siliphaivanh, Phieng
- Palani, Anandan
Publication details: ACS medicinal chemistry letters Jul 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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