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Synthesis of Cyclobutane-Fused Tetracyclic Scaffolds via Visible-Light Photocatalysis for Building Molecular Complexity. [electronic resource] by
- Oderinde, Martins S
- Mao, Edna
- Ramirez, Antonio
- Pawluczyk, Joseph
- Jorge, Christine
- Cornelius, Lyndon A M
- Kempson, James
- Vetrichelvan, Muthalagu
- Pitchai, Manivel
- Gupta, Anuradha
- Gupta, Arun Kumar
- Meanwell, Nicholas A
- Mathur, Arvind
- Dhar, T G Murali
Producer: 20200824
In:
Journal of the American Chemical Society vol. 142
Availability: No items available.
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Discovery of 4'-[(imidazol-1-yl)methyl]biphenyl-2-sulfonamides as dual endothelin/angiotensin II receptor antagonists. [electronic resource] by
- Tellew, John E
- Baska, Rose Ann F
- Beyer, Sophie M
- Carlson, Kenneth E
- Cornelius, Lyndon A
- Fadnis, Leena
- Gu, Zhengxiang
- Kunst, Bridgette L
- Kowala, Mark C
- Monshizadegan, Hossain
- Murugesan, Natesan
- Ryan, Carol S
- Valentine, Maria T
- Yang, Yifan
- Macor, John E
Producer: 20031027
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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4.
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Discovery of orally active pyrrolopyridine- and aminopyridine-based Met kinase inhibitors. [electronic resource] by
- Cai, Zhen-Wei
- Wei, Donna
- Schroeder, Gretchen M
- Cornelius, Lyndon A M
- Kim, Kyoung
- Chen, Xiao-Tao
- Schmidt, Robert J
- Williams, David K
- Tokarski, John S
- An, Yongmi
- Sack, John S
- Manne, Veeraswamy
- Kamath, Amrita
- Zhang, Yueping
- Marathe, Punit
- Hunt, John T
- Lombardo, Louis J
- Fargnoli, Joseph
- Borzilleri, Robert M
Producer: 20080709
In:
Bioorganic & medicinal chemistry letters vol. 18
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Discovery of N-isoxazolyl biphenylsulfonamides as potent dual angiotensin II and endothelin A receptor antagonists. [electronic resource] by
- Murugesan, Natesan
- Tellew, John E
- Gu, Zhengxiang
- Kunst, Bridgette L
- Fadnis, Leena
- Cornelius, Lyndon A
- Baska, Rose Ann F
- Yang, Yifan
- Beyer, Sophie M
- Monshizadegan, Hossain
- Dickinson, Kenneth E
- Panchal, Balkrushna
- Valentine, Maria T
- Chong, Saeho
- Morrison, Richard A
- Carlson, Kenneth E
- Powell, James R
- Moreland, Suzanne
- Barrish, Joel C
- Kowala, Mark C
- Macor, John E
Producer: 20020923
In:
Journal of medicinal chemistry vol. 45
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6.
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Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors. [electronic resource] by
- Qin, Lan-Ying
- Ruan, Zheming
- Cherney, Robert J
- Dhar, T G Murali
- Neels, James
- Weigelt, Carolyn A
- Sack, John S
- Srivastava, Anurag S
- Cornelius, Lyndon A M
- Tino, Joseph A
- Stefanski, Kevin
- Gu, Xiaomei
- Xie, Jenny
- Susulic, Vojkan
- Yang, Xiaoxia
- Yarde-Chinn, Melissa
- Skala, Stacey
- Bosnius, Ruth
- Goldstein, Christine
- Davies, Paul
- Ruepp, Stefan
- Salter-Cid, Luisa
- Bhide, Rajeev S
- Poss, Michael A
Producer: 20170704
In:
Bioorganic & medicinal chemistry letters vol. 27
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7.
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Discovery of N-(2-chloro-6-methyl- phenyl)-2-(6-(4-(2-hydroxyethyl)- piperazin-1-yl)-2-methylpyrimidin-4- ylamino)thiazole-5-carboxamide (BMS-354825), a dual Src/Abl kinase inhibitor with potent antitumor activity in preclinical assays. [electronic resource] by
- Lombardo, Louis J
- Lee, Francis Y
- Chen, Ping
- Norris, Derek
- Barrish, Joel C
- Behnia, Kamelia
- Castaneda, Stephen
- Cornelius, Lyndon A M
- Das, Jagabandhu
- Doweyko, Arthur M
- Fairchild, Craig
- Hunt, John T
- Inigo, Ivan
- Johnston, Kathy
- Kamath, Amrita
- Kan, David
- Klei, Herbert
- Marathe, Punit
- Pang, Suhong
- Peterson, Russell
- Pitt, Sidney
- Schieven, Gary L
- Schmidt, Robert J
- Tokarski, John
- Wen, Mei-Li
- Wityak, John
- Borzilleri, Robert M
Producer: 20050214
In:
Journal of medicinal chemistry vol. 47
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8.
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Synthesis and SAR of pyrrolotriazine-4-one based Eg5 inhibitors. [electronic resource] by
- Kim, Kyoung Soon
- Lu, Songfeng
- Cornelius, Lyndon A
- Lombardo, Louis J
- Borzilleri, Robert M
- Schroeder, Gretchen M
- Sheng, Christopher
- Rovnyak, George
- Crews, Donald
- Schmidt, Robert J
- Williams, David K
- Bhide, Rajeev S
- Traeger, Sarah C
- McDonnell, Patricia A
- Mueller, Luciano
- Sheriff, Steven
- Newitt, John A
- Pudzianowski, Andrew T
- Yang, Zheng
- Wild, Robert
- Lee, Frances Y
- Batorsky, Roberta
- Ryder, James S
- Ortega-Nanos, Marie
- Shen, Henry
- Gottardis, Marco
- Roussell, Deborah L
Producer: 20060911
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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9.
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Discovery of N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide (BMS-777607), a selective and orally efficacious inhibitor of the Met kinase superfamily. [electronic resource] by
- Schroeder, Gretchen M
- An, Yongmi
- Cai, Zhen-Wei
- Chen, Xiao-Tao
- Clark, Cheryl
- Cornelius, Lyndon A M
- Dai, Jun
- Gullo-Brown, Johnni
- Gupta, Ashok
- Henley, Benjamin
- Hunt, John T
- Jeyaseelan, Robert
- Kamath, Amrita
- Kim, Kyoung
- Lippy, Jonathan
- Lombardo, Louis J
- Manne, Veeraswamy
- Oppenheimer, Simone
- Sack, John S
- Schmidt, Robert J
- Shen, Guoxiang
- Stefanski, Kevin
- Tokarski, John S
- Trainor, George L
- Wautlet, Barri S
- Wei, Donna
- Williams, David K
- Zhang, Yingru
- Zhang, Yueping
- Fargnoli, Joseph
- Borzilleri, Robert M
Producer: 20100629
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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