In vivo SPECT imaging of [¹²³I]-labeled pentamidine pro-drugs for the treatment of human African trypanosomiasis, pharmacokinetics, and bioavailability studies in rats. [electronic resource]
Producer: 20160321Description: 167-75 p. digitalISSN:- 1873-3476
- Administration, Oral
- Animals
- Biological Availability
- Blood-Brain Barrier -- metabolism
- Brain -- metabolism
- Humans
- Male
- Pentamidine -- analogs & derivatives
- Prodrugs
- Rats
- Rats, Sprague-Dawley
- Succinates -- pharmacokinetics
- Time Factors
- Tissue Distribution
- Tomography, Emission-Computed, Single-Photon -- methods
- Trypanocidal Agents -- pharmacokinetics
- Trypanosomiasis, African -- drug therapy
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Publication Type: Comparative Study; Journal Article
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