Results
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1.
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Non-acidic pyrazole EP1 receptor antagonists with in vivo analgesic efficacy. [electronic resource] by
- Hall, Adrian
- Billinton, Andy
- Brown, Susan H
- Clayton, Nicholas M
- Chowdhury, Anita
- Giblin, Gerard M P
- Goldsmith, Paul
- Hayhow, Thomas G
- Hurst, David N
- Kilford, Ian R
- Naylor, Alan
- Passingham, Barry
- Winyard, Lisa
Producer: 20080709
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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2.
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Discovery of GSK345931A: An EP(1) receptor antagonist with efficacy in preclinical models of inflammatory pain. [electronic resource] by
- Hall, Adrian
- Brown, Susan H
- Budd, Christopher
- Clayton, Nicholas M
- Giblin, Gerard M P
- Goldsmith, Paul
- Hayhow, Thomas G
- Hurst, David N
- Naylor, Alan
- Anthony Rawlings, D
- Scoccitti, Tiziana
- Wilson, Alexander W
- Winchester, Wendy J
Producer: 20090302
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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3.
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Discovery of sodium 6-[(5-chloro-2-{[(4-chloro-2-fluorophenyl)methyl]oxy}phenyl)methyl]-2-pyridinecarboxylate (GSK269984A) an EP(1) receptor antagonist for the treatment of inflammatory pain. [electronic resource] by
- Hall, Adrian
- Billinton, Andy
- Brown, Susan H
- Chowdhury, Anita
- Clayton, Nicholas M
- Giblin, Gerard M P
- Gibson, Mairi
- Goldsmith, Paul A
- Hurst, David N
- Naylor, Alan
- Peet, Caroline F
- Scoccitti, Tiziana
- Wilson, Alexander W
- Winchester, Wendy
Producer: 20090821
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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4.
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1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists: Structure-activity relationships of 4- and 5-substituted benzoic acid derivatives. [electronic resource] by
- Hall, Adrian
- Brown, Susan H
- Chessell, Iain P
- Chowdhury, Anita
- Clayton, Nicholas M
- Coleman, Tanya
- Giblin, Gerard M P
- Hammond, Beverley
- Healy, Mark P
- Johnson, Matthew R
- Metcalf, Ann
- Michel, Anton D
- Naylor, Alan
- Novelli, Riccardo
- Spalding, David J
- Sweeting, Jennifer
Producer: 20070403
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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5.
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1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists. Structure-activity relationships of 6-substituted and 5,6-disubstituted benzoic acid derivatives. [electronic resource] by
- Hall, Adrian
- Brown, Susan H
- Chessell, Iain P
- Chowdhury, Anita
- Clayton, Nicholas M
- Coleman, Tanya
- Giblin, Gerard M P
- Hammond, Beverley
- Healy, Mark P
- Johnson, Matthew R
- Metcalf, Ann
- Michel, Anton D
- Naylor, Alan
- Novelli, Riccardo
- Spalding, David J
- Sweeting, Jennifer
- Winyard, Lisa
Producer: 20070413
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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6.
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Structure-activity relationships of 1,5-biaryl pyrroles as EP1 receptor antagonists. [electronic resource] by
- Hall, Adrian
- Atkinson, Stephen
- Brown, Susan H
- Chessell, Iain P
- Chowdhury, Anita
- Clayton, Nicholas M
- Coleman, Tanya
- Giblin, Gerard M P
- Gleave, Robert J
- Hammond, Beverley
- Healy, Mark P
- Johnson, Matthew R
- Michel, Anton D
- Naylor, Alan
- Novelli, Riccardo
- Spalding, David J
- Tang, Sac P
Producer: 20060925
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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7.
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Discovery of {4-[4,9-bis(ethyloxy)-1-oxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-2-fluorophenyl}acetic acid (GSK726701A), a novel EP [electronic resource] by
- Healy, Mark P
- Allan, Amanda C
- Bailey, Kristin
- Billinton, Andy
- Chessell, Iain P
- Clayton, Nicholas M
- Giblin, Gerard M P
- Kay, Melanie A
- Khaznadar, Tarik
- Michel, Anton D
- Naylor, Alan
- Price, Helen
- Spalding, David J
- Stevens, David A
- Swarbrick, Martin E
- Wilson, Alexander W
Producer: 20181227
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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8.
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The discovery of 6-[2-(5-chloro-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)-1-cyclopenten-1-yl]-2-pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin EP1 receptor antagonist for the treatment of inflammatory pain. [electronic resource] by
- Giblin, Gerard M P
- Bit, Rino A
- Brown, Susan H
- Chaignot, Hélène M
- Chowdhury, Anita
- Chessell, Iain P
- Clayton, Nicholas M
- Coleman, Tanya
- Hall, Adrian
- Hammond, Beverley
- Hurst, David N
- Michel, Anton D
- Naylor, Alan
- Novelli, Riccardo
- Scoccitti, Tiziana
- Spalding, David
- Tang, Sac P
- Wilson, Alex W
- Wilson, Rich
Producer: 20070409
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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