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Bioactivation of GPR40 Agonist MK-8666: Formation of Protein Adducts in Vitro from Reactive Acyl Glucuronide and Acyl CoA Thioester. [electronic resource] by
- Shang, Jackie
- Tschirret-Guth, Richard
- Cancilla, Mark
- Samuel, Koppara
- Chen, Qing
- Chobanian, Harry R
- Thomas, Ann
- Tong, Wei
- Josien, Hubert
- Buevich, Alexei V
- Mitra, Kaushik
Producer: 20210121
In:
Chemical research in toxicology vol. 33
Availability: No items available.
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8.
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Pyridinesulfonylureas and pyridinesulfonamides as selective bombesin receptor subtype-3 (BRS-3) agonists. [electronic resource] by
- Lo, Michael M-C
- Chobanian, Harry R
- Palyha, Oksana
- Kan, Yanqing
- Kelly, Theresa M
- Guan, Xiao-Ming
- Reitman, Marc L
- Dragovic, Jasminka
- Lyons, Kathryn A
- Nargund, Ravi P
- Lin, Linus S
Producer: 20110711
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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9.
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Differentiation of Deprotonated Acyl-, [electronic resource] by
- Niyonsaba, Edouard
- Easton, McKay W
- Feng, Erlu
- Yu, Zaikuan
- Zhang, Zhoupeng
- Sheng, Huaming
- Kong, John
- Easterling, Leah F
- Milton, Jacob
- Chobanian, Harry R
- Deprez, Nicholas R
- Cancilla, Mark T
- Kilaz, Gozdem
- Kenttämaa, Hilkka I
Producer: 20200928
In:
Analytical chemistry vol. 91
Availability: No items available.
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10.
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Improved Stability of Proline-Derived Direct Thrombin Inhibitors through Hydroxyl to Heterocycle Replacement. [electronic resource] by
- Chobanian, Harry R
- Pio, Barbara
- Guo, Yan
- Shen, Hong
- Huffman, Mark A
- Madeira, Maria
- Salituro, Gino
- Terebetski, Jenna L
- Ormes, James
- Jochnowitz, Nina
- Hoos, Lizbeth
- Zhou, Yuchen
- Lewis, Dale
- Hawes, Brian
- Mitnaul, Lyndon
- O'Neill, Kim
- Ellsworth, Kenneth
- Wang, Liangsu
- Biftu, Tesfaye
- Duffy, Joseph L
Producer: 20150525
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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11.
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The design and synthesis of novel spirocyclic heterocyclic sulfone ROMK inhibitors as diuretics. [electronic resource] by
- Chobanian, Harry R
- Guo, Yan
- Pio, Barbara
- Tang, Haifeng
- Teumelsan, Nardos
- Clements, Matthew
- Frie, Jessica
- Ferguson, Ronald
- Guo, Zach
- Thomas-Fowlkes, Brande S
- Felix, John P
- Liu, Jessica
- Kohler, Martin
- Priest, Birgit
- Hampton, Caryn
- Pai, Lee-Yuh
- Corona, Aaron
- Metzger, Joseph
- Tong, Vincent
- Joshi, Elizabeth M
- Xu, Ling
- Owens, Karen
- Maloney, Kevin
- Sullivan, Kathleen
- Pasternak, Alexander
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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12.
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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent. [electronic resource] by
- Pachanski, Michele J
- Kirkland, Melissa E
- Kosinski, Daniel T
- Mane, Joel
- Cheewatrakoolpong, Boonlert
- Xue, Jiyan
- Szeto, Daphne
- Forrest, Gail
- Miller, Corin
- Bunzel, Michelle
- Plummer, Christopher W
- Chobanian, Harry R
- Miller, Michael W
- Souza, Sarah
- Thomas-Fowlkes, Brande S
- Ogawa, Aimie M
- Weinglass, Adam B
- Di Salvo, Jerry
- Li, Xiaoyan
- Feng, Yue
- Tatosian, Daniel A
- Howard, Andrew D
- Colletti, Steven L
- Trujillo, Maria E
Producer: 20171121
In:
PloS one vol. 12
Availability: No items available.
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13.
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Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity. [electronic resource] by
- Chobanian, Harry R
- Guo, Yan
- Liu, Ping
- Chioda, Marc
- Lanza, Thomas J
- Chang, Linda
- Kelly, Theresa M
- Kan, Yanqing
- Palyha, Oksana
- Guan, Xiao-Ming
- Marsh, Donald J
- Metzger, Joseph M
- Gorski, Judith N
- Raustad, Kate
- Wang, Sheng-Ping
- Strack, Alison M
- Miller, Randy
- Pang, Jianmei
- Madeira, Maria
- Lyons, Kathy
- Dragovic, Jasminka
- Reitman, Marc L
- Nargund, Ravi P
- Lin, Linus S
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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14.
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Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs. [electronic resource] by
- Pio, Barbara
- Chobanian, Harry R
- Guo, Yan
- Josien, Hubert
- Hagmann, William K
- Miller, Michael
- Trujillo, Maria E
- Kirkland, Melissa
- Kosinski, Daniel
- Mane, Joel
- Pachanski, Michele
- Cheewatrakoolpong, Boonlert
- Ashley, Eric
- Orr, Robert
- Wright, Michael J
- Bugianesi, Randal
- Souza, Sarah
- Zhang, Xiaoping
- Di Salvo, Jerry
- Weinglass, Adam B
- Tschirret-Guth, Richard
- Samuel, Koppara
- Chen, Qing
- Shang, Jackie
- Lamca, James
- Ehrhart, Juliann
- Nargund, Ravi
- Howard, Andrew D
- Colletti, Steven L
Producer: 20200909
In:
Bioorganic & medicinal chemistry letters vol. 29
Availability: No items available.
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15.
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Structure-Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs. [electronic resource] by
- Chen, Helen Y
- Plummer, Christopher W
- Xiao, Dong
- Chobanian, Harry R
- DeMong, Duane
- Miller, Michael
- Trujillo, Maria E
- Kirkland, Melissa
- Kosinski, Daniel
- Mane, Joel
- Pachanski, Michele
- Cheewatrakoolpong, Boonlert
- Di Salvo, Jerry
- Thomas-Fowlkes, Brande
- Souza, Sarah
- Tatosian, Daniel A
- Chen, Qing
- Hafey, Michael J
- Houle, Robert
- Nolting, Andrew F
- Orr, Robert
- Ehrhart, Juliann
- Weinglass, Adam B
- Tschirret-Guth, Richard
- Howard, Andrew D
- Colletti, Steven L
Publication details: ACS medicinal chemistry letters Jul 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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16.
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The design and synthesis of potent, selective benzodiazepine sulfonamide bombesin receptor subtype 3 (BRS-3) agonists with an increased barrier of atropisomerization. [electronic resource] by
- Chobanian, Harry R
- Guo, Yan
- Liu, Ping
- Lanza, Thomas J
- Chioda, Marc
- Chang, Linda
- Kelly, Theresa M
- Kan, Yanqing
- Palyha, Oksana
- Guan, Xiao-Ming
- Marsh, Donald J
- Metzger, Joseph M
- Raustad, Katie
- Wang, Sheng-Ping
- Strack, Alison M
- Gorski, Judith N
- Miller, Randy
- Pang, Jianmei
- Lyons, Kathy
- Dragovic, Jasminka
- Ning, Jian G
- Schafer, Wes A
- Welch, Christopher J
- Gong, Xiaoyi
- Gao, Ying-Duo
- Hornak, Viktor
- Reitman, Marc L
- Nargund, Ravi P
- Lin, Linus S
Producer: 20120810
In:
Bioorganic & medicinal chemistry vol. 20
Availability: No items available.
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17.
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Discovery of benzodiazepine sulfonamide-based bombesin receptor subtype 3 agonists and their unusual chirality. [electronic resource] by
- Liu, Ping
- Lanza, Thomas J
- Chioda, Marc
- Jones, Carrie
- Chobanian, Harry R
- Guo, Yan
- Chang, Linda
- Kelly, Theresa M
- Kan, Yanqing
- Palyha, Oksana
- Guan, Xiao-Ming
- Marsh, Donald J
- Metzger, Joseph M
- Ramsay, Katie
- Wang, Sheng-Ping
- Strack, Alison M
- Miller, Randy
- Pang, Jianmei
- Lyons, Kathy
- Dragovic, Jasminka
- Ning, Jian G
- Schafer, Wes A
- Welch, Christopher J
- Gong, Xiaoyi
- Gao, Ying-Duo
- Hornak, Viktor
- Ball, Richard G
- Tsou, Nancy
- Reitman, Marc L
- Wyvratt, Matthew J
- Nargund, Ravi P
- Lin, Linus S
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 2
Availability: No items available.
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18.
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Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40. [electronic resource] by
- Lu, Jun
- Byrne, Noel
- Wang, John
- Bricogne, Gerard
- Brown, Frank K
- Chobanian, Harry R
- Colletti, Steven L
- Di Salvo, Jerry
- Thomas-Fowlkes, Brande
- Guo, Yan
- Hall, Dawn L
- Hadix, Jennifer
- Hastings, Nicholas B
- Hermes, Jeffrey D
- Ho, Thu
- Howard, Andrew D
- Josien, Hubert
- Kornienko, Maria
- Lumb, Kevin J
- Miller, Michael W
- Patel, Sangita B
- Pio, Barbara
- Plummer, Christopher W
- Sherborne, Bradley S
- Sheth, Payal
- Souza, Sarah
- Tummala, Srivanya
- Vonrhein, Clemens
- Webb, Maria
- Allen, Samantha J
- Johnston, Jennifer M
- Weinglass, Adam B
- Sharma, Sujata
- Soisson, Stephen M
Producer: 20170717
In:
Nature structural & molecular biology vol. 24
Availability: No items available.
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19.
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Discovery of MK-4409, a Novel Oxazole FAAH Inhibitor for the Treatment of Inflammatory and Neuropathic Pain. [electronic resource] by
- Chobanian, Harry R
- Guo, Yan
- Liu, Ping
- Chioda, Marc D
- Fung, Selena
- Lanza, Thomas J
- Chang, Linda
- Bakshi, Raman K
- Dellureficio, James P
- Hong, Qingmei
- McLaughlin, Mark
- Belyk, Kevin M
- Krska, Shane W
- Makarewicz, Amanda K
- Martel, Elliot J
- Leone, Joseph F
- Frey, Lisa
- Karanam, Bindhu
- Madeira, Maria
- Alvaro, Raul
- Shuman, Joyce
- Salituro, Gino
- Terebetski, Jenna L
- Jochnowitz, Nina
- Mistry, Shruti
- McGowan, Erin
- Hajdu, Richard
- Rosenbach, Mark
- Abbadie, Catherine
- Alexander, Jessica P
- Shiao, Lin-Lin
- Sullivan, Kathleen M
- Nargund, Ravi P
- Wyvratt, Matthew J
- Lin, Linus S
- DeVita, Robert J
Producer: 20140619
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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20.
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Discovery of MK-3168: A PET Tracer for Imaging Brain Fatty Acid Amide Hydrolase. [electronic resource] by
- Liu, Ping
- Hamill, Terence G
- Chioda, Marc
- Chobanian, Harry
- Fung, Selena
- Guo, Yan
- Chang, Linda
- Bakshi, Raman
- Hong, Qingmei
- Dellureficio, James
- Lin, Linus S
- Abbadie, Catherine
- Alexander, Jessica
- Jin, Hong
- Mandala, Suzanne
- Shiao, Lin-Lin
- Li, Wenping
- Sanabria, Sandra
- Williams, David
- Zeng, Zhizhen
- Hajdu, Richard
- Jochnowitz, Nina
- Rosenbach, Mark
- Karanam, Bindhu
- Madeira, Maria
- Salituro, Gino
- Powell, Joyce
- Xu, Ling
- Terebetski, Jenna L
- Leone, Joseph F
- Miller, Patricia
- Cook, Jacquelynn
- Holahan, Marie
- Joshi, Aniket
- O'Malley, Stacey
- Purcell, Mona
- Posavec, Diane
- Chen, Tsing-Bau
- Riffel, Kerry
- Williams, Mangay
- Hargreaves, Richard
- Sullivan, Kathleen A
- Nargund, Ravi P
- DeVita, Robert J
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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