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Discovery of 5-phenoxy-1,3-dimethyl-1H-pyrazole-4-carboxamides as potent agonists of TGR5 via sequential combinatorial libraries. [electronic resource] by
- Londregan, Allyn T
- Piotrowski, David W
- Futatsugi, Kentaro
- Warmus, Joseph S
- Boehm, Markus
- Carpino, Philip A
- Chin, Janice E
- Janssen, Ann M
- Roush, Nicole S
- Buxton, Joanne
- Hinchey, Terri
Producer: 20140113
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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Chemical Probe Identification Platform for Orphan GPCRs Using Focused Compound Screening: GPR39 as a Case Example. [electronic resource] by
- Boehm, Markus
- Hepworth, David
- Loria, Paula M
- Norquay, Lisa D
- Filipski, Kevin J
- Chin, Janice E
- Cameron, Kimberly O
- Brenner, Martin
- Bonnette, Peter
- Cabral, Shawn
- Conn, Edward
- Ebner, David C
- Gautreau, Denise
- Hadcock, John
- Lee, Esther C Y
- Mathiowetz, Alan M
- Morin, Michelle
- Rogers, Lucy
- Smith, Aaron
- VanVolkenburg, Maria
- Carpino, Philip A
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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5.
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Discovery of N-benzyl-2-[(4S)-4-(1H-indol-3-ylmethyl)-5-oxo-1-phenyl-4,5-dihydro-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-6-yl]-N-isopropylacetamide, an orally active, gut-selective CCK1 receptor agonist for the potential treatment of obesity. [electronic resource] by
- Elliott, Richard L
- Cameron, Kimberly O
- Chin, Janice E
- Bartlett, Jeremy A
- Beretta, Elena E
- Chen, Yue
- Jardine, Paul Da Silva
- Dubins, Jeffrey S
- Gillaspy, Melissa L
- Hargrove, Diane M
- Kalgutkar, Amit S
- LaFlamme, Janet A
- Lame, Mary E
- Martin, Kelly A
- Maurer, Tristan S
- Nardone, Nancy A
- Oliver, Robert M
- Scott, Dennis O
- Sun, Dexue
- Swick, Andrew G
- Trebino, Catherine E
- Zhang, Yingxin
Producer: 20110329
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Identification of Tetrahydropyrido[4,3-d]pyrimidine Amides as a New Class of Orally Bioavailable TGR5 Agonists. [electronic resource] by
- Piotrowski, David W
- Futatsugi, Kentaro
- Warmus, Joseph S
- Orr, Suvi T M
- Freeman-Cook, Kevin D
- Londregan, Allyn T
- Wei, Liuqing
- Jennings, Sandra M
- Herr, Michael
- Coffey, Steven B
- Jiao, Wenhua
- Storer, Gregory
- Hepworth, David
- Wang, Jian
- Lavergne, Sophie Y
- Chin, Janice E
- Hadcock, John R
- Brenner, Martin B
- Wolford, Angela C
- Janssen, Ann M
- Roush, Nicole S
- Buxton, Joanne
- Hinchey, Terri
- Kalgutkar, Amit S
- Sharma, Raman
- Flynn, Declan A
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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