Results
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Structure of the complex of trypsin with a highly potent synthetic inhibitor at 0.97 A resolution. [electronic resource] by
- Sherawat, Manashi
- Kaur, Punit
- Perbandt, Markus
- Betzel, Christian
- Slusarchyk, William A
- Bisacchi, Gregory S
- Chang, Chiehying
- Jacobson, Bruce L
- Einspahr, Howard M
- Singh, Tej P
Producer: 20070607
In:
Acta crystallographica. Section D, Biological crystallography vol. 63
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4.
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Discovery of furo[2,3-d][1,3]thiazinamines as beta amyloid cleaving enzyme-1 (BACE1) inhibitors. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Rajamani, Ramkumar
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Muckelbauer, Jodi
- Chang, ChiehYing
- Camac, Dan
- Macor, John E
- Thompson, Lorin A
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
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The structure of human tau-tubulin kinase 1 both in the apo form and in complex with an inhibitor. [electronic resource] by
- Kiefer, Susan E
- Chang, Chiehying J
- Kimura, S Roy
- Gao, Mian
- Xie, Dianlin
- Zhang, Yaqun
- Zhang, Guifen
- Gill, Martin B
- Mastalerz, Harold
- Thompson, Lorin A
- Cacace, Angela M
- Sheriff, Steven
Producer: 20141114
In:
Acta crystallographica. Section F, Structural biology communications vol. 70
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Novel 1H-(benzimidazol-2-yl)-1H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinase. [electronic resource] by
- Wittman, Mark D
- Balasubramanian, Balu
- Stoffan, Karen
- Velaparthi, Upender
- Liu, Pieying
- Krishnanathan, Subramaniam
- Carboni, Joan
- Li, Aixin
- Greer, Ann
- Attar, Ricardo
- Gottardis, Marco
- Chang, Chiehying
- Jacobson, Bruce
- Sun, Yax
- Hansel, Steven
- Zoeckler, Mary
- Vyas, Dolatrai M
Producer: 20070413
In:
Bioorganic & medicinal chemistry letters vol. 17
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7.
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Design and synthesis of carbazole carboxamides as promising inhibitors of Bruton's tyrosine kinase (BTK) and Janus kinase 2 (JAK2). [electronic resource] by
- Liu, Qingjie
- Batt, Douglas G
- Lippy, Jonathan S
- Surti, Neha
- Tebben, Andrew J
- Muckelbauer, Jodi K
- Chen, Lin
- An, Yongmi
- Chang, Chiehying
- Pokross, Matt
- Yang, Zheng
- Wang, Haiqing
- Burke, James R
- Carter, Percy H
- Tino, Joseph A
Producer: 20160524
In:
Bioorganic & medicinal chemistry letters vol. 25
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Discovery of S3-Truncated, C-6 Heteroaryl Substituted Aminothiazine β-Site APP Cleaving Enzyme-1 (BACE1) Inhibitors. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Shi, Jianliang
- Marcin, Lawrence
- Higgins, Mendi
- Rajamani, Ramkumar
- Muckelbauer, Jodi
- Lewis, Hal
- Chang, ChiehYing
- Camac, Dan
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Macor, John E
- Thompson, Lorin A
Producer: 20170612
In:
Journal of medicinal chemistry vol. 59
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Design of LFA-1 antagonists based on a 2,3-dihydro-1H-pyrrolizin-5(7aH)-one scaffold. [electronic resource] by
- Dodd, Dharmpal S
- Sheriff, Steven
- Chang, ChiehYing J
- Stetsko, Dawn K
- Phillips, Linda M
- Zhang, Yingru
- Launay, Michele
- Potin, Dominique
- Vaccaro, Wayne
- Poss, Michael A
- McKinnon, Murray
- Barrish, Joel C
- Suchard, Suzanne J
- Murali Dhar, T G
Producer: 20070725
In:
Bioorganic & medicinal chemistry letters vol. 17
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Targeting the BACE1 Active Site Flap Leads to a Potent Inhibitor That Elicits Robust Brain Aβ Reduction in Rodents. [electronic resource] by
- Wu, Yong-Jin
- Guernon, Jason
- Yang, Fukang
- Snyder, Lawrence
- Shi, Jianliang
- Mcclure, Andrea
- Rajamani, Ramkumar
- Park, Hyunsoo
- Ng, Alicia
- Lewis, Hal
- Chang, ChiehYing
- Camac, Dan
- Toyn, Jeremy H
- Ahlijanian, Michael K
- Albright, Charles F
- Macor, John E
- Thompson, Lorin A
Producer: 20160317
In:
ACS medicinal chemistry letters vol. 7
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11.
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Discovery and initial SAR of 3-(1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-ones as inhibitors of insulin-like growth factor 1-receptor (IGF-1R). [electronic resource] by
- Velaparthi, Upender
- Wittman, Mark
- Liu, Peiying
- Stoffan, Karen
- Zimmermann, Kurt
- Sang, Xiaopeng
- Carboni, Joan
- Li, Aixin
- Attar, Ricardo
- Gottardis, Marco
- Greer, Ann
- Chang, ChiehYing Y
- Jacobsen, Bruce L
- Sack, John S
- Sun, Yax
- Langley, David R
- Balasubramanian, Balu
- Vyas, Dolatrai
Producer: 20070530
In:
Bioorganic & medicinal chemistry letters vol. 17
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Molecular design and structure--activity relationships leading to the potent, selective, and orally active thrombin active site inhibitor BMS-189664. [electronic resource] by
- Das, Jagabandhu
- Kimball, S David
- Hall, Steven E
- Han, Wen Ching
- Iwanowicz, Edwin
- Lin, James
- Moquin, Robert V
- Reid, Joyce A
- Sack, John S
- Malley, Mary F
- Chang, Chiehying Y
- Chong, Saeho
- Wang-Iverson, David B
- Roberts, Daniel G M
- Seiler, Steven M
- Schumacher, William A
- Ogletree, Martin L
Producer: 20021004
In:
Bioorganic & medicinal chemistry letters vol. 12
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De novo design, synthesis, and in vitro activity of LFA-1 antagonists based on a bicyclic[5.5]hydantoin scaffold. [electronic resource] by
- Potin, Dominique
- Launay, Michele
- Nicolai, Eric
- Fabreguette, Maud
- Malabre, Patrice
- Caussade, François
- Besse, Dominique
- Skala, Stacey
- Stetsko, Dawn K
- Todderud, Gordon
- Beno, Brett R
- Cheney, Daniel L
- Chang, Chiehying J
- Sheriff, Steven
- Hollenbaugh, Diane L
- Barrish, Joel C
- Iwanowicz, Edwin J
- Suchard, Suzanne J
- Dhar, T G Murali
Producer: 20050615
In:
Bioorganic & medicinal chemistry letters vol. 15
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Tyrosine Kinase 2-mediated Signal Transduction in T Lymphocytes Is Blocked by Pharmacological Stabilization of Its Pseudokinase Domain. [electronic resource] by
- Tokarski, John S
- Zupa-Fernandez, Adriana
- Tredup, Jeffrey A
- Pike, Kristen
- Chang, ChiehYing
- Xie, Dianlin
- Cheng, Lihong
- Pedicord, Donna
- Muckelbauer, Jodi
- Johnson, Stephen R
- Wu, Sophie
- Edavettal, Suzanne C
- Hong, Yang
- Witmer, Mark R
- Elkin, Lisa L
- Blat, Yuval
- Pitts, William J
- Weinstein, David S
- Burke, James R
Producer: 20150703
In:
The Journal of biological chemistry vol. 290
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15.
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Purine derivatives as potent Bruton's tyrosine kinase (BTK) inhibitors for autoimmune diseases. [electronic resource] by
- Shi, Qing
- Tebben, Andrew
- Dyckman, Alaric J
- Li, Hedy
- Liu, Chunjian
- Lin, James
- Spergel, Steve
- Burke, James R
- McIntyre, Kim W
- Olini, Gilbert C
- Strnad, Joann
- Surti, Neha
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Cheng, Lin
- Ruan, Qian
- Leftheris, Katerina
- Carter, Percy H
- Tino, Joseph
- De Lucca, George V
Producer: 20141201
In:
Bioorganic & medicinal chemistry letters vol. 24
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16.
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Discovery of azetidinone acids as conformationally-constrained dual PPARalpha/gamma agonists. [electronic resource] by
- Wang, Wei
- Devasthale, Pratik
- Farrelly, Dennis
- Gu, Liqun
- Harrity, Thomas
- Cap, Michael
- Chu, Cuixia
- Kunselman, Lori
- Morgan, Nathan
- Ponticiello, Randy
- Zebo, Rachel
- Zhang, Litao
- Locke, Kenneth
- Lippy, Jonathan
- O'Malley, Kevin
- Hosagrahara, Vinayak
- Zhang, Lisa
- Kadiyala, Pathanjali
- Chang, Chiehying
- Muckelbauer, Jodi
- Doweyko, Arthur M
- Zahler, Robert
- Ryono, Denis
- Hariharan, Narayanan
- Cheng, Peter T W
Producer: 20080609
In:
Bioorganic & medicinal chemistry letters vol. 18
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17.
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Synthesis and structure-activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARalpha selective activators- PPARalpha and PPARgamma selectivity modulation. [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie
- Zhang, Hao
- Locke, Kenneth T
- O'Malley, Kevin
- Zhang, Litao
- Srivastava, Raijit
- Miao, Bowman
- Meyers, Daniel
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Lippy, Jonathan
- Twamley, Celeste
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Hosagrahara, Vinayak
- Zhang, Lisa
- Yang, T-J
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100727
In:
Bioorganic & medicinal chemistry letters vol. 20
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18.
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Design, synthesis and structure-activity relationships of azole acids as novel, potent dual PPAR alpha/gamma agonists. [electronic resource] by
- Zhang, Hao
- Ryono, Denis E
- Devasthale, Pratik
- Wang, Wei
- O'Malley, Kevin
- Farrelly, Dennis
- Gu, Liqun
- Harrity, Thomas
- Cap, Michael
- Chu, Cuixia
- Locke, Kenneth
- Zhang, Litao
- Lippy, Jonathan
- Kunselman, Lori
- Morgan, Nathan
- Flynn, Neil
- Moore, Lisa
- Hosagrahara, Vinayak
- Zhang, Lisa
- Kadiyala, Pathanjali
- Xu, Carrie
- Doweyko, Arthur M
- Bell, Aneka
- Chang, Chiehying
- Muckelbauer, Jodi
- Zahler, Robert
- Hariharan, Narayanan
- Cheng, Peter T W
Producer: 20090828
In:
Bioorganic & medicinal chemistry letters vol. 19
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19.
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Identification of [electronic resource] by
- Moslin, Ryan
- Zhang, Yanlei
- Wrobleski, Stephen T
- Lin, Shuqun
- Mertzman, Michael
- Spergel, Steven
- Tokarski, John S
- Strnad, Joann
- Gillooly, Kathleen
- McIntyre, Kim W
- Zupa-Fernandez, Adriana
- Cheng, Lihong
- Sun, Huadong
- Chaudhry, Charu
- Huang, Christine
- D'Arienzo, Celia
- Heimrich, Elizabeth
- Yang, Xiaoxia
- Muckelbauer, Jodi K
- Chang, ChiehYing
- Tredup, Jeffrey
- Mulligan, Dawn
- Xie, Dianlin
- Aranibar, Nelly
- Chiney, Manoj
- Burke, James R
- Lombardo, Louis
- Carter, Percy H
- Weinstein, David S
Producer: 20200706
In:
Journal of medicinal chemistry vol. 62
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20.
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Discovery of a (1H-benzoimidazol-2-yl)-1H-pyridin-2-one (BMS-536924) inhibitor of insulin-like growth factor I receptor kinase with in vivo antitumor activity. [electronic resource] by
- Wittman, Mark
- Carboni, Joan
- Attar, Ricardo
- Balasubramanian, Balu
- Balimane, Praveen
- Brassil, Patrick
- Beaulieu, Francis
- Chang, Chiehying
- Clarke, Wendy
- Dell, Janet
- Eummer, Jeffrey
- Frennesson, David
- Gottardis, Marco
- Greer, Ann
- Hansel, Steven
- Hurlburt, Warren
- Jacobson, Bruce
- Krishnananthan, Subramaniam
- Lee, Francis Y
- Li, Aixin
- Lin, Tai-An
- Liu, Peiying
- Ouellet, Carl
- Sang, Xiaopeng
- Saulnier, Mark G
- Stoffan, Karen
- Sun, Yax
- Velaparthi, Upender
- Wong, Henry
- Yang, Zheng
- Zimmermann, Kurt
- Zoeckler, Mary
- Vyas, Dolatrai
Producer: 20051101
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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