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Ethyl (3S,4aR,6S,8aR)-6-(4-ethoxycar- bonylimidazol-1-ylmethyl)decahydroiso-quinoline-3-carboxylic ester: a prodrug of a GluR5 kainate receptor antagonist active in two animal models of acute migraine. [electronic resource] by
- Filla, Sandra A
- Winter, Mark A
- Johnson, Kirk W
- Bleakman, David
- Bell, Michael G
- Bleisch, Thomas J
- Castaño, Ana M
- Clemens-Smith, Amy
- del Prado, Miriam
- Dieckman, Donna K
- Dominguez, Esteban
- Escribano, Ana
- Ho, Ken H
- Hudziak, Kevin J
- Katofiasc, Mary A
- Martinez-Perez, Jose A
- Mateo, Ana
- Mathes, Brian M
- Mattiuz, Edward L
- Ogden, Ann Marie L
- Phebus, Lee A
- Stack, Douglas R
- Stratford, Robert E
- Ornstein, Paul L
Producer: 20021021
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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5.
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GluK1 antagonists from 6-(carboxy)phenyl decahydroisoquinoline derivatives. SAR and evaluation of a prodrug strategy for oral efficacy in pain models. [electronic resource] by
- Martinez-Perez, Jose A
- Iyengar, Smriti
- Shannon, Harlan E
- Bleakman, David
- Alt, Andrew
- Arnold, Brian M
- Bell, Michael G
- Bleisch, Thomas J
- Castaño, Ana M
- Del Prado, Miriam
- Dominguez, Esteban
- Escribano, Ana M
- Filla, Sandra A
- Ho, Ken H
- Hudziak, Kevin J
- Jones, Carrie K
- Mateo, Ana
- Mathes, Brian M
- Mattiuz, Edward L
- Ogden, Ann Marie L
- Simmons, Rosa Maria A
- Stack, Douglas R
- Stratford, Robert E
- Winter, Mark A
- Wu, Zhipei
- Ornstein, Paul L
Producer: 20140817
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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6.
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Two prodrugs of potent and selective GluR5 kainate receptor antagonists actives in three animal models of pain. [electronic resource] by
- Dominguez, Esteban
- Iyengar, Smriti
- Shannon, Harlan E
- Bleakman, David
- Alt, Andrew
- Arnold, Brian M
- Bell, Michael G
- Bleisch, Thomas J
- Buckmaster, Jennifer L
- Castano, Ana M
- Del Prado, Miriam
- Escribano, Ana
- Filla, Sandra A
- Ho, Ken H
- Hudziak, Kevin J
- Jones, Carrie K
- Martinez-Perez, Jose A
- Mateo, Ana
- Mathes, Brian M
- Mattiuz, Edward L
- Ogden, Ann Marie L
- Simmons, Rosa Maria A
- Stack, Douglas R
- Stratford, Robert E
- Winter, Mark A
- Wu, Zhipei
- Ornstein, Paul L
Producer: 20050823
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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7.
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GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: in vitro profile and in vivo analgesic efficacy. [electronic resource] by
- Martinez-Perez, Jose A
- Iyengar, Smriti
- Shannon, Harlan E
- Bleakman, David
- Alt, Andrew
- Clawson, David K
- Arnold, Brian M
- Bell, Michael G
- Bleisch, Thomas J
- Castaño, Ana M
- Del Prado, Miriam
- Dominguez, Esteban
- Escribano, Ana M
- Filla, Sandra A
- Ho, Ken H
- Hudziak, Kevin J
- Jones, Carrie K
- Mateo, Ana
- Mathes, Brian M
- Mattiuz, Edward L
- Ogden, Ann Marie L
- Simmons, Rosa Maria A
- Stack, Douglas R
- Stratford, Robert E
- Winter, Mark A
- Wu, Zhipei
- Ornstein, Paul L
Producer: 20140817
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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