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Quinazolinedione sulfonamides: a novel class of competitive AMPA receptor antagonists with oral activity. [electronic resource] by
- Koller, Manuel
- Lingenhoehl, Kurt
- Schmutz, Markus
- Vranesic, Ivan-Toma
- Kallen, Joerg
- Auberson, Yves P
- Carcache, David A
- Mattes, Henri
- Ofner, Silvio
- Orain, David
- Urwyler, Stephan
Producer: 20110914
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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7.
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Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists. [electronic resource] by
- Hintermann, Samuel
- Guntermann, Christine
- Mattes, Henri
- Carcache, David A
- Wagner, Juergen
- Vulpetti, Anna
- Billich, Andreas
- Dawson, Janet
- Kaupmann, Klemens
- Kallen, Joerg
- Stringer, Rowan
- Orain, David
Producer: 20170710
In:
ChemMedChem vol. 11
Availability: No items available.
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8.
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6-Amino quinazolinedione sulfonamides as orally active competitive AMPA receptor antagonists. [electronic resource] by
- Orain, David
- Ofner, Silvio
- Koller, Manuel
- Carcache, David A
- Froestl, Wolfgang
- Allgeier, Hans
- Rasetti, Vittorio
- Nozulak, Joachim
- Mattes, Henri
- Soldermann, Nicolas
- Floersheim, Philipp
- Desrayaud, Sandrine
- Kallen, Joerg
- Lingenhoehl, Kurt
- Urwyler, Stephan
Producer: 20120824
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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9.
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Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model. [electronic resource] by
- Carcache, David A
- Vulpetti, Anna
- Kallen, Joerg
- Mattes, Henri
- Orain, David
- Stringer, Rowan
- Vangrevelinghe, Eric
- Wolf, Romain M
- Kaupmann, Klemens
- Ottl, Johannes
- Dawson, Janet
- Cooke, Nigel G
- Hoegenauer, Klemens
- Billich, Andreas
- Wagner, Juergen
- Guntermann, Christine
- Hintermann, Samuel
Producer: 20190618
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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