Results
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1.
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2' biaryl amides as novel and subtype selective M1 agonists. Part I: Identification, synthesis, and initial SAR. [electronic resource] by
- Budzik, Brian
- Garzya, Vincenzo
- Shi, Dongchuan
- Foley, James J
- Rivero, Ralph A
- Langmead, Christopher J
- Watson, Jeannette
- Wu, Zining
- Forbes, Ian T
- Jin, Jian
Producer: 20100913
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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2.
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2' biaryl amides as novel and subtype selective M1 agonists. Part II: Further optimization and profiling. [electronic resource] by
- Budzik, Brian
- Garzya, Vincenzo
- Shi, Dongchuan
- Walker, Graham
- Lauchart, Yann
- Lucas, Adam J
- Rivero, Ralph A
- Langmead, Christopher J
- Watson, Jeannette
- Wu, Zining
- Forbes, Ian T
- Jin, Jian
Producer: 20100913
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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4.
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Novel N-Substituted Benzimidazolones as Potent, Selective, CNS-Penetrant, and Orally Active M1 mAChR Agonists. [electronic resource] by
- Budzik, Brian
- Garzya, Vincenzo
- Shi, Dongchuan
- Walker, Graham
- Woolley-Roberts, Marie
- Pardoe, Joanne
- Lucas, Adam
- Tehan, Ben
- Rivero, Ralph A
- Langmead, Christopher J
- Watson, Jeannette
- Wu, Zining
- Forbes, Ian T
- Jin, Jian
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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5.
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The development of an in vitro assay to screen lipid based nanoparticles for siRNA delivery. [electronic resource] by
- Zhang, Ye
- Arrington, Leticia
- Boardman, David
- Davis, Jared
- Xu, Yan
- DiFelice, Katie
- Stirdivant, Steve
- Wang, Weimin
- Budzik, Brian
- Bawiec, Jack
- Deng, James
- Beutner, Greg
- Seifried, Darla
- Stanton, Matthew
- Gindy, Marian
- Leone, Anthony
Producer: 20140912
In:
Journal of controlled release : official journal of the Controlled Release Society vol. 174
Availability: No items available.
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6.
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M3 muscarinic acetylcholine receptor antagonists: SAR and optimization of bi-aryl amines. [electronic resource] by
- Budzik, Brian
- Wang, Yonghui
- Shi, Dongchuan
- Wang, Feng
- Xie, Haibo
- Wan, Zehong
- Zhu, Chongye
- Foley, James J
- Nuthulaganti, Parvathi
- Kallal, Lorena A
- Sarau, Henry M
- Morrow, Dwight M
- Moore, Michael L
- Rivero, Ralph A
- Palovich, Michael
- Salmon, Michael
- Belmonte, Kristen E
- Laine, Dramane I
- Jin, Jian
Producer: 20090820
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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7.
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Discovery of biphenyl piperazines as novel and long acting muscarinic acetylcholine receptor antagonists. [electronic resource] by
- Jin, Jian
- Budzik, Brian
- Wang, Yonghui
- Shi, Dongchuan
- Wang, Feng
- Xie, Haibo
- Wan, Zehong
- Zhu, Chongye
- Foley, James J
- Webb, Edward F
- Berlanga, Manuela
- Burman, Miriam
- Sarau, Henry M
- Morrow, Dwight M
- Moore, Michael L
- Rivero, Ralph A
- Palovich, Michael
- Salmon, Michael
- Belmonte, Kristen E
- Lainé, Dramane I
Producer: 20081030
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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8.
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Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists. [electronic resource] by
- Jin, Jian
- Morales-Ramos, Angel
- Eidam, Patrick
- Mecom, John
- Li, Yue
- Brooks, Carl
- Hilfiker, Mark
- Zhang, David
- Wang, Ning
- Shi, Dongchuan
- Tseng, Pei-San
- Wheless, Karen
- Budzik, Brian
- Evans, Karen
- Jaworski, Jon-Paul
- Jugus, Jack
- Leon, Lisa
- Wu, Charlene
- Pullen, Mark
- Karamshi, Bhumika
- Rao, Parvathi
- Ward, Emma
- Laping, Nicholas
- Evans, Christopher
- Leach, Colin
- Holt, Dennis
- Su, Xin
- Morrow, Dwight
- Fries, Harvey
- Thorneloe, Kevin
- Edwards, Richard
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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9.
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Discovery of 3-aryl-4-isoxazolecarboxamides as TGR5 receptor agonists. [electronic resource] by
- Evans, Karen A
- Budzik, Brian W
- Ross, Sean A
- Wisnoski, David D
- Jin, Jian
- Rivero, Ralph A
- Vimal, Mythily
- Szewczyk, George R
- Jayawickreme, Channa
- Moncol, David L
- Rimele, Thomas J
- Armour, Susan L
- Weaver, Susan P
- Griffin, Robert J
- Tadepalli, Sarva M
- Jeune, Michael R
- Shearer, Todd W
- Chen, Zibin B
- Chen, Lihong
- Anderson, Donald L
- Becherer, J David
- De Los Frailes, Maite
- Colilla, Francisco Javier
Producer: 20100106
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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10.
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Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid-4 with in Vivo Activity in a Pulmonary Edema Model. [electronic resource] by
- Pero, Joseph E
- Matthews, Jay M
- Behm, David J
- Brnardic, Edward J
- Brooks, Carl
- Budzik, Brian W
- Costell, Melissa H
- Donatelli, Carla A
- Eisennagel, Stephen H
- Erhard, Karl
- Fischer, Michael C
- Holt, Dennis A
- Jolivette, Larry J
- Li, Huijie
- Li, Peng
- McAtee, John J
- McCleland, Brent W
- Pendrak, Israil
- Posobiec, Lorraine M
- Rivera, Katrina L K
- Rivero, Ralph A
- Roethke, Theresa J
- Sender, Matthew R
- Shu, Arthur
- Terrell, Lamont R
- Vaidya, Kalindi
- Xu, Xiaoping
- Lawhorn, Brian G
Producer: 20191028
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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