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A new orally bioavailable dual adenosine A2B/A3 receptor antagonist with therapeutic potential. [electronic resource] by
- Press, Neil J
- Taylor, Roger J
- Fullerton, Joseph D
- Tranter, Pamela
- McCarthy, Clive
- Keller, Thomas H
- Brown, Lyndon
- Cheung, Robert
- Christie, Julie
- Haberthuer, Sandra
- Hatto, Julia D I
- Keenan, Mark
- Mercer, Mark K
- Press, Nicola E
- Sahri, Helene
- Tuffnell, Andrew R
- Tweed, Morris
- Fozard, John R
Producer: 20050919
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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7.
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Discovery and Optimization of 4-(8-(3-Fluorophenyl)-1,7-naphthyridin-6-yl)transcyclohexanecarboxylic Acid, an Improved PDE4 Inhibitor for the Treatment of Chronic Obstructive Pulmonary Disease (COPD). [electronic resource] by
- Press, Neil J
- Taylor, Roger J
- Fullerton, Joseph D
- Tranter, Pamela
- McCarthy, Clive
- Keller, Thomas H
- Arnold, Nicola
- Beer, David
- Brown, Lyndon
- Cheung, Robert
- Christie, Julie
- Denholm, Alastair
- Haberthuer, Sandra
- Hatto, Julia D I
- Keenan, Mark
- Mercer, Mark K
- Oakman, Helen
- Sahri, Helene
- Tuffnell, Andrew R
- Tweed, Morris
- Trifilieff, Alexandre
Producer: 20151214
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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8.
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The identification of 7-[(R)-2-((1S,2S)-2-benzyloxycyclopentylamino)-1-hydroxyethyl]-4-hydroxybenzothiazolone as an inhaled long-acting β2-adrenoceptor agonist. [electronic resource] by
- Arnold, Nicola
- Beattie, David
- Bradley, Michelle
- Brearley, Andrew
- Brown, Lyndon
- Charlton, Steven J
- Fairhurst, Robin A
- Farr, David
- Fozard, John
- Fullerton, Joe
- Gosling, Martin
- Hatto, Julia
- Janus, Diana
- Jones, Darryl
- Jordan, Lynne
- Lewis, Christine
- Maas, Janet
- McCarthy, Clive
- Mercer, Mark
- Oakman, Helen
- Press, Neil
- Profit, Rachel
- Schuerch, Friedrich
- Sykes, David
- Taylor, Roger J
- Trifilieff, Alexandre
- Tuffnell, Andrew
Producer: 20150330
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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9.
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Solubility-driven optimization of phosphodiesterase-4 inhibitors leading to a clinical candidate. [electronic resource] by
- Press, Neil J
- Taylor, Roger J
- Fullerton, Joseph D
- Tranter, Pamela
- McCarthy, Clive
- Keller, Thomas H
- Arnold, Nicola
- Beer, David
- Brown, Lyndon
- Cheung, Robert
- Christie, Julie
- Denholm, Alastair
- Haberthuer, Sandra
- Hatto, Julia D I
- Keenan, Mark
- Mercer, Mark K
- Oakman, Helen
- Sahri, Helene
- Tuffnell, Andrew R
- Tweed, Morris
- Tyler, John W
- Wagner, Trixie
- Fozard, John R
- Trifilieff, Alexandre
Producer: 20121231
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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10.
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Correction to "Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP [electronic resource] by
- Sandham, David A
- Barker, Lucy
- Brown, Lyndon
- Brown, Zarin
- Budd, David
- Charlton, Steven J
- Chatterjee, Devnandan
- Cox, Brian
- Dubois, Gerald
- Duggan, Nicholas
- Hall, Edward
- Hatto, Julia
- Leblanc, Catherine
- Maas, Janet
- Manini, Jodie
- Profit, Rachael
- Riddy, Darren
- Ritchie, Catherine
- Sohal, Bindi
- Shaw, Duncan
- Stringer, Rowan
- Sykes, David A
- Thomas, Matthew
- Turner, Katharine L
- Watson, Simon J
- West, Ryan
- Willard, Elisabeth
- Williams, Gareth
- Willis, Jennifer
Publication details: ACS medicinal chemistry letters Sep 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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11.
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Discovery of Fevipiprant (NVP-QAW039), a Potent and Selective DP [electronic resource] by
- Sandham, David A
- Barker, Lucy
- Brown, Lyndon
- Brown, Zarin
- Budd, David
- Charlton, Steven J
- Chatterjee, Devnandan
- Cox, Brian
- Dubois, Gerald
- Duggan, Nicholas
- Hall, Edward
- Hatto, Julia
- Maas, Janet
- Manini, Jodie
- Profit, Rachael
- Riddy, Darren
- Ritchie, Catherine
- Sohal, Bindi
- Shaw, Duncan
- Stringer, Rowan
- Sykes, David A
- Thomas, Matthew
- Turner, Katharine L
- Watson, Simon J
- West, Ryan
- Willard, Elisabeth
- Williams, Gareth
- Willis, Jennifer
Publication details: ACS medicinal chemistry letters May 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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12.
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Discovery and characterization of NVP-QAV680, a potent and selective CRTh2 receptor antagonist suitable for clinical testing in allergic diseases. [electronic resource] by
- Sandham, David A
- Arnold, Nicola
- Aschauer, Heinrich
- Bala, Kamlesh
- Barker, Lucy
- Brown, Lyndon
- Brown, Zarin
- Budd, David
- Cox, Brian
- Docx, Cerys
- Dubois, Gerald
- Duggan, Nicholas
- England, Karen
- Everatt, Brian
- Furegati, Marcus
- Hall, Edward
- Kalthoff, Frank
- King, Anna
- Leblanc, Catherine J
- Manini, Jodie
- Meingassner, Josef
- Profit, Rachael
- Schmidt, Alfred
- Simmons, Jennifer
- Sohal, Bindi
- Stringer, Rowan
- Thomas, Matthew
- Turner, Katharine L
- Walker, Christoph
- Watson, Simon J
- Westwick, John
- Willis, Jennifer
- Williams, Gareth
- Wilson, Caroline
Producer: 20140526
In:
Bioorganic & medicinal chemistry vol. 21
Availability: No items available.
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