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Conversion of human-selective PPARalpha agonists to human/mouse dual agonists: a molecular modeling analysis. [electronic resource] by
- Wang, Minmin
- Winneroski, Leonard L
- Ardecky, Robert J
- Babine, Robert E
- Brooks, Dawn A
- Etgen, Garret J
- Hutchison, Darrell R
- Kauffman, Raymond F
- Kunkel, Aaron
- Mais, Dale E
- Montrose-Rafizadeh, Chahrzad
- Ogilvie, Kathleen M
- Oldham, Brian A
- Peters, Mary K
- Rito, Christopher J
- Rungta, Deepa K
- Tripp, Allie E
- Wilson, Sarah B
- Xu, Yanping
- Zink, Richard W
- McCarthy, James R
Producer: 20050420
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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9.
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A tailored therapy for the metabolic syndrome: the dual peroxisome proliferator-activated receptor-alpha/gamma agonist LY465608 ameliorates insulin resistance and diabetic hyperglycemia while improving cardiovascular risk factors in preclinical models. [electronic resource] by
- Etgen, Garret J
- Oldham, Brian A
- Johnson, William T
- Broderick, Carol L
- Montrose, Chahrzad R
- Brozinick, Joseph T
- Misener, Elizabeth A
- Bean, James S
- Bensch, William R
- Brooks, Dawn A
- Shuker, Anthony J
- Rito, Christopher J
- McCarthy, James R
- Ardecky, Robert J
- Tyhonas, John S
- Dana, Sharon L
- Bilakovics, James M
- Paterniti, James R
- Ogilvie, Kathleen M
- Liu, Sha
- Kauffman, Raymond F
Producer: 20020510
In:
Diabetes vol. 51
Availability: No items available.
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10.
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2-Alkoxydihydrocinnamates as PPAR agonists. Activity modulation by the incorporation of phenoxy substituents. [electronic resource] by
- Martín, José A
- Brooks, Dawn A
- Prieto, Lourdes
- González, Rosario
- Torrado, Alicia
- Rojo, Isabel
- López de Uralde, Beatriz
- Lamas, Carlos
- Ferritto, Rafael
- Dolores Martín-Ortega, María
- Agejas, Javier
- Parra, Francisco
- Rizzo, John R
- Rhodes, Gary A
- Robey, Roger L
- Alt, Charles A
- Wendel, Samuel R
- Zhang, Tony Y
- Reifel-Miller, Anne
- Montrose-Rafizadeh, Chahrzad
- Brozinick, Joseph T
- Hawkins, Eric
- Misener, Elizabeth A
- Briere, Daniel A
- Ardecky, Robert
- Fraser, James D
- Warshawsky, Alan M
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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11.
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Design and synthesis of alpha-aryloxy-alpha-methylhydrocinnamic acids: a novel class of dual peroxisome proliferator-activated receptor alpha/gamma agonists. [electronic resource] by
- Xu, Yanping
- Rito, Christopher J
- Etgen, Garret J
- Ardecky, Robert J
- Bean, James S
- Bensch, William R
- Bosley, Jacob R
- Broderick, Carol L
- Brooks, Dawn A
- Dominianni, Samuel J
- Hahn, Patric J
- Liu, Sha
- Mais, Dale E
- Montrose-Rafizadeh, Chahrzad
- Ogilvie, Kathy M
- Oldham, Brian A
- Peters, Mary
- Rungta, Deepa K
- Shuker, Anthony J
- Stephenson, Gregory A
- Tripp, Allie E
- Wilson, Sarah B
- Winneroski, Leonard L
- Zink, Richard
- Kauffman, Raymond F
- McCarthy, James R
Producer: 20040616
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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12.
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The Discovery, Preclinical, and Early Clinical Development of Potent and Selective GPR40 Agonists for the Treatment of Type 2 Diabetes Mellitus (LY2881835, LY2922083, and LY2922470). [electronic resource] by
- Hamdouchi, Chafiq
- Kahl, Steven D
- Patel Lewis, Anjana
- Cardona, Guemalli R
- Zink, Richard W
- Chen, Keyue
- Eessalu, Thomas E
- Ficorilli, James V
- Marcelo, Marialuisa C
- Otto, Keith A
- Wilbur, Kelly L
- Lineswala, Jayana P
- Piper, Jared L
- Coffey, D Scott
- Sweetana, Stephanie A
- Haas, Joseph V
- Brooks, Dawn A
- Pratt, Edward J
- Belin, Ruth M
- Deeg, Mark A
- Ma, Xiaosu
- Cannady, Ellen A
- Johnson, Jason T
- Yumibe, Nathan P
- Chen, Qi
- Maiti, Pranab
- Montrose-Rafizadeh, Chahrzad
- Chen, Yanyun
- Reifel Miller, Anne
Producer: 20170619
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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