Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of Aurora-A kinase. [electronic resource]
Producer: 20111109Description: 312-9 p. digitalISSN:- 1520-4804
- Administration, Oral
- Antineoplastic Agents -- chemical synthesis
- Aurora Kinase B
- Aurora Kinases
- Biological Availability
- Cell Line, Tumor
- Crystallography, X-Ray
- Drug Screening Assays, Antitumor
- Humans
- Models, Molecular
- Molecular Structure
- Phthalazines -- chemical synthesis
- Protein Serine-Threonine Kinases -- antagonists & inhibitors
- Pyrazoles -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article
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