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Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acne. [electronic resource] by
- Thoreau, Etienne
- Arlabosse, Jean-Marie
- Bouix-Peter, Claire
- Chambon, Sandrine
- Chantalat, Laurent
- Daver, Sébastien
- Dumais, Laurence
- Duvert, Gwenaëlle
- Feret, Angélique
- Ouvry, Gilles
- Pascau, Jonathan
- Raffin, Catherine
- Rodeville, Nicolas
- Soulet, Catherine
- Tabet, Samuel
- Talano, Sandrine
- Portal, Thibaud
Producer: 20181218
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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3.
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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists. [electronic resource] by
- Ouvry, Gilles
- Bouix-Peter, Claire
- Ciesielski, Fabrice
- Chantalat, Laurent
- Christin, Olivier
- Comino, Catherine
- Duvert, Denis
- Feret, Christophe
- Harris, Craig S
- Lamy, Laurent
- Luzy, Anne-Pascale
- Musicki, Branislav
- Orfila, Danielle
- Pascau, Jonathan
- Parnet, Véronique
- Perrin, Agnès
- Pierre, Romain
- Polge, Gaëlle
- Raffin, Catherine
- Rival, Yves
- Taquet, Nathalie
- Thoreau, Etienne
- Hennequin, Laurent F
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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4.
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Identification of novel TACE inhibitors compatible with topical application. [electronic resource] by
- Ouvry, Gilles
- Berton, Yaël
- Bhurruth-Alcor, Yushma
- Bonnary, Laetitia
- Bouix-Peter, Claire
- Bouquet, Karine
- Bourotte, Marilyne
- Chambon, Sandrine
- Comino, Catherine
- Deprez, Benoît
- Duvert, Denis
- Duvert, Gwenaëlle
- Hacini-Rachinel, Feriel
- Harris, Craig S
- Luzy, Anne-Pascale
- Mathieu, Arnaud
- Millois, Corinne
- Pascau, Jonathan
- Pinto, Artur
- Polge, Gaëlle
- Reitz, Arnaud
- Reversé, Kevin
- Rosignoli, Carine
- Taquet, Nathalie
- Hennequin, Laurent F
Producer: 20170718
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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5.
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Sulfoximines as potent RORγ inverse agonists. [electronic resource] by
- Ouvry, Gilles
- Bihl, Franck
- Bouix-Peter, Claire
- Christin, Olivier
- Defoin-Platel, Claire
- Deret, Sophie
- Feret, Christophe
- Froude, David
- Hacini-Rachinel, Feriel
- Harris, Craig S
- Hervouet, Catherine
- Lafitte, Guillaume
- Luzy, Anne-Pascale
- Musicki, Branislav
- Orfila, Danielle
- Parnet, Veronique
- Pascau, Coralie
- Pascau, Jonathan
- Pierre, Romain
- Raffin, Catherine
- Rossio, Patricia
- Spiesse, Delphine
- Taquet, Nathalie
- Thoreau, Etienne
- Vatinel, Rodolphe
- Vial, Emmanuel
- Hennequin, Laurent F
Producer: 20190227
In:
Bioorganic & medicinal chemistry letters vol. 28
Availability: No items available.
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6.
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Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne. [electronic resource] by
- Fournier, Jean-François
- Clary, Laurence
- Chambon, Sandrine
- Dumais, Laurence
- Harris, Craig Steven
- Millois, Corinne
- Pierre, Romain
- Talano, Sandrine
- Thoreau, Étienne
- Aubert, Jérome
- Aurelly, Michèle
- Bouix-Peter, Claire
- Brethon, Anne
- Chantalat, Laurent
- Christin, Olivier
- Comino, Catherine
- El-Bazbouz, Ghizlane
- Ghilini, Anne-Laurence
- Isabet, Tatiana
- Lardy, Claude
- Luzy, Anne-Pascale
- Mathieu, Céline
- Mebrouk, Kenny
- Orfila, Danielle
- Pascau, Jonathan
- Reverse, Kevin
- Roche, Didier
- Rodeschini, Vincent
- Hennequin, Laurent François
Producer: 20190528
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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7.
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Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis. [electronic resource] by
- Boiteau, Jean-Guy
- Ouvry, Gilles
- Arlabosse, Jean-Marie
- Astri, Stéphanie
- Beillard, Audrey
- Bhurruth-Alcor, Yushma
- Bonnary, Laetitia
- Bouix-Peter, Claire
- Bouquet, Karine
- Bourotte, Marilyne
- Cardinaud, Isabelle
- Comino, Catherine
- Deprez, Benoît
- Duvert, Denis
- Féret, Angélique
- Hacini-Rachinel, Feriel
- Harris, Craig S
- Luzy, Anne-Pascale
- Mathieu, Arnaud
- Millois, Corinne
- Orsini, Nicolas
- Pascau, Jonathan
- Pinto, Artur
- Piwnica, David
- Polge, Gaëlle
- Reitz, Arnaud
- Reversé, Kevin
- Rodeville, Nicolas
- Rossio, Patricia
- Spiesse, Delphine
- Tabet, Samuel
- Taquet, Nathalie
- Tomas, Loïc
- Vial, Emmanuel
- Hennequin, Laurent F
Producer: 20180907
In:
Bioorganic & medicinal chemistry vol. 26
Availability: No items available.
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8.
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Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis. [electronic resource] by
- Ouvry, Gilles
- Atrux-Tallau, Nicolas
- Bihl, Franck
- Bondu, Aline
- Bouix-Peter, Claire
- Carlavan, Isabelle
- Christin, Olivier
- Cuadrado, Marie-Josée
- Defoin-Platel, Claire
- Deret, Sophie
- Duvert, Denis
- Feret, Christophe
- Forissier, Mathieu
- Fournier, Jean-François
- Froude, David
- Hacini-Rachinel, Fériel
- Harris, Craig Steven
- Hervouet, Catherine
- Huguet, Hélène
- Lafitte, Guillaume
- Luzy, Anne-Pascale
- Musicki, Branislav
- Orfila, Danielle
- Ozello, Benjamin
- Pascau, Coralie
- Pascau, Jonathan
- Parnet, Véronique
- Peluchon, Guillaume
- Pierre, Romain
- Piwnica, David
- Raffin, Catherine
- Rossio, Patricia
- Spiesse, Delphine
- Taquet, Nathalie
- Thoreau, Etienne
- Vatinel, Rodolphe
- Vial, Emmanuel
- Hennequin, Laurent François
Producer: 20190122
In:
ChemMedChem vol. 13
Availability: No items available.
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