New Cav2 calcium channel gating modifiers with agonist activity and therapeutic potential to treat neuromuscular disease. [electronic resource]
Producer: 20181113Description: 176-189 p. digitalISSN:- 1873-7064
- Animals
- Biophysics
- Calcium Channel Agonists -- chemistry
- Calcium Channels, N-Type -- genetics
- Cell Line
- Dose-Response Relationship, Drug
- Electric Stimulation
- Green Fluorescent Proteins -- genetics
- HEK293 Cells
- Humans
- Ion Channel Gating -- drug effects
- Membrane Potentials -- drug effects
- Neuroblastoma -- pathology
- Neurotransmitter Agents -- metabolism
- Patch-Clamp Techniques
- Purines -- chemistry
- Synaptic Transmission -- drug effects
- Thiophenes -- chemistry
- Time Factors
- Transfection
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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