Results
|
1.
|
Discovery of novel insulin-like growth factor-1 receptor inhibitors with unique time-dependent binding kinetics. [electronic resource] by
- Jin, Meizhong
- Petronella, Brenda A
- Cooke, Andy
- Kadalbajoo, Mridula
- Siu, Kam W
- Kleinberg, Andrew
- May, Earl W
- Gokhale, Prafulla C
- Schulz, Ryan
- Kahler, Jennifer
- Bittner, Mark A
- Foreman, Kenneth
- Pachter, Jonathan A
- Wild, Robert
- Epstein, David
- Mulvihill, Mark J
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
|
|
2.
|
Discovery of potent, selective and orally bioavailable imidazo[1,5-a]pyrazine derived ACK1 inhibitors. [electronic resource] by
- Jin, Meizhong
- Wang, Jing
- Kleinberg, Andrew
- Kadalbajoo, Mridula
- Siu, Kam W
- Cooke, Andrew
- Bittner, Mark A
- Yao, Yan
- Thelemann, April
- Ji, Qunsheng
- Bhagwat, Shripad
- Mulvihill, Kristen M
- Rechka, Josef A
- Pachter, Jonathan A
- Crew, Andrew P
- Epstein, David
- Mulvihill, Mark J
Producer: 20131031
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
|
|
3.
|
Potent and selective cyclohexyl-derived imidazopyrazine insulin-like growth factor 1 receptor inhibitors with in vivo efficacy. [electronic resource] by
- Jin, Meizhong
- Kleinberg, Andrew
- Cooke, Andy
- Gokhale, Prafulla C
- Foreman, Kenneth
- Dong, Hanqing
- Siu, Kam W
- Bittner, Mark A
- Mulvihill, Kristen M
- Yao, Yan
- Landfair, Darla
- O'Connor, Matthew
- Mak, Gilda
- Pachter, Jonathan A
- Wild, Robert
- Rosenfeld-Franklin, Maryland
- Ji, Qunsheng
- Mulvihill, Mark J
Producer: 20110523
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
|
|
4.
|
Discovery of an Orally Efficacious Imidazo[5,1-f][1,2,4]triazine Dual Inhibitor of IGF-1R and IR. [electronic resource] by
- Jin, Meizhong
- Gokhale, Prafulla C
- Cooke, Andy
- Foreman, Kenneth
- Buck, Elizabeth
- May, Earl W
- Feng, Lixin
- Bittner, Mark A
- Kadalbajoo, Mridula
- Landfair, Darla
- Siu, Kam W
- Stolz, Kathryn M
- Werner, Douglas S
- Laufer, Radoslaw S
- Li, An-Hu
- Dong, Hanqing
- Steinig, Arno G
- Kleinberg, Andrew
- Yao, Yan
- Pachter, Jonathan A
- Wild, Robert
- Mulvihill, Mark J
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
|
|
5.
|
Imidazo[1,5-a]pyrazines: orally efficacious inhibitors of mTORC1 and mTORC2. [electronic resource] by
- Crew, Andrew P
- Bhagwat, Shripad V
- Dong, Hanqing
- Bittner, Mark A
- Chan, Anna
- Chen, Xin
- Coate, Heather
- Cooke, Andrew
- Gokhale, Prafulla C
- Honda, Ayako
- Jin, Meizhong
- Kahler, Jennifer
- Mantis, Christine
- Mulvihill, Mark J
- Tavares-Greco, Paula A
- Volk, Brian
- Wang, Jing
- Werner, Douglas S
- Arnold, Lee D
- Pachter, Jonathan A
- Wild, Robert
- Gibson, Neil W
Producer: 20110711
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
|
|
6.
|
OSI-930: a novel selective inhibitor of Kit and kinase insert domain receptor tyrosine kinases with antitumor activity in mouse xenograft models. [electronic resource] by
- Garton, Andrew J
- Crew, Andrew P A
- Franklin, Maryland
- Cooke, Andrew R
- Wynne, Graham M
- Castaldo, Linda
- Kahler, Jennifer
- Winski, Shannon L
- Franks, April
- Brown, Eric N
- Bittner, Mark A
- Keily, John F
- Briner, Paul
- Hidden, Chris
- Srebernak, Mary C
- Pirrit, Carrie
- O'Connor, Matthew
- Chan, Anna
- Vulevic, Bojana
- Henninger, Dwight
- Hart, Karen
- Sennello, Regina
- Li, An-Hu
- Zhang, Tao
- Richardson, Frank
- Emerson, David L
- Castelhano, Arlindo L
- Arnold, Lee D
- Gibson, Neil W
Producer: 20060214
In:
Cancer research vol. 66
Availability: No items available.
|