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	1.	Concise and efficient synthesis of 4-fluoro-1H-pyrrolo[2,3-b]pyridine. [electronic resource] by Thibault, Carl L'Heureux, Alexandre Bhide, Rajeev S Ruel, Réjean Producer: 20041026 In: Organic letters vol. 5 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	2.	Preclinical pharmacokinetics and in vitro metabolism of brivanib (BMS-540215), a potent VEGFR2 inhibitor and its alanine ester prodrug brivanib alaninate. [electronic resource] by Marathe, Punit H Kamath, Amrita V Zhang, Yueping D'Arienzo, Celia Bhide, Rajeev Fargnoli, Joseph Producer: 20091013 In: Cancer chemotherapy and pharmacology vol. 65 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	3.	Identification of highly potent and selective PI3Kδ inhibitors. [electronic resource] by Marcoux, David Qin, Lan-Ying Ruan, Zheming Shi, Qing Ruan, Qian Weigelt, Carolyn Qiu, Hongchen Schieven, Gary Hynes, John Bhide, Rajeev Poss, Michael Tino, Joseph Producer: 20170818 In: Bioorganic & medicinal chemistry letters vol. 27 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	4.	Metabolism of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)-N-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine (BMS-645737): identification of an unusual N-acetylglucosamine conjugate in the cynomolgus monkey. [electronic resource] by Johnson, Benjamin M Kamath, Amrita V Leet, John E Liu, Xiaohong Bhide, Rajeev S Tejwani, Ravindra W Zhang, Yueping Qian, Ligang Wei, Donna D Lombardo, Louis J Shu, Yue-Zhong Producer: 20090605 In: Drug metabolism and disposition: the biological fate of chemicals vol. 36 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	5.	Discovery and structure-based design of 4,6-diaminonicotinamides as potent and selective IRAK4 inhibitors. [electronic resource] by Bhide, Rajeev S Keon, Alec Weigelt, Carolyn Sack, John S Schmidt, Robert J Lin, Shuqun Xiao, Hai-Yun Spergel, Steven H Kempson, James Pitts, William J Carman, Julie Poss, Michael A Producer: 20171206 In: Bioorganic & medicinal chemistry letters vol. 27 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	6.	Discovery of the pyrrolo[2,1-f][1,2,4]triazine nucleus as a new kinase inhibitor template. [electronic resource] by Hunt, John T Mitt, Toomas Borzilleri, Robert Gullo-Brown, Johnni Fargnoli, Joseph Fink, Brian Han, Wen-Ching Mortillo, Steven Vite, Gregory Wautlet, Barri Wong, Tai Yu, Chiang Zheng, Xiaoping Bhide, Rajeev Producer: 20040824 In: Journal of medicinal chemistry vol. 47 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	7.	Synthesis, SAR, and Evaluation of 4-[2,4-Difluoro-5-(cyclopropylcarbamoyl)phenylamino]pyrrolo[2,1-f][1,2,4]triazine-based VEGFR-2 kinase inhibitors. [electronic resource] by Cai, Zhen-Wei Wei, Donna Borzilleri, Robert M Qian, Ligang Kamath, Amrita Mortillo, Steven Wautlet, Barri Henley, Benjamin J Jeyaseelan, Robert Tokarski, John Hunt, John T Bhide, Rajeev S Fargnoli, Joseph Lombardo, Louis J Producer: 20080512 In: Bioorganic & medicinal chemistry letters vol. 18 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	8.	Synthesis and SAR of 4-(3-hydroxyphenylamino)pyrrolo[2,1-f][1,2,4]triazine based VEGFR-2 kinase inhibitors. [electronic resource] by Borzilleri, Robert M Cai, Zhen-Wei Ellis, Christopher Fargnoli, Joseph Fura, Aberra Gerhardt, Tracy Goyal, Bindu Hunt, John T Mortillo, Steven Qian, Ligang Tokarski, John Vyas, Viral Wautlet, Barri Zheng, Xioping Bhide, Rajeev S Producer: 20050705 In: Bioorganic & medicinal chemistry letters vol. 15 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	9.	Design, synthesis, functional and structural characterization of an inhibitor of N-acetylneuraminate-9-phosphate phosphatase: observation of extensive dynamics in an enzyme/inhibitor complex. [electronic resource] by Kim, Soong-Hoon Constantine, Keith L Duke, Gerald J Goldfarb, Valentina Hunt, John T Johnson, Stephen Kish, Kevin Klei, Herbert E McDonnell, Patricia A Metzler, William J Mueller, Luciano Poss, Michael A Fairchild, Craig R Bhide, Rajeev S Producer: 20140121 In: Bioorganic & medicinal chemistry letters vol. 23 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	10.	The antiangiogenic activity in xenograft models of brivanib, a dual inhibitor of vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 kinases. [electronic resource] by Bhide, Rajeev S Lombardo, Louis J Hunt, John T Cai, Zhen-Wei Barrish, Joel C Galbraith, Susan Jeyaseelan, Robert Mortillo, Steven Wautlet, Barri S Krishnan, Bala Kukral, Daniel Malone, Harold Lewin, Anne C Henley, Benjamin J Fargnoli, Joseph Producer: 20101110 In: Molecular cancer therapeutics vol. 9 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	11.	Discovery and evaluation of N-cyclopropyl- 2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a selective and orally efficacious inhibitor of vascular endothelial growth factor receptor-2. [electronic resource] by Borzilleri, Robert M Bhide, Rajeev S Barrish, Joel C D'Arienzo, Celia J Derbin, George M Fargnoli, Joseph Hunt, John T Jeyaseelan, Robert Kamath, Amrita Kukral, Daniel W Marathe, Punit Mortillo, Steve Qian, Ligang Tokarski, John S Wautlet, Barri S Zheng, Xiaoping Lombardo, Louis J Producer: 20060816 In: Journal of medicinal chemistry vol. 49 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	12.	Design, synthesis, and evaluation of orally active 4-(2,4-difluoro-5-(methoxycarbamoyl)phenylamino)pyrrolo[2,1-f][1,2,4]triazines as dual vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 inhibitors. [electronic resource] by Borzilleri, Robert M Zheng, Xiaoping Qian, Ligang Ellis, Christopher Cai, Zhen-wei Wautlet, Barri S Mortillo, Steve Jeyaseelan, Robert Kukral, Daniel W Fura, Aberra Kamath, Amrita Vyas, Viral Tokarski, John S Barrish, Joel C Hunt, John T Lombardo, Louis J Fargnoli, Joseph Bhide, Rajeev S Producer: 20050706 In: Journal of medicinal chemistry vol. 48 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	13.	Design, synthesis, and structure-activity relationships of tetrahydroquinoline-based farnesyltransferase inhibitors. [electronic resource] by Lombardo, Louis J Camuso, Amy Clark, John Fager, Krista Gullo-Brown, Johnni Hunt, John T Inigo, Ivan Kan, David Koplowitz, Barry Lee, Francis McGlinchey, Kelly Qian, Ligang Ricca, Carolyn Rovnyak, George Traeger, Sarah Tokarski, John Williams, David K Wu, Laurence I Zhao, Yufen Manne, Veeraswamy Bhide, Rajeev S Producer: 20050805 In: Bioorganic & medicinal chemistry letters vol. 15 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	14.	Discovery and SAR of pyrrolo[2,1-f][1,2,4]triazin-4-amines as potent and selective PI3Kδ inhibitors. [electronic resource] by Bhide, Rajeev S Neels, James Qin, Lan-Ying Ruan, Zheming Stachura, Sylwia Weigelt, Carolyn Sack, John S Stefanski, Kevin Gu, Xiaomei Xie, Jenny H Goldstine, Christine B Skala, Stacey Pedicord, Donna L Ruepp, Stefan Dhar, T G Murali Carter, Percy H Salter-Cid, Luisa M Poss, Michael A Davies, Paul Producer: 20170726 In: Bioorganic & medicinal chemistry letters vol. 26 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	15.	Discovery and preclinical studies of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)-N-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine (BMS-645737), an in vivo active potent VEGFR-2 inhibitor. [electronic resource] by Ruel, Réjean Thibeault, Carl L'Heureux, Alexandre Martel, Alain Cai, Zhen-Wei Wei, Donna Qian, Ligang Barrish, Joel C Mathur, Arvind D'Arienzo, Celia Hunt, John T Kamath, Amrita Marathe, Punit Zhang, Yueping Derbin, George Wautlet, Barri Mortillo, Steven Jeyaseelan, Robert Henley, Benjamin Tejwani, Ravindra Bhide, Rajeev S Trainor, George L Fargnoli, Joseph Lombardo, Louis J Producer: 20080715 In: Bioorganic & medicinal chemistry letters vol. 18 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	16.	Discovery of brivanib alaninate ((S)-((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), a novel prodrug of dual vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 kinase inhibitor (BMS-540215). [electronic resource] by Cai, Zhen-wei Zhang, Yongzheng Borzilleri, Robert M Qian, Ligang Barbosa, Stephanie Wei, Donna Zheng, Xiaoping Wu, Lawrence Fan, Junying Shi, Zhongping Wautlet, Barri S Mortillo, Steve Jeyaseelan, Robert Kukral, Daniel W Kamath, Amrita Marathe, Punit D'Arienzo, Celia Derbin, George Barrish, Joel C Robl, Jeffrey A Hunt, John T Lombardo, Louis J Fargnoli, Joseph Bhide, Rajeev S Producer: 20080611 In: Journal of medicinal chemistry vol. 51 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	17.	Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors. [electronic resource] by Qin, Lan-Ying Ruan, Zheming Cherney, Robert J Dhar, T G Murali Neels, James Weigelt, Carolyn A Sack, John S Srivastava, Anurag S Cornelius, Lyndon A M Tino, Joseph A Stefanski, Kevin Gu, Xiaomei Xie, Jenny Susulic, Vojkan Yang, Xiaoxia Yarde-Chinn, Melissa Skala, Stacey Bosnius, Ruth Goldstein, Christine Davies, Paul Ruepp, Stefan Salter-Cid, Luisa Bhide, Rajeev S Poss, Michael A Producer: 20170704 In: Bioorganic & medicinal chemistry letters vol. 27 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	18.	Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an in vivo active potent VEGFR-2 inhibitor. [electronic resource] by Bhide, Rajeev S Cai, Zhen-Wei Zhang, Yong-Zheng Qian, Ligang Wei, Donna Barbosa, Stephanie Lombardo, Louis J Borzilleri, Robert M Zheng, Xiaoping Wu, Laurence I Barrish, Joel C Kim, Soong-Hoon Leavitt, Kenneth Mathur, Arvind Leith, Leslie Chao, Sam Wautlet, Barri Mortillo, Steven Jeyaseelan, Robert Kukral, Daniel Hunt, John T Kamath, Amrita Fura, Aberra Vyas, Viral Marathe, Punit D'Arienzo, Celia Derbin, George Fargnoli, Joseph Producer: 20060502 In: Journal of medicinal chemistry vol. 49 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	19.	Synthesis and SAR of pyrrolotriazine-4-one based Eg5 inhibitors. [electronic resource] by Kim, Kyoung Soon Lu, Songfeng Cornelius, Lyndon A Lombardo, Louis J Borzilleri, Robert M Schroeder, Gretchen M Sheng, Christopher Rovnyak, George Crews, Donald Schmidt, Robert J Williams, David K Bhide, Rajeev S Traeger, Sarah C McDonnell, Patricia A Mueller, Luciano Sheriff, Steven Newitt, John A Pudzianowski, Andrew T Yang, Zheng Wild, Robert Lee, Frances Y Batorsky, Roberta Ryder, James S Ortega-Nanos, Marie Shen, Henry Gottardis, Marco Roussell, Deborah L Producer: 20060911 In: Bioorganic & medicinal chemistry letters vol. 16 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	20.	Identification of a Potent, Selective, and Efficacious Phosphatidylinositol 3-Kinase δ (PI3Kδ) Inhibitor for the Treatment of Immunological Disorders. [electronic resource] by Liu, Qingjie Shi, Qing Marcoux, David Batt, Douglas G Cornelius, Lyndon Qin, Lan-Ying Ruan, Zheming Neels, James Beaudoin-Bertrand, Myra Srivastava, Anurag S Li, Ling Cherney, Robert J Gong, Hua Watterson, Scott H Weigelt, Carolyn Gillooly, Kathleen M McIntyre, Kim W Xie, Jenny H Obermeier, Mary T Fura, Aberra Sleczka, Bogdan Stefanski, Kevin Fancher, R M Padmanabhan, Shweta Rp, Thatipamula Kundu, Ipsit Rajareddy, Kallem Smith, Rodney Hennan, James K Xing, Dezhi Fan, Jingsong Levesque, Paul C Ruan, Qian Pitt, Sidney Zhang, Rosemary Pedicord, Donna Pan, Jie Yarde, Melissa Lu, Hao Lippy, Jonathan Goldstine, Christine Skala, Stacey Rampulla, Richard A Mathur, Arvind Gupta, Anuradha Arunachalam, Pirama Nayagam Sack, John S Muckelbauer, Jodi K Cvijic, Mary Ellen Salter-Cid, Luisa M Bhide, Rajeev S Poss, Michael A Hynes, John Carter, Percy H Macor, John E Ruepp, Stefan Schieven, Gary L Tino, Joseph A Producer: 20170811 In: Journal of medicinal chemistry vol. 60 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)

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