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MAP4K4 Is a Threonine Kinase That Phosphorylates FARP1. [electronic resource] by
- Schwaid, Adam G
- Su, Chunyan
- Loos, Paula
- Wu, Jiang
- Nguyen, Chuong
- Stone, Kathryn L
- Kanyo, Jean
- Geoghegan, Kieran F
- Bhattacharya, Samit K
- Dow, Robert L
- Buckbinder, Leonard
- Carpino, Philip A
Producer: 20161005
In:
ACS chemical biology vol. 10
Availability: No items available.
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9.
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Achieving selectivity between highly homologous tyrosine kinases: a novel selective erbB2 inhibitor. [electronic resource] by
- Bhattacharya, Samit K
- Cox, Eric D
- Kath, John C
- Mathiowetz, Alan M
- Morris, Joel
- Moyer, James D
- Pustilnik, Leslie R
- Rafidi, Kris
- Richter, Daniel T
- Su, Chunyan
- Wessel, Matthew D
Producer: 20030916
In:
Biochemical and biophysical research communications vol. 307
Availability: No items available.
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10.
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The discovery of highly selective erbB2 (Her2) inhibitors for the treatment of cancer. [electronic resource] by
- Lippa, Blaise
- Kauffman, Goss S
- Arcari, Joel
- Kwan, Tricia
- Chen, Jinshan
- Hungerford, William
- Bhattacharya, Samit
- Zhao, Xumiao
- Williams, Courtney
- Xiao, Jun
- Pustilnik, Leslie
- Su, Chunyan
- Moyer, James D
- Ma, Ling
- Campbell, Mary
- Steyn, Stefanus
Producer: 20070807
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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11.
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2-Aminopyridine-Based Mitogen-Activated Protein Kinase Kinase Kinase Kinase 4 (MAP4K4) Inhibitors: Assessment of Mechanism-Based Safety. [electronic resource] by
- Dow, Robert L
- Ammirati, Mark
- Bagley, Scott W
- Bhattacharya, Samit K
- Buckbinder, Leonard
- Cortes, Christian
- El-Kattan, Ayman F
- Ford, Kristen
- Freeman, Gary B
- Guimarães, Cristiano R W
- Liu, Shenping
- Niosi, Mark
- Skoura, Athanasia
- Tess, David
Producer: 20190417
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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12.
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Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). [electronic resource] by
- Filipski, Kevin J
- Sammons, Matthew F
- Bhattacharya, Samit K
- Panteleev, Jane
- Brown, Janice A
- Loria, Paula M
- Boehm, Markus
- Smith, Aaron C
- Shavnya, Andre
- Conn, Edward L
- Song, Kun
- Weng, Yan
- Facemire, Carie
- Jüppner, Harald
- Clerin, Valerie
Publication details: ACS medicinal chemistry letters May 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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13.
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Endothelial protein kinase MAP4K4 promotes vascular inflammation and atherosclerosis. [electronic resource] by
- Roth Flach, Rachel J
- Skoura, Athanasia
- Matevossian, Anouch
- Danai, Laura V
- Zheng, Wei
- Cortes, Christian
- Bhattacharya, Samit K
- Aouadi, Myriam
- Hagan, Nana
- Yawe, Joseph C
- Vangala, Pranitha
- Menendez, Lorena Garcia
- Cooper, Marcus P
- Fitzgibbons, Timothy P
- Buckbinder, Leonard
- Czech, Michael P
Producer: 20160517
In:
Nature communications vol. 6
Availability: No items available.
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14.
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Discovery and pharmacologic characterization of CP-724,714, a selective ErbB2 tyrosine kinase inhibitor. [electronic resource] by
- Jani, Jitesh P
- Finn, Richard S
- Campbell, Mary
- Coleman, Kevin G
- Connell, Richard D
- Currier, Nicolas
- Emerson, Erling O
- Floyd, Eugenia
- Harriman, Shawn
- Kath, John C
- Morris, Joel
- Moyer, James D
- Pustilnik, Leslie R
- Rafidi, Kristina
- Ralston, Sherry
- Rossi, Ann Marie K
- Steyn, Stefanus J
- Wagner, Larry
- Winter, Steven M
- Bhattacharya, Samit K
Producer: 20071212
In:
Cancer research vol. 67
Availability: No items available.
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15.
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The discovery of novel calcium sensing receptor negative allosteric modulators. [electronic resource] by
- Balan, Gayatri
- Bauman, Jonathan
- Bhattacharya, Samit
- Castrodad, Mayda
- Healy, David R
- Herr, Michael
- Humphries, Paul
- Jennings, Sandra
- Kalgutkar, Amit S
- Kapinos, Brendon
- Khot, Vishal
- Lazarra, Kimberly
- Li, Mei
- Li, Yan
- Neagu, Constantin
- Oliver, Robert
- Piotrowski, David W
- Price, David
- Qi, Hong
- Simmons, Holly A
- Southers, James
- Wei, Liuqing
- Zhang, Yan
- Paralkar, Vishwas M
Producer: 20090821
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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16.
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Evaluation and synthesis of polar aryl- and heteroaryl spiroazetidine-piperidine acetamides as ghrelin inverse agonists. [electronic resource] by
- Orr, Suvi T M
- Beveridge, Ramsay
- Bhattacharya, Samit K
- Cameron, Kimberly O
- Coffey, Steven
- Fernando, Dilinie
- Hepworth, David
- Jackson, Margaret V
- Khot, Vishal
- Kosa, Rachel
- Lapham, Kimberly
- Loria, Paula M
- McClure, Kim F
- Patel, Jigna
- Rose, Colin
- Saenz, James
- Stock, Ingrid A
- Storer, Gregory
- von Volkenburg, Maria
- Vrieze, Derek
- Wang, Guoqiang
- Xiao, Jun
- Zhang, Yingxin
Producer: 20150220
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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17.
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PF-03814735, an orally bioavailable small molecule aurora kinase inhibitor for cancer therapy. [electronic resource] by
- Jani, Jitesh P
- Arcari, Joel
- Bernardo, Vincent
- Bhattacharya, Samit K
- Briere, David
- Cohen, Bruce D
- Coleman, Kevin
- Christensen, James G
- Emerson, Erling O
- Jakowski, Amy
- Hook, Kenneth
- Los, Gerrit
- Moyer, James D
- Pruimboom-Brees, Ingrid
- Pustilnik, Leslie
- Rossi, Ann Marie
- Steyn, Stefan J
- Su, Chunyan
- Tsaparikos, Konstantinos
- Wishka, Donn
- Yoon, Kwansik
- Jakubczak, John L
Producer: 20100707
In:
Molecular cancer therapeutics vol. 9
Availability: No items available.
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18.
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Design and synthesis of truncated EGF-A peptides that restore LDL-R recycling in the presence of PCSK9 in vitro. [electronic resource] by
- Schroeder, Christina I
- Swedberg, Joakim E
- Withka, Jane M
- Rosengren, K Johan
- Akcan, Muharrem
- Clayton, Daniel J
- Daly, Norelle L
- Cheneval, Olivier
- Borzilleri, Kris A
- Griffor, Matt
- Stock, Ingrid
- Colless, Barbara
- Walsh, Phillip
- Sunderland, Philip
- Reyes, Allan
- Dullea, Robert
- Ammirati, Mark
- Liu, Shenping
- McClure, Kim F
- Tu, Meihua
- Bhattacharya, Samit K
- Liras, Spiros
- Price, David A
- Craik, David J
Producer: 20141016
In:
Chemistry & biology vol. 21
Availability: No items available.
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19.
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Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate. [electronic resource] by
- Bhattacharya, Samit K
- Andrews, Kim
- Beveridge, Ramsay
- Cameron, Kimberly O
- Chen, Chiliu
- Dunn, Matthew
- Fernando, Dilinie
- Gao, Hua
- Hepworth, David
- Jackson, V Margaret
- Khot, Vishal
- Kong, Jimmy
- Kosa, Rachel E
- Lapham, Kimberly
- Loria, Paula M
- Londregan, Allyn T
- McClure, Kim F
- Orr, Suvi T M
- Patel, Jigna
- Rose, Colin
- Saenz, James
- Stock, Ingrid A
- Storer, Gregory
- VanVolkenburg, Maria
- Vrieze, Derek
- Wang, Guoqiang
- Xiao, Jun
- Zhang, Yingxin
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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20.
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Discovery of an in Vivo Tool to Establish Proof-of-Concept for MAP4K4-Based Antidiabetic Treatment. [electronic resource] by
- Ammirati, Mark
- Bagley, Scott W
- Bhattacharya, Samit K
- Buckbinder, Leonard
- Carlo, Anthony A
- Conrad, Rebecca
- Cortes, Christian
- Dow, Robert L
- Dowling, Matthew S
- El-Kattan, Ayman
- Ford, Kristen
- Guimarães, Cristiano R W
- Hepworth, David
- Jiao, Wenhua
- LaPerle, Jennifer
- Liu, Shenping
- Londregan, Allyn
- Loria, Paula M
- Mathiowetz, Alan M
- Munchhof, Michael
- Orr, Suvi T M
- Petersen, Donna N
- Price, David A
- Skoura, Athanasia
- Smith, Aaron C
- Wang, Jian
Producer: 20151130
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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