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	1.	Fragment-based approaches to the discovery of kinase inhibitors. [electronic resource] by Mortenson, Paul N Berdini, Valerio O'Reilly, Marc Producer: 20150707 In: Methods in enzymology vol. 548 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	2.	Crystal structure of Schistosoma purine nucleoside phosphorylase complexed with a novel monocyclic inhibitor. [electronic resource] by Pereira, Humberto M Berdini, Valério Ferri, Mariana R Cleasby, Anne Garratt, Richard C Producer: 20100525 In: Acta tropica vol. 114 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	3.	Virtual screening using protein-ligand docking: avoiding artificial enrichment. [electronic resource] by Verdonk, Marcel L Berdini, Valerio Hartshorn, Michael J Mooij, Wijnand T M Murray, Christopher W Taylor, Richard D Watson, Paul Producer: 20050321 In: Journal of chemical information and computer sciences vol. 44 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	4.	Carbocysteine lysine salt monohydrate (SCMC-LYS) is a selective scavenger of reactive oxygen intermediates (ROIs). [electronic resource] by Brandolini, Laura Allegretti, Marcello Berdini, Valerio Cervellera, Maria Neve Mascagni, Patrizia Rinaldi, Matteo Melillo, Gabriella Ghezzi, Pietro Mengozzi, Manuela Bertini, Riccardo Producer: 20040122 In: European cytokine network vol. 14 Availability: No items available. Save to lists Add to cart (remove)
	5.	Perspective on computational and structural aspects of kinase discovery from IPK2014. [electronic resource] by Martin, Eric Knapp, Stefan Engh, Richard A Moebitz, Henrik Varin, Thibault Roux, Benoit Meiler, Jens Berdini, Valerio Baumann, Alexander Vieth, Michal Producer: 20151209 In: Biochimica et biophysica acta vol. 1854 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	6.	Rapid evolution of 6-phenylpurine inhibitors of protein kinase B through structure-based design. [electronic resource] by Donald, Alastair McHardy, Tatiana Rowlands, Martin G Hunter, Lisa-Jane K Davies, Thomas G Berdini, Valerio Boyle, Robert G Aherne, G Wynne Garrett, Michelle D Collins, Ian Producer: 20070706 In: Journal of medicinal chemistry vol. 50 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	7.	Identification of inhibitors of protein kinase B using fragment-based lead discovery. [electronic resource] by Saxty, Gordon Woodhead, Steven J Berdini, Valerio Davies, Thomas G Verdonk, Marcel L Wyatt, Paul G Boyle, Robert G Barford, David Downham, Robert Garrett, Michelle D Carr, Robin A Producer: 20070706 In: Journal of medicinal chemistry vol. 50 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	8.	Crystal structure of human soluble adenylate cyclase reveals a distinct, highly flexible allosteric bicarbonate binding pocket. [electronic resource] by Saalau-Bethell, Susanne M Berdini, Valerio Cleasby, Anne Congreve, Miles Coyle, Joseph E Lock, Victoria Murray, Christopher W O'Brien, M Alistair Rich, Sharna J Sambrook, Tracey Vinkovic, Mladen Yon, Jeff R Jhoti, Harren Producer: 20141215 In: ChemMedChem vol. 9 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	9.	2-Arylpropionic CXC chemokine receptor 1 (CXCR1) ligands as novel noncompetitive CXCL8 inhibitors. [electronic resource] by Allegretti, Marcello Bertini, Riccardo Cesta, Maria Candida Bizzarri, Cinzia Di Bitondo, Rosa Di Cioccio, Vito Galliera, Emanuela Berdini, Valerio Topai, Alessandra Zampella, Giuseppe Russo, Vincenzo Di Bello, Nicoletta Nano, Giuseppe Nicolini, Luca Locati, Massimo Fantucci, Piercarlo Florio, Saverio Colotta, Francesco Producer: 20050823 In: Journal of medicinal chemistry vol. 48 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	10.	Structure-based design of isoquinoline-5-sulfonamide inhibitors of protein kinase B. [electronic resource] by Collins, Ian Caldwell, John Fonseca, Tatiana Donald, Alastair Bavetsias, Vassilios Hunter, Lisa-Jane K Garrett, Michelle D Rowlands, Martin G Aherne, G Wynne Davies, Thomas G Berdini, Valerio Woodhead, Steven J Davis, Deborah Seavers, Lisa C A Wyatt, Paul G Workman, Paul McDonald, Edward Producer: 20060317 In: Bioorganic & medicinal chemistry vol. 14 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	11.	Fragment-based discovery of type I inhibitors of maternal embryonic leucine zipper kinase. [electronic resource] by Johnson, Christopher N Berdini, Valerio Beke, Lijs Bonnet, Pascal Brehmer, Dirk Coyle, Joseph E Day, Phillip J Frederickson, Martyn Freyne, Eddy J E Gilissen, Ron A H J Hamlett, Christopher C F Howard, Steven Meerpoel, Lieven McMenamin, Rachel Patel, Sahil Rees, David C Sharff, Andrew Sommen, François Wu, Tongfei Linders, Joannes T M Producer: 20150115 In: ACS medicinal chemistry letters vol. 6 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	12.	Structure-Based Design of Type II Inhibitors Applied to Maternal Embryonic Leucine Zipper Kinase. [electronic resource] by Johnson, Christopher N Adelinet, Christophe Berdini, Valerio Beke, Lijs Bonnet, Pascal Brehmer, Dirk Calo, Frederick Coyle, Joseph E Day, Phillip J Frederickson, Martyn Freyne, Eddy J E Gilissen, Ron A H J Hamlett, Christopher C F Howard, Steven Meerpoel, Lieven Mevellec, Laurence McMenamin, Rachel Pasquier, Elisabeth Patel, Sahil Rees, David C Linders, Joannes T M Producer: 20150115 In: ACS medicinal chemistry letters vol. 6 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	13.	Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors. [electronic resource] by Murray, Christopher W Berdini, Valerio Buck, Ildiko M Carr, Maria E Cleasby, Anne Coyle, Joseph E Curry, Jayne E Day, James E H Day, Phillip J Hearn, Keisha Iqbal, Aman Lee, Lydia Y W Martins, Vanessa Mortenson, Paul N Munck, Joanne M Page, Lee W Patel, Sahil Roomans, Susan Smith, Kirsten Tamanini, Emiliano Saxty, Gordon Producer: 20150720 In: ACS medicinal chemistry letters vol. 6 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	14.	Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA [electronic resource] by Woolford, Alison J-A Day, Philip J Bénéton, Véronique Berdini, Valerio Coyle, Joseph E Dudit, Yann Grondin, Pascal Huet, Pascal Lee, Lydia Y W Manas, Eric S McMenamin, Rachel L Murray, Christopher W Page, Lee W Patel, Vipulkumar K Potvain, Florent Rich, Sharna J Sang, Yingxia Somers, Don O Trottet, Lionel Wan, Zehong Zhang, Xiaomin Producer: 20170615 In: Journal of medicinal chemistry vol. 59 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	15.	Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives. [electronic resource] by Tisi, Dominic Chiarparin, Elisabetta Tamanini, Emiliano Pathuri, Puja Coyle, Joseph E Hold, Adam Holding, Finn P Amin, Nader Martin, Agnes C L Rich, Sharna J Berdini, Valerio Yon, Jeff Acklam, Paul Burke, Rosemary Drouin, Ludovic Harmer, Jenny E Jeganathan, Fiona van Montfort, Rob L M Newbatt, Yvette Tortorici, Marcello Westlake, Maura Wood, Amy Hoelder, Swen Heightman, Tom D Producer: 20170622 In: ACS chemical biology vol. 11 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	16.	Fragment-based discovery of the pyrazol-4-yl urea (AT9283), a multitargeted kinase inhibitor with potent aurora kinase activity. [electronic resource] by Howard, Steven Berdini, Valerio Boulstridge, John A Carr, Maria G Cross, David M Curry, Jayne Devine, Lindsay A Early, Theresa R Fazal, Lynsey Gill, Adrian L Heathcote, Michelle Maman, Sarita Matthews, Julia E McMenamin, Rachel L Navarro, Eva F O'Brien, Michael A O'Reilly, Marc Rees, David C Reule, Matthias Tisi, Dominic Williams, Glyn Vinković, Mladen Wyatt, Paul G Producer: 20090223 In: Journal of medicinal chemistry vol. 52 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	17.	Identification of N-(4-piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide (AT7519), a novel cyclin dependent kinase inhibitor using fragment-based X-ray crystallography and structure based drug design. [electronic resource] by Wyatt, Paul G Woodhead, Andrew J Berdini, Valerio Boulstridge, John A Carr, Maria G Cross, David M Davis, Deborah J Devine, Lindsay A Early, Theresa R Feltell, Ruth E Lewis, E Jonathan McMenamin, Rachel L Navarro, Eva F O'Brien, Michael A O'Reilly, Marc Reule, Matthias Saxty, Gordon Seavers, Lisa C A Smith, Donna-Michelle Squires, Matt S Trewartha, Gary Walker, Margaret T Woolford, Alison J-A Producer: 20080910 In: Journal of medicinal chemistry vol. 51 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	18.	Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening. [electronic resource] by Woolford, Alison J-A Pero, Joseph E Aravapalli, Sridhar Berdini, Valerio Coyle, Joseph E Day, Philip J Dodson, Andrew M Grondin, Pascal Holding, Finn P Lee, Lydia Y W Li, Peng Manas, Eric S Marino, Joseph Martin, Agnes C L McCleland, Brent W McMenamin, Rachel L Murray, Christopher W Neipp, Christopher E Page, Lee W Patel, Vipulkumar K Potvain, Florent Rich, Sharna Rivero, Ralph A Smith, Kirsten Somers, Donald O Trottet, Lionel Velagaleti, Ranganadh Williams, Glyn Xie, Ren Producer: 20170606 In: Journal of medicinal chemistry vol. 59 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	19.	Potent, selective inhibitors of fibroblast growth factor receptor define fibroblast growth factor dependence in preclinical cancer models. [electronic resource] by Squires, Matthew Ward, George Saxty, Gordan Berdini, Valerio Cleasby, Anne King, Peter Angibaud, Patrick Perera, Tim Fazal, Lynsey Ross, Douglas Jones, Charlotte Griffiths Madin, Andrew Benning, Rajdeep K Vickerstaffe, Emma O'Brien, Alistair Frederickson, Martyn Reader, Michael Hamlett, Christopher Batey, Michael A Rich, Sharna Carr, Maria Miller, Darcey Feltell, Ruth Thiru, Abarna Bethell, Susanne Devine, Lindsay A Graham, Brent L Pike, Andrew Cosme, Jose Lewis, Edward J Freyne, Eddy Lyons, John Irving, Julie Murray, Christopher Newell, David R Thompson, Neil T Producer: 20120123 In: Molecular cancer therapeutics vol. 10 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	20.	Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. [electronic resource] by Heightman, Tom D Berdini, Valerio Braithwaite, Hannah Buck, Ildiko M Cassidy, Megan Castro, Juan Courtin, Aurélie Day, James E H East, Charlotte Fazal, Lynsey Graham, Brent Griffiths-Jones, Charlotte M Lyons, John F Martins, Vanessa Muench, Sandra Munck, Joanne M Norton, David O'Reilly, Marc Palmer, Nick Pathuri, Puja Reader, Michael Rees, David C Rich, Sharna J Richardson, Caroline Saini, Harpreet Thompson, Neil T Wallis, Nicola G Walton, Hugh Wilsher, Nicola E Woolford, Alison J-A Cooke, Michael Cousin, David Onions, Stuart Shannon, Jonathan Watts, John Murray, Christopher W Producer: 20190520 In: Journal of medicinal chemistry vol. 61 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)

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